Patent classifications
C07C235/52
Use of picolinamide compounds as fungicides
This disclosure relates to picolinamides of Formula I and their use as fungicides. ##STR00001##
Amide derivatives as lysophosphatidic acid receptor antagonists
The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, formula (I) wherein R.sup.1, X, m, R.sup.2, Y, R.sup.3, Z, n, R.sup.4, A and B are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.
##STR00001##
Amide derivatives as lysophosphatidic acid receptor antagonists
The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, formula (I) wherein R.sup.1, X, m, R.sup.2, Y, R.sup.3, Z, n, R.sup.4, A and B are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.
##STR00001##
NOVEL PHENOLIC ACID DERIVATIVE COMPOUND AND USE THEREOF
The present invention relates to a novel phenolic acid derivative compound with whitening and antioxidant activities and use thereof. The phenolic acid derivative compound is a compound represented by Formula 1, which is described in the specification, an isomer thereof or a salt thereof. The compound of the present invention has skin whitening activity to inhibit tyrosinase, thus being suitable for use in a pharmaceutical composition or cosmetic product for skin whitening. In addition, the compound of the present invention is suitable for the prevention or treatment of oxidation-derived skin abnormality or disease such as skin aging due to its antioxidant activity.
FATTY ACID ACETYLATED SALICYLATES AND THEIR USES
The invention relates to Fatty Acid Acetylated Salicylate Derivatives; compositions comprising an effective amount of a Fatty Acid Acetylated Salicylate Derivative; and methods for treating or preventing an inflammatory disorder comprising the administration of an effective amount of a Fatty Acid Acetylated Salicylate Derivative.
FATTY ACID ACETYLATED SALICYLATES AND THEIR USES
The invention relates to Fatty Acid Acetylated Salicylate Derivatives; compositions comprising an effective amount of a Fatty Acid Acetylated Salicylate Derivative; and methods for treating or preventing an inflammatory disorder comprising the administration of an effective amount of a Fatty Acid Acetylated Salicylate Derivative.
Therapeutic compounds and methods of use thereof
The invention provides compounds having the general Formula (I); ##STR00001##
and pharmaceutically acceptable salts thereof; wherein the variables R.sup.A, R.sup.AA, subscript n, subscript q, ring A, X.sup.2, L, subscript m, X.sup.1, R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, D and E have the meaning as described herein, and compositions containing such compounds and methods for using such compounds and compositions.
Amide derivatives as lysophosphatidic acid receptor antagonists
The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, ##STR00001##
wherein R.sup.1, X, m, R.sup.2, Y, R.sup.3, Z, n, R.sup.4, A and B are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.
Amide derivatives as lysophosphatidic acid receptor antagonists
The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, ##STR00001##
wherein R.sup.1, X, m, R.sup.2, Y, R.sup.3, Z, n, R.sup.4, A and B are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.
PHENYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS
The invention relates to a compound of formula (I)
##STR00001##
wherein R.sup.1 to R.sup.3 are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.