C07D231/16

ADSORPTION OF FLUORINATED ANESTHETICS WITHIN THE PORES OF MOLECULAR CRYSTALS

A method of delivering or sequestering anesthetic agents by adsorption of such agents by porous partially fluorinated compounds which display high weight adsorption capacities.

SUBSTITUTED PYRAZOLYLPYRAZOLE DERIVATIVE AND USE OF SAME AS HERBICIDE
20170367341 · 2017-12-28 · ·

Provided is a compound capable of effectively control worst weeds of higher leaf stages that present practical problems. A specific pyrazolylpyrazole derivative of formula (I) is disclosed that is able to solve the above-mentioned problems.

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Process for the preparation of 5-fluoro-1H-pyrazoles

A new process for the preparation of 5-fluoro-1H-pyrazoles of the general formula (I) as described herein comprising reacting an olefin with an hydrazine.

Process for the preparation of 5-fluoro-1H-pyrazoles

A new process for the preparation of 5-fluoro-1H-pyrazoles of the general formula (I) as described herein comprising reacting an olefin with an hydrazine.

Tetrazolinone compounds and their use as pesticides

The present invention provides a compound having an excellent efficacy for controlling pests. A tetrazolinone compound of a formula (1) [wherein Q represents a group selected from the following group: Q1, Q2, Q3 or Q4: R.sup.1, R.sup.2, R.sup.3 and R.sup.11 represent independently of each other a halogen atom, an CI-C6 alkyl group, etc.; R.sup.4 and R.sup.5 represent independently of each other a hydrogen atom, a halogen atom or an C1-C3 alkyl group, etc.; R.sup.6 represents a halogen atom, an C1-C4 alkyl group, etc.; R.sup.7, R.sup.8 and R.sup.9 represent independently of each other a hydrogen atom, a halogen atom, etc.; and R.sup.10 represents an C1-C3 alkyl group, etc.] shows an excellent controlling efficacy on pests. ##STR00001##

Tetrazolinone compounds and their use as pesticides

The present invention provides a compound having an excellent efficacy for controlling pests. A tetrazolinone compound of a formula (1) [wherein Q represents a group selected from the following group: Q1, Q2, Q3 or Q4: R.sup.1, R.sup.2, R.sup.3 and R.sup.11 represent independently of each other a halogen atom, an CI-C6 alkyl group, etc.; R.sup.4 and R.sup.5 represent independently of each other a hydrogen atom, a halogen atom or an C1-C3 alkyl group, etc.; R.sup.6 represents a halogen atom, an C1-C4 alkyl group, etc.; R.sup.7, R.sup.8 and R.sup.9 represent independently of each other a hydrogen atom, a halogen atom, etc.; and R.sup.10 represents an C1-C3 alkyl group, etc.] shows an excellent controlling efficacy on pests. ##STR00001##

IMIDAZOLE 3-OXIDE DERIVATIVE BASED ACSS2 INHIBITORS AND METHODS OF USE THEREOF

The present invention relates to novel ACSS2 inhibitors having activity as anti-cancer therapy, treatment of alcoholism, and viral infection (e.g., CMV), composition and methods of preparation thereof, and uses thereof for treating viral infection, alcoholism, alcoholic steatohepatitis (ASH), non-alcoholic steatohepatitis (NASH), obesity/weight gain, anxiety, depression, post-traumatic stress disorder, inflammatory/autoimmune conditions and cancer, including metastatic cancer, advanced cancer, and drug resistant cancer of various types.

AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURAL FRAGMENTS AND PREPARATION METHOD AND APPLICATION THEREOF

The present invention discloses an amide compound containing substituted acetophenone structural fragments, having a structure shown by general formula I:

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The definitions of substituents in the formula are shown in the description. The compound of the present invention has broad-spectrum fungal activity, and has excellent control effects on cucumber downy mildew, wheat powdery mildew, corn rust, cucumber anthracnose, cucumber botrytis and tomato botrytis.

AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURAL FRAGMENTS AND PREPARATION METHOD AND APPLICATION THEREOF

The present invention discloses an amide compound containing substituted acetophenone structural fragments, having a structure shown by general formula I:

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The definitions of substituents in the formula are shown in the description. The compound of the present invention has broad-spectrum fungal activity, and has excellent control effects on cucumber downy mildew, wheat powdery mildew, corn rust, cucumber anthracnose, cucumber botrytis and tomato botrytis.

HERBICIDAL COMPOUNDS

The present invention relates to a compound of formula (I) wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7, R.sup.8, R.sup.9, R.sup.10, R.sup.11 and G are as defined herein; and wherein the compound of formula (I) is optionally present as an agrochemically acceptable salt thereof. These compounds are suitable for use as herbicides. The invention therefore also relates to a method of controlling weeds, especially grassy monocotyledonous weeds, in crops of useful plants, comprising applying a compound of formula (I), or a herbicidal composition comprising such a compound, to the plants or to the locus thereof.

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