C07D265/28

Process for the preparation of bazedoxifene

The invention relates to a process for preparation of the compound 3-methyl-5-benzyloxy-2-(4-benzyloxyphenyl)-1H-indole 5, an intermediate for the synthesis of bazedoxifene and bazedoxifene acetate. ##STR00001##

ELECTROCHROMIC COMPOUND, ELECTROCHROMIC COMPOSITION, AND ELECTROCHROMIC DISPLAY ELEMENT

Provided is an electrochromic compound represented by the following general formula (I) or (II) where R.sub.1 to R.sub.13 are each independently a hydrogen atom, a halogen atom, a monovalent organic group, or a polymerizable functional group, and at least one of the R.sub.1 to the R.sub.13 is a polymerizable functional group.

##STR00001##

ELECTROCHROMIC COMPOUND, ELECTROCHROMIC COMPOSITION, AND ELECTROCHROMIC DISPLAY ELEMENT

Provided is an electrochromic compound represented by the following general formula (I) or (II) where R.sub.1 to R.sub.13 are each independently a hydrogen atom, a halogen atom, a monovalent organic group, or a polymerizable functional group, and at least one of the R.sub.1 to the R.sub.13 is a polymerizable functional group.

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NOVEL ARYL ETHENE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT

The present invention relates to an aryl ethene derivative, for inhibiting an estrogen-related receptor gamma (ERR) activity, a prodrug of same, a solvate of same, a stereoisomer of same or pharmaceutically acceptable salts of same, and a pharmaceutical composition containing same as an active ingredient.

NOVEL ARYL ETHENE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT

The present invention relates to an aryl ethene derivative, for inhibiting an estrogen-related receptor gamma (ERR) activity, a prodrug of same, a solvate of same, a stereoisomer of same or pharmaceutically acceptable salts of same, and a pharmaceutical composition containing same as an active ingredient.

Pyrrolopyrimidine compounds used as TLR7 agonist

The present invention relates to a pyrrolopyrimidine compound as TLR7 agonist, and particularly relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, a preparation process thereof, a pharmaceutical composition containing such compounds and use thereof for manufacturing a medicament against viral infection. ##STR00001##

Pyrrolopyrimidine compounds used as TLR7 agonist

The present invention relates to a pyrrolopyrimidine compound as TLR7 agonist, and particularly relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, a preparation process thereof, a pharmaceutical composition containing such compounds and use thereof for manufacturing a medicament against viral infection. ##STR00001##

Electrochromic compound, electrochromic composition, and electrochromic display element

Provided is an electrochromic compound represented by the following general formula (I) or (II) where R.sub.1 to R.sub.13 are each independently a hydrogen atom, a halogen atom, a monovalent organic group, or a polymerizable functional group, and at least one of the R.sub.1 to the R.sub.13 is a polymerizable functional group.

Electrochromic compound, electrochromic composition, and electrochromic display element

Provided is an electrochromic compound represented by the following general formula (I) or (II) where R.sub.1 to R.sub.13 are each independently a hydrogen atom, a halogen atom, a monovalent organic group, or a polymerizable functional group, and at least one of the R.sub.1 to the R.sub.13 is a polymerizable functional group.

NEW PROCESS FOR EARLY SACUBITRIL INTERMEDIATES
20190256454 · 2019-08-22 ·

The invention relates to a new enantioselective process for producing useful intermediates for the manufacture of NEP inhibitors or prodrugs thereof, in particular NEP inhibitors comprising a -amino--biphenyl--methylalkanoic acid, or acid ester, backbone.