C07D273/01

Heterocyclic GLP-1 agonists

This disclosure relates to GLP-1 agonists of Formula I: ##STR00001##
including pharmaceutically acceptable salts and solvates thereof, and pharmaceutical compositions including the same.

ORGANIC COMPOUNDS AND USES THEREOF

Disclosed are organic compounds including a structure of formula (I). The organic compound has a good rigid structure, so that the organic compound has good thermal stability, and high efficiency and the long lifetime of an OLED device are realized. Also provided are formulations containing the organic compounds, and at least one organic solvent. Further provided are organic electronic devices containing a functional layer, the functional layer comprises the organic compounds.

ORGANIC COMPOUNDS AND USES THEREOF

Disclosed are organic compounds including a structure of formula (I). The organic compound has a good rigid structure, so that the organic compound has good thermal stability, and high efficiency and the long lifetime of an OLED device are realized. Also provided are formulations containing the organic compounds, and at least one organic solvent. Further provided are organic electronic devices containing a functional layer, the functional layer comprises the organic compounds.

METHOD FOR CONTROLLING SOYBEAN RUST FUNGUS HAVING RESISTANCE AGAINST Qo SITE INHIBITOR

The present invention provides a method for controlling a soybean rust fungus having an amino acid substitution of F129L on mitochondrial cytochrome b protein, by applying a compound represented by formula (I) [wherein Q represents a group represented by the following Q1, Q2, Q3, Q4 or Q5 (in the formulae, represents a binding site to benzene ring); X represents an oxygen atom or NH; L represents CH.sub.2, an oxygen atom or NCH.sub.3; E represents a C6-C10 aryl group, etc.; R.sup.1 represents a C1-C3 chain hydrocarbon group or a cyclopropyl group, etc.; R.sup.2 represents a C1-C3 chain hydrocarbon group or a cyclopropyl group, etc.; R.sup.3 represents a C1-C3 alkoxy group or a C1-C3 chain hydrocarbon group, etc.; and n is 0, 1, 2, or 3] or its N oxide or an agriculturally acceptable salt thereof.

##STR00001##

1,3, 5-Dioxazine Derivatives, Method of Preparation and Application Thereof as Sulfide Scavenger
20190300515 · 2019-10-03 ·

The present disclosure relates to 1,3,5-dioxazine derivatives of formula (I) capable of reducing or eliminating hydrogen sulfide and other objectionable sulfides from oil field produced hydrocarbon fluids such as petroleum, fuel oil, gasoline, diesel, liquid propane, liquid butane, an aquaculture and production/processing of syngas/natural gas. The present disclosure further provides a method for preparing 1,3,5-dioxazine derivatives of formula I, and a method for scavenging sulfur-based species including, but not limited to hydrogen sulfide or alkyl/aryl mercaptans from a medium.

1,3, 5-Dioxazine Derivatives, Method of Preparation and Application Thereof as Sulfide Scavenger
20190300515 · 2019-10-03 ·

The present disclosure relates to 1,3,5-dioxazine derivatives of formula (I) capable of reducing or eliminating hydrogen sulfide and other objectionable sulfides from oil field produced hydrocarbon fluids such as petroleum, fuel oil, gasoline, diesel, liquid propane, liquid butane, an aquaculture and production/processing of syngas/natural gas. The present disclosure further provides a method for preparing 1,3,5-dioxazine derivatives of formula I, and a method for scavenging sulfur-based species including, but not limited to hydrogen sulfide or alkyl/aryl mercaptans from a medium.

PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF PIMAVANSERIN

The present disclosure relates to novel, safe and efficient processes for the synthesis of Pimavanserin and salts thereof, as well as novel intermediates that can be used in these processes.

PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF PIMAVANSERIN

The present disclosure relates to novel, safe and efficient processes for the synthesis of Pimavanserin and salts thereof, as well as novel intermediates that can be used in these processes.