Heterocyclic compound and arthropod pest control composition containing same
11779018 · 2023-10-10
Assignee
Inventors
- Ryota Maehata (Takarazuka, JP)
- Kohei Orimoto (Takarazuka, JP)
- Takamasa Tanabe (Chuo-ku, JP)
- Yasumasa Saito (Takarazuka, JP)
Cpc classification
A01N43/80
HUMAN NECESSITIES
C07D413/04
CHEMISTRY; METALLURGY
C07D277/22
CHEMISTRY; METALLURGY
C07D401/04
CHEMISTRY; METALLURGY
C07D409/04
CHEMISTRY; METALLURGY
C07D417/04
CHEMISTRY; METALLURGY
International classification
A01N43/80
HUMAN NECESSITIES
C07D277/22
CHEMISTRY; METALLURGY
C07D401/04
CHEMISTRY; METALLURGY
C07D409/04
CHEMISTRY; METALLURGY
C07D413/04
CHEMISTRY; METALLURGY
Abstract
The present invention provides a compound that has an excellent control effect on arthropod pests, and is represented by formula (I) [wherein Q represents a group represented by Q1, or the like, n is 0, 1, or 2, R.sup.2 represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, or the like, Y.sup.a represents an oxygen atom, a sulfur atom, or NR.sup.3a, G.sup.1 represents a nitrogen atom or CR.sup.5a, G.sup.2 represents a nitrogen atom or CR.sup.5b, A.sup.2 represents a nitrogen atom or CR.sup.4a, A.sup.3 represents a nitrogen atom or CR.sup.4b, A.sup.4 represents a nitrogen atom or CR.sup.4c, and R.sup.3a, R.sup.4a, R.sup.4b, R.sup.4c, R.sup.5a, and R.sup.5b represent a C1-C6 chain hydrocarbon group or the like, and T represents a C1-C10 chain hydrocarbon group which may optionally have one or more halogen atoms, or the like]. ##STR00001##
Claims
1. A compound represented by formula (I): ##STR00142## wherein Q represents a group represented by formula Q1, a group represented by formula Q2, or a group represented by formula Q3, ##STR00143## n is 0, 1 or 2, R.sup.2 represents a C2-C6 alkyl group which may optionally have one or more halogen atoms, a cyclopropyl group, or a cyclopropylmethyl group, Y.sup.a represents an oxygen atom, a sulfur atom, or NR.sup.3a, Y.sup.b represents an oxygen atom, a sulfur atom, or NR.sup.3b, Y.sup.c represents an oxygen atom, a sulfur atom, or NR.sup.3c, G.sup.1 represents a nitrogen atom, or CR.sup.5a, G.sup.2 represents a nitrogen atom, or CR.sup.5b, G.sup.3 represents a nitrogen atom, or CR.sup.5c, R.sup.3a, R.sup.3b, and R.sup.3c are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more substituents selected from Group B, a C3-C7 cycloalkyl group which may optionally have one or more substituents selected from Group E, a phenyl group which may optionally have one or more substituents selected from Group H, a 5- or 6-membered aromatic heterocyclic group which may optionally have one or more substituents selected from Group H, C(O)R.sup.13, C(O)OR.sup.17, C(O)NR.sup.15aR.sup.16a, C(O)NR.sup.11S(O).sub.2R.sup.23, or a hydrogen atom, R.sup.5a, R.sup.5b and R.sup.5c are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more substituents selected from Group B, a C3-C7 cycloalkyl group which may optionally have one or more substituents selected from Group E, a phenyl group which may optionally have one or more substituents selected from Group H, a 5- or 6-membered aromatic heterocyclic group which may optionally have one or more substituents selected from Group H, OR.sup.12, NR.sup.11R.sup.12, NR.sup.11aR.sup.12a, NR.sup.24NR.sup.11R.sup.12, NR.sup.24OR.sup.11, NR.sup.11C(O)R.sup.13, NR.sup.24NR.sup.11C(O)R.sup.13, NR.sup.11C(O)OR.sup.14, NR.sup.24NR.sup.11R.sup.12, NR.sup.24OR.sup.14, NR.sup.11C(O)NR.sup.15aR.sup.16a, NR.sup.24NR.sup.11C(O)NR.sup.15aR.sup.16a, N═CHNR.sup.15aR.sup.16a, N═S(O).sub.xR.sup.15R.sup.16, C(O)R.sup.13, C(O)OR.sup.17, C(O)NR.sup.15aR.sup.16a, C(O)NR.sup.11S(O).sub.2R.sup.23, CR.sup.24═NOR.sup.17, NR.sup.11CR.sup.24═NOR.sup.17, a cyano group, a nitro group, a halogen atom, or a hydrogen atom, x is 0 or 1, A.sup.2 represents CR.sup.4a, A.sup.3 represents CR.sup.4b, A.sup.4 represents CR.sup.4c, R.sup.4a,R.sup.4b, and R.sup.4c are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a nitro group, OR.sup.18, NR.sup.18R.sup.19, a cyan® group, a halogen atom, or a hydrogen atom, R.sup.18 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen acorns, R.sup.19 represents a C1-C6 chain hydrocarbon group which optionally have one or more halogen atoms, or a hydrogen atom, T represents a C1-C10 chain hydrocarbon group which has one or more halogen atoms, a (C1-C5 alkoxy)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkylsulfanyl)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkylsulfinyl)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkysulfonyl group)C2-C5 alkyl group which has one or more halogen atoms, a (C3-C7 cycloalkyl)C1-C3 alkyl group which may optionally have one or more substituents selected from Group G, a C3-C7 cycloalkyl group which may optionally have one or more substituents selected from Group G, OR.sup.1, S(O).sub.mR.sup.1, OS(O).sub.2R.sup.1, NR.sup.1R.sup.29, C(O)R.sup.1, C(O)NR.sup.1R.sup.29, CR.sup.29C(O)R.sup.1, N═CR.sup.1R.sup.30, ##STR00144## ##STR00145## X.sup.1 represents a nitrogen atom, or CR.sup.1a, X.sup.2 represents a nitrogen atom or CR.sup.1b, X.sup.3 represents a nitrogen atom or CR.sup.1c, X.sup.4 represents a nitrogen atom or CR.sup.1d, X.sup.5 represents a nitrogen atom or CR.sup.1e, R.sup.1a, R.sup.1b, R.sup.1c, R.sup.1d, and R.sup.1e are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C3-C6 cycloalkyl group which may optionally have one or more halogen atoms, a halogen atom, or a hydrogen atom, Y.sup.1 represents NR.sup.25, an oxygen atom, or a sulfur atom, Y.sup.2 represents a nitrogen atom, or CR.sup.26, Y.sup.3 represents a nitrogen atom, or CR.sup.27, Y.sup.4 represents a nitrogen atom, or CR.sup.28, R.sup.25 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a C3-C7 cycloalkyl group which may optionally have one or more halogen atoms, a (C3-C7 cycloalkyl) C1-C6 alkyl group which may optionally have one or more halogen atoms, or a hydrogen atom, R.sup.26, R.sup.27, and R.sup.28 are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C3-C6 cycloalkyl group which may optionally have one or more halogen atoms, a halogen atom, or a hydrogen atom, R.sup.1x represents OR.sup.7, OS(O).sub.2R.sup.7, S(O).sub.mR.sup.7, NR.sup.8S(O).sub.2R.sup.7, a C1-C5 chain hydrocarbon group which has one or more halogen atoms, a cyano group, or a halogen atom, R.sup.1y represents OR.sup.7, OS(O).sub.2R.sup.7, S(O).sub.mR.sup.7, NR.sup.8S(O).sub.2R.sup.7, a cyano group, a C1-C5 chain hydrocarbon group which has one or more halogen atoms, or a halogen atom, R.sup.1ay and R.sup.7 are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which has one or more halogen atoms, R.sup.8 represents a C7-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, or a hydrogen atom, m is 0, 1, or 2, R.sup.1 represents a C1-C10 chain hydrocarbon group which has one or more halogen atoms, a (C1-C5 alkoxy)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkylsulfanyl)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkylsulfinyl group)C2-C5 alkyl group which has one or more halogen atoms, a (C1-C5 alkylsulfonyl)C2-C5 alkyl group which has one or more halogen atoms, a (C3-C7 cycloalkyl)C1-C3 alkyl group which has one or more substituents selected from Group G, or a C3-C7 cycloalkyl group which has one or more substituents selected from Group G, R.sup.11, R.sup.17, R.sup.24, and R.sup.29 are identical to or different from each other, and each represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, or a hydrogen atom, R.sup.30 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, or a hydrogen atom, R.sup.12 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C1-C6 alkyl group having one substituent selected from Group F, a phenyl group which may optionally have one or more substituents selected from Group H, a 5- or 6-membered aromatic heterocyclic group which may optionally have one or more substituents selected from Group H, S(O).sub.2R.sup.23, or a hydrogen atom, R.sup.23 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, or a phenyl group which may optionally have one or more substituents selected from Group D, R.sup.11a and R.sup.12a combined together with a nitrogen atom to which they are attached to form a 3 to 7 membered nonaromatic heterocyclic group which may optionally have one or more substituents selected from Group E, R.sup.13 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C3-C7 cycloalkyl group which may optionally have one or more halogen atoms, a (C3-C6 cycloalkyl)C1-C3 alkyl group which may optionally have one or more halogen atoms, a phenyl group which may optionally have one or more substituents selected from Group D, a 5- or 6-membered aromatic heterocyclic group which may optionally have one or more substituents selected from Group D, or a hydrogen atom, R.sup.14 represents a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C3-C7 cycloalkyl group which may optionally have one or more halogen atoms, a (C3-C6 cycloalkyl)C1-C3 alkyl group which may optionally have one or more halogen atoms, or a phenyl C1-C3 alkyl group wherein the phenyl moiety in the phenyl C1-C3 alkyl group may have optionally one or more substituents selected from Group D, R.sup.15 and R.sup.16 are identical to or different from each other, and each represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, R.sup.15a represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, or a hydrogen atom, and R.sup.16a a represents a C1-C6 chain hydrocarbon group which may optionally have one or more substituents selected from Group F, a C3-C7 cycloalkyl group which may optionally have one or more substituents selected from Group J, or a hydrogen atom, Group B: a group consisting of a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a C3-C6 alkenyloxy group which may optionally have one or more halogen atoms, a C3-C6 alkynyloxy group which may optionally have one or more halogen atoms, a C1-C6 alkylsulfanyl group which may optionally have one or more halogen atoms, a C1-C6 alkylsulfinyl group which may optionally have one or more halogen atoms, a C1-C6 alkylsulfonyl group which may optionally have one or more halogen atoms, a C3-C6 cycloalkyl group which may optionally have one or more halogen atoms, a cyano group, a hydroxy group, and a halogen atom, Group C: a group consisting of a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a C3-C6 alkenyloxy group which may optionally have one or more halogen atoms, a C3-C6 alkynyloxy group which may optionally have one or more halogen atoms, and a halogen atom, Group D: a group consisting of a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a hydroxy group, a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a C3-C6 alkenyloxy group which may optionally have one or more halogen atoms, a C3-C6 alkynyloxy group which may optionally have one or more halogen atoms, a sulfanyl group, a C1-C6 alkylsulfanyl group which may optionally have one or more halogen atoms, a C1-C6 alkylsulfinyl group which may optionally have one or more halogen atoms, a C1-C6 alkylsulfonyl group which may optionally have one or more halogen atoms, an amino group, NHR.sup.21, NR.sup.21R.sup.22, C(O)R.sup.21, OC(O)R.sup.21, C(O)OR.sup.21, a cyano group, a nitro group, and a halogen atom, R.sup.21 and R.sup.22 are identical to or different from each other, and each represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, Group E: a group consisting of a C1-C6 chain hydrocarbon group which may optionally have one or more halogen atoms, a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a C3-C6 alkenyloxy group which may optionally have one or more halogen atoms, a C3-C6 alkynyloxy group which may optionally have one or more halogen atoms, a halogen atom, an oxo group, a hydroxy group, a cyano group, and a nitro group, Group F: a group consisting of a C1-C6 alkoxy group which may optionally have one or more halogen atoms, a phenyl group which may optionally have one or more substituents selected from Group D, a 5- or 6- membered aromatic heterocyclic group which may optionally have one or more substituents selected from Group D, a C3-C7 cycloalkyl group which may optionally have one or more halogen atoms, a 3 to 7 membered nonaromatic heterocyclic group which may optionally have one or more substituents selected from Group C, an amino group, NHR.sup.21, NR.sup.21R.sup.22, and a cyano group, Group G: a group consisting of a C1-C6 alkyl group which has one or more halogen atoms, and a halogen atom, Group H: a group consisting of a C1-C6 alkyl group which may optionally have one or more halogen atoms, OR.sup.10, NR.sup.9R.sup.10, C(O)R.sup.10, C(O)NR.sup.9R.sup.10, OC(O)R.sup.9, OC(O)OR.sup.9, NR.sup.10C(O)R.sup.9, NR.sup.10C(O)OR.sup.9, C(O)OR.sup.10, a halogen atom, a nitro group, a cyano group, an amino group, and a 5- or 6-membered aromatic heterocyclic group, R.sup.9 represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, or a C3-C6 cycloalkyl group which may optionally have one or more halogen atoms, R.sup.10 represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, a C3-C6 cycloalkyl group which may optionally have one or more halogen atoms, or a hydrogen atom, Group J: a group consisting of a C1-C6 alkyl group which may optionally have one or more halogen atoms, a halogen atom, and a cyano group.
2. The compound according to claim 1, wherein R.sup.2 represents a C1-C6 alkyl group, R.sup.3a, R.sup.3b, and R.sup.3c are identical to or different from each other, and each represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, a phenyl group, a pyridyl group, a pyrimidinyl group, a pyrazolyl group, a triazolyl group, wherein the phenyl group, the pyridyl group, the pyrimidinyl group, the pyrazolyl group, and the triazolyl group may optionally have one or more substituents selected from Group HUN, or a hydrogen atom, R.sup.4a, R.sup.4b, and R.sup.4c are identical to or different from each other, and each presents a hydrogen atom, or a halogen atom, T represents OR.sup.1, and R.sup.1 represents a C1-C5 chain hydrocarbon group which has one or more halogen atoms, Q represents a group represented by formula Q1, or a group represented by formula Q3, and R.sup.5a, R.sup.5b, and R.sup.5c are identical to or different from each other, and each represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, a phenyl group, a pyridyl group, a pyrimidinyl group, a pyrazolyl group, a triazolyl group, wherein the phenyl group, the pyridyl group, the pyrimidinyl group, the pyrazolyl group, and the triazolyl group may optionally have one or more substituents selected from Group H, OR.sup.12, NR.sup.11R.sup.12NR.sup.11C(O)OR.sup.14, a halogen atom, or a hydrogen atom.
3. The compound according to claim 1, wherein R.sup.1 represents a C1-C5 alkyl group having three or more fluorine atoms, R.sup.3a, R.sup.3b, and R.sup.3c are identical to or different from each other, and each represent a C1-C6 alkyl group which may optionally have one or more halogen atoms, or a hydrogen atom, R.sup.4a, R.sup.4b, and R.sup.4c represent a hydrogen atom, and R.sup.5a, R.sup.5b, and R.sup.5c are identical to or different from each other, and each represents a C1-C6 alkyl group which may optionally have one or more halogen atoms, OR.sup.12, a halogen atom, or a hydrogen atom.
4. The compound of claim 1, wherein R.sup.2 represents an ethyl group.
5. The compound of claim 1, wherein Q represents a group represented by formula Q1.
6. The compound of claim 1, wherein Q represents a group represented by formula Q3.
7. A composition for controlling a harmful arthropod comprising the compound of claim 1 and an inert carrier.
8. A method for controlling a harmful arthropod, the method comprising: applying an effective amount of the compound of claim 1 to a harmful arthropod or a habitat where a harmful arthropod lives.
9. A composition comprising one or more ingredients selected from Group (a) and Group (b), and the compound of claim 1: Group (a): a group consisting of insecticidal ingredients, miticide ingredients, and nematicidal ingredients; and Group (b): fungicidal ingredient.
10. A method for controlling a, harmful arthropod, the method comprising: applying an effective amount of the composition of claim 9 to a harmful arthropod or a habitat where the harmful arthropod lives.
11. A seed or vegetative reproductive organ carrying an effective amount of the compound of claim 1.
Description
EXAMPLES
(1) Hereinafter, the present invention is explained in more detail by using the Preparation Example, the Reference Preparation Example, the Formulation Example, and the Test Example, however, the present invention should not be limited to these examples.
Preparation Example 1
(2) A mixture of 2,4-dibromothiazole 15 g, 4-fluorophenyl boronic acid 9.5 g, palladium (II) acetate 690 mg, 4,5′-bis(diphenylphoshino)-9,9′-dimethyl xanthene 1.8 g, tripotassium phosphate 39 g, and THF 300 mL was stirred at 60° C. for 10 hours. Water was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to silica gel column chromatography to obtain an intermediate compound 1 represented by the below-mentioned formula 12 g.
(3) ##STR00059##
(4) Intermediate compound 1: .sup.1H-NMR (CDCl.sub.3) δ: 7.95-7.91 (2H, m), 7.21 (1H, s), 7.16-7.11 (2H, m).
Preparation Example 2
(5) To a mixture of diisopropyl amine 1.2 mL and THF 5 mL was added butyl lithium (1.6 M hexane solution) 5.7 mL at −50° C., and the mixture was stirred for 20 minutes. To the resulting mixture was added a mixture of the intermediate compound 1 1.5 g and THF 7 mL, and the mixture was stirred for 1 hour. To the resulting mixture was added zinc chloride (1.0 M diethyl ether solution) 15 mL. The resulting mixture was raised gradually from −50° C. to room temperature, and the mixture was stirred at room temperature for 2 hours. To the resulting mixture were added 2-bromo-5-(2,2,3,3,3-pentafluoropropoxy)pyridine 0.59 g, which was prepared according to the method described in WO 2016/121969, tetrakis(triphenylphosphine)palladium (0) 340 mg, and THE 5 mL, and the mixture was stirred at 50° C. for 3 hours. To the resulting mixture was added 2N hydrochloric acid, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to silica gel column chromatography to obtain an intermediate compound 2 represented by the below-mentioned formula 920 mg.
(6) ##STR00060##
(7) Intermediate compound 2: .sup.1H-NMR (CDCl.sub.3) δ: 8.39 (1H, d), 8.37 (1H, d), 7.97 (2H, dd), 7.38 (1H, dd), 7.15 (2H, t), 4.53 (2H, t).
Preparation Example 3
(8) To a mixture of the intermediate compound 2 920 mg, sodium hydride (60%, oily) 76 mg, and DMF 5 mL was added ethanethiol 0.14 mL, and the mixture was stirred at room temperature for 8 hours. To the resulting mixture was added saturated aqueous sodium hydrocarbonate solution, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 1 represented by the below-mentioned formula 270 mg.
(9) ##STR00061##
(10) Present compound 1: .sup.1H-NMR (CDCl.sub.3) δ: 8.38-8.36 (2H, m), 8.00-7.93 (2H, m), 7.38-7.33 (1H, m), 7.17-7.12 (2H, m), 4.53 (2H, t), 3.02 (2H, q), 1.37 (3H, t).
Preparation Example 4
(11) To a mixture of the present compound 1 270 mg, and ethyl acetate 5 mL was added m-chloroperbenzoic acid (74%) 320 mg under ice-cooling, and the mixture was raised to room temperature, and thereafter, the mixture was stirred for 4 hours. To the resulting mixture were added saturated aqueous sodium thiosulfate solution and saturated aqueous sodium hydrogen carbonate solution, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 2 represented by the below-mentioned formula 150 mg.
(12) ##STR00062##
(13) Present compound 2: .sup.1H-NMR (CDCl.sub.3) δ: 8.38 (1H, d), 8.26 (1H, d), 7.98-7.94 (2H, m), 7.35 (1H, dd), 7.20-7.14 (2H, m), 4.53 (2H, t), 3.62 (2H, q), 1.42 (3H, t).
Preparation Example 5
(14) An intermediate compound 3 was obtained by using cyclopropyl boronic acid in place of 4-fluorophenyl boronic acid according to the method described in the Preparation Example 1.
(15) ##STR00063##
(16) Intermediate compound 3: .sup.1H-NMR (CDCl.sub.3) δ: 6.96 (1H, s), 2.34-2.24 (1H, m), 1.18-1.07 (4H, m).
Preparation Example 6
(17) An intermediate compound 4 was obtained by using the intermediate compound 3 in place of the intermediate compound 1 according to the method described in the Preparation Example 2.
(18) ##STR00064##
(19) Intermediate compound 4: .sup.1H-NMR (CDCl.sub.3) δ: 8.32 (1H, dd), 8.28 (1H, dd), 7.34 (1H, dd), 4.56-4.43 (2H, m), 2.34-2.26 (1H, m), 1.23-1.08 (4H, m).
Preparation Example 7
(20) A mixture of the intermediate compound 705 mg, ethanethiol 190 μL, tris(benzylideneacetone)palladium (0) 300 mg, 4,5′-bis(diphenylphoshino)-9,9′-dimethylxanthene 380 mg, diisopropylethylamine 840 μL, and cyclopently methyl ether 5 mL was stirred at 100° C. for 8 hours. The resulting mixture was allowed to cool, and thereafter, thereto was added saturated aqueous sodium hydrogen carbonate solution, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 3 represented by the below-mentioned formula 490 mg.
(21) ##STR00065##
(22) Present compound 3: .sup.1H-NMR (CDCl.sub.3) δ: 8.31 (1H, d), 8.03 (1H, dd), 7.42-7.28 (1H, m), 4.53-4.45 (2H, m), 3.32-3.11 (2H, m), 2.40-2.24 (1H, m), 1.33 (3H, t), 1.18-1.09 (4H, m).
Preparation Example 8
(23) The present compound 4 was obtained by using the present compound 3 in place of the present compound 1 according to the method described in the Preparation Example 4.
(24) ##STR00066##
(25) Present compound 4: 1H-NMR (CDCl.sub.3) δ: 8.33 (1H, dd), 8.12 (1H, dd), 7.31 (1H, dd), 4.50 (2H, d), 3.48 (2H, q), 2.36-2.28 (1H, m), 1.34 (3H, t), 1.25-1.18 (2H, m), 1.14-1.10 (2H, m).
Preparation Example 9
(26) A mixture of ethyl chloro(hydroxyimimo) acetate 0.15 g, which was prepared according to the method described in WO 2012/117421, 2-ethanesulfonyl-1-[5-(2,2,3,3,3-pentafluoropropoxy)pyridin-2-yl]ethanone (hereinafter, referred to as “Intermediate compound 5”), which was prepared according to the method described in WO 2016/121969, 0.38 g, trimethylamine 0.22 g, and ethanol 3 mL was stirred at room temperature for 12 hours. To the resulting mixture was added water, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 5 represented by the below-mentioned formula 100 mg.
(27) ##STR00067##
(28) Present compound 5: 1H-NMR (CDCl.sub.3) δ: 8.54 (1H, d), 7.97 (1H, d), 7.42 (1H, dd), 4.57 (2H, t), 4.51 (2H, q), 3.77 (2H, q), 1.47-1.28 (6H, m).
Preparation Example 10
(29) A mixture of the present compound 5 400 mg, 1N aqueous lithium hydroxide solution 1 mL, and THF 3 mL was stirred at room temperature for 5 hours. To the resulting mixture was added water 5 mL, and the mixture was extracted with MTBE. To the resulting aqueous layer was added 2N hydrochloric acid to adjust pH to 4, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate and concentrated under reduced pressure. The resulting residue was added to a mixture of triethylamine 222 mg, 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride salt 0.38 g, and isobutyl amine 141 mg under ice-cooling. The resulting mixture was raised to room temperature, and stirred for 8 hours. To the resulting mixture was added water, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 6 represented by the below-mentioned formula 260 mg.
(30) ##STR00068##
(31) Present compound 6: 1H-NMR (CDCl.sub.3) δ: 8.52 (1H, d), 7.90 (1H, d), 7.40 (1H, dd), 6.63 (1H, br s), 4.56 (2H, t), 3.80 (2H, q), 3.33 (2H, t), 1.98-1.91 (1H, m), 1.45 (3H, t), 1.01 (6H, d).
Preparation Example 11
(32) The present compound 7 and the present compound 8 each represented by the below-mentioned formula were obtained according to the Preparation Example 9.
(33) ##STR00069##
(34) Present compound 7: 1H-NMR (CDCl.sub.3) δ: 8.56 (1H, t), 8.13 (2H, s), 8.07-8.03 (2H, m), 7.47 (1H, dd), 4.60 (2H, t), 3.77 (2H, q), 1.37 (3H, t).
(35) ##STR00070##
(36) Present compound 8: 1H-NMR (CDCl.sub.3) δ: 8.54 (1H, dd), 7.99 (1H, dd), 7.72-7.66 (2H, m), 7.44 (1H, dd), 7.23-7.15 (2H, m), 4.58 (2H, t), 3.55 (2H, q), 1.29 (3H, t).
Preparation Example 12
(37) To a mixture of the intermediate compound 5 1.7 g, and ally bromide 320 mg, and DMSO 10 mL was added potassium hydroxide 320 mg at room temperature under nitrogen atmosphere, and the mixture was stirred at 80° C. for 30 minutes. To the resulting mixture was added water at room temperature, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. To the resulting residue was added methanol 10 mL, and ozone was bubbled to the resulting mixture at room temperature for 10 minutes. To the resulting mixture was added dimethyl sulfide 530 μL at −78° C., and the mixture was stirred at room temperature for 1 day. The resulting mixture was concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain an intermediate compound 6 represented by the below-mentioned formula 1.2 g.
(38) ##STR00071##
(39) Intermediate compound 6: .sup.1H-NMR (CDCl.sub.3) δ: 9.77 (1H, s), 8.49 (1H, d), 8.18 (1H, d), 7.41 (1H, dd), 6.39 (1H, dd), 4.59 (2H, t), 3.62-3.53 (2H, m), 3.30-3.07 (2H, m), 1.40 (3H, t).
Preparation Example 13
(40) To a mixture of the intermediate compound 6 250 mg and ethanol 2 mL was added ammonium acetate 53 mg at room temperature under nitrogen atmosphere, and the mixture was stirred at 80° C. for 1 hour. To the resulting mixture was added water at room temperature, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, and dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 9 represented by the below-mentioned formula 31 mg.
(41) ##STR00072##
(42) Present compound 9: .sup.1H-NMR (CDCl.sub.3) δ: 10.13 (1H, s), 8.55 (1H, dd), 8.32 (1H, d), 7.32 (1H, dd), 6.90 (1H, t), 6.74 (1H, t), 4.51 (2H, t), 3.14 (2H, q), 1.26 (3H, t).
Preparation Example 14
(43) To a mixture of the present compound 9 200 mg, methyl iodide 160 μL and DMF 2 mL was added sodium hydride (60%, oily) 23 mg at room temperature, and the mixture was stirred for 30 minutes. To the resulting mixture was added water, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 10 represented by the below-mentioned formula 120 mg.
(44) ##STR00073##
(45) Present compound 10: 1H-NMR (CDCl.sub.3) δ: 8.44 (1H, dd), 7.74 (1H, dd), 7.35 (1H, dd), 6.73 (1H, d), 6.63 (1H, d), 4.53 (2H, t), 3.58 (3H, s), 2.92 (2H, q), 1.14 (3H, t).
Preparation Example 15
(46) The present compound 11 was obtained by using isopropyl iodide in place of methyl iodide according to the Preparation Example 14.
(47) ##STR00074##
(48) Present compound 11: .sup.1H-NMR (CDCl.sub.3) δ: 8.44 (1H, dd), 7.67 (1H, dd), 7.35 (1H, dd), 6.88 (1H, d), 6.67 (1H, d), 4.53 (2H, t), 4.31-4.24 (1H, m), 2.91 (2H, q), 1.37 (6H, d), 1.15 (3H, t).
Preparation Example 16
(49) To a mixture of the intermediate compound 6 240 mg and toluene 10 mL was added lowesson reagent 630 mg at room temperature, and the mixture was stirred at 80° C. for 1 hour. To the resulting mixture was added water at room temperature, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 12 represented by the below-mentioned formula 190 mg.
(50) ##STR00075##
(51) Present compound 12: .sup.1H-NMR (CDCl.sub.3) δ: 8.44 (1H, d), 7.94 (1H, d), 7.53 (1H, d), 7.42 (1H, d), 7.36 (1H, dd), 4.54 (2H, t), 3.34 (2H, q), 1.27 (3H, t).
Preparation Example 17
(52) To a mixture of the intermediate compound 5 10 g and chloroform 40 mL were added N-chlorosuccinimide 4.1 g and p-toluenesulfonic acid 530 mg successively, and the mixture was stirred at 60° C. for 2 hours. The resulting mixture was allowed to cool to room temperature, and thereto was added aqueous sodium thiosulfate solution, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting reside was subjected to a silica gel column chromatography to obtain the intermediate compound 7 represented by the below-mentioned formula 2.1 g.
(53) ##STR00076##
(54) Intermediate compound 7: .sup.1H-NMR (CDCl.sub.3) δ: 8.46 (1H, d), 8.19 (1H, d), 7.41 (1H, dd), 4.59 (2H, t), 3.61-3.47 (1H, m), 3.43-3.28 (2H, m), 1.46 (3H, t).
Preparation Example 18
(55) To a mixture of the intermediate compound 7 1.0 g and ethanol 40 mL were added thiourea 580 mg and pyridine 400 mg successively at room temperature, and the mixture was stirred under reflux for 2 hours. The resulting mixture was allowed to cool to room temperature, water was added thereto, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, and dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 13 represented by the below-mentioned formula 200 mg.
(56) ##STR00077##
(57) Present compound 13: .sup.1H-NMR (CDCl.sub.3) δ: 8.40 (1H, dd), 7.93 (1H, dd), 7.32 (1H, dd), 5.40 (2H, s), 4.52 (2H, t), 3.87 (2H, q), 1.41 (3H, t).
Preparation Example 19
(58) To a mixture of the intermediate compound 7 500 mg and ethanol 5 mL was added thiobenzamide 520 mg at room temperature, and the mixture was stirred at 100° C. for 30 minutes. The resulting mixture was allowed to cool to room temperature, and water was added thereto, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to silica gel column chromatography to obtain the present compound 14 represented by the below-mentioned formula 74 mg.
(59) ##STR00078##
(60) Present compound 14: .sup.1H-NMR (CDCl.sub.3) δ: 8.45 (1H, d), 8.23 (1H, d), 8.02 (2H, dd), 7.56-7.48 (3H, m), 7.40 (1H, dd), 4.56 (2H, t), 4.05 (2H, q), 1.46 (3H, t).
Preparation Example 20
(61) To a mixture of the present compound 13 230 mg and DMF 2 mL was added t-butyl nitrite 80 μL at 60° C., and the mixture was stirred under reflux for 30 minutes. The resulting mixture was allowed to cool to room temperature, water was added thereto, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 15 represented by the below-mentioned formula 73 mg.
(62) ##STR00079##
(63) Present compound 15: .sup.1H-NMR (CDCl.sub.3) δ: 8.99 (1H, s), 8.44 (1H, d), 8.14 (1H, d), 7.39 (1H, dd), 4.55 (2H, t), 4.04 (2H, q), 1.42 (3H, t).
Preparation Example 21
(64) A mixture of the intermediate compound 5 30 g and N,N-dimethylformamide dimethyl acetal 120 mL was stirred at room temperature for 12 hours. The precipitated out-solids were filtered, and washed with MTBE. The resulting solids were dried under reduced pressure to obtain the intermediate compound 8 represented by the below-mentioned formula 24 g.
(65) ##STR00080##
(66) Intermediate compound 8: .sup.1H-NMR (CDCl.sub.3) δ: 8.30 (1H, dd), 7.96 (1H, dd), 7.84 (1H, s), 7.34 (1H, dd), 4.52 (2H, t), 3.47 (2H, q), 3.26 (3H, s), 2.70 (3H, s), 1.33 (3H, t).
Preparation Example 22
(67) To a mixture of the intermediate compound 8 0.5 mg, sodium hydrogen carbonate 0.2 g, and ethanol 3 mL was added 4-fluorophenyl hydrazine hydrochloride salt 0.3 mg, and the mixture was stirred under reflux for 5 hours. The resulting mixture was allowed to cool to room temperature, water was added thereto, and the mixture was extracted with MTBE. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography to obtain the present compound 16 represented by the below-mentioned formula 0.53 g.
(68) ##STR00081##
(69) Present compound 16: .sup.1H-NMR (CDCl.sub.3) δ: 8.38 (1H, d), 8.13 (1H, d), 7.36-7.33 (1H, m), 7.25-7.22 (3H, m), 7.07-7.00 (2H, m), 4.49 (2H, t), 3.29 (2H, q), 1.31 (3H, t).
(70) Next, examples of the present compounds which are prepared by either the Preparation Examples described in Examples or the Process described herein are shown below.
(71) As used herein, “Me” represents a methyl group, “Et” represents an ethyl group, “Pr” represents a propyl group, “i-Pr” represents an isopropyl group, “c-Pr” represents a cyclopropyl group, “Ph” represents a phenyl group, “Py2” represents a 2-pyridyl group, “Py3” represents a 3-pyridyl group, “Py4” represents a 4-pyridyl group, and “Bn” represents a benzyl group. When c-Pr, Ph, Py2, Py3, and Py4 have a substituent, the substituent is written with its substituted position before the symbol. For example, “1-CN-c-Pr” represents a 1-cyanocyclopropyl group, “3,4-F.sub.2-Ph” represents a 3,4-difluorophenyl group, “4-CF.sub.3—Py2” represents a 4-(trifluoromethyl)-2-pyridyl group, and “5-OCH.sub.2CF.sub.2CF.sub.3-Py2” represents a 5-(2,2,3,3,3-pentafluoropropoxy)-2-pyridyl group.
(72) Here Q10 to Q28 represents the following groups respectively.
(73) ##STR00082## ##STR00083## ##STR00084##
(74) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX1”).
(75) [Table 1]
(76) TABLE-US-00001 TABLE 1A CF.sub.3 CHF.sub.2 CH.sub.2CF.sub.3 CF.sub.2CF.sub.3 CH.sub.2CF.sub.2CF.sub.3 CF.sub.2CF.sub.2CF.sub.3 CF.sub.2CF.sub.2CF.sub.2CF.sub.3 CF.sub.2CF.sub.2CF.sub.2CF.sub.2CF.sub.3 OCF.sub.3 OCHF.sub.2 OCH.sub.2CF.sub.3 OCH.sub.2CHF.sub.2 OCF.sub.2CF.sub.3 OCH(CH.sub.3)CF.sub.3 OCH.sub.2CF.sub.2CHF.sub.2 OCH.sub.2CF.sub.2CF.sub.3 OCF.sub.2CF.sub.2CF.sub.3 OCH.sub.2CF.sub.2CHFCF.sub.3 OCH.sub.2CF.sub.2CF.sub.2CF.sub.3 OCF.sub.2CF.sub.2CF.sub.2CF.sub.3 OCH.sub.2CF.sub.2CF.sub.2CF.sub.2CF.sub.3
(77) TABLE-US-00002 TABLE 2A SCF.sub.3 SCH.sub.2CF.sub.3 SCF.sub.2CF.sub.3 SCH.sub.2CF.sub.2CF.sub.3 SCF.sub.2CF.sub.2CF.sub.3 SCH.sub.2CF.sub.2CF.sub.2CF.sub.3 SCF.sub.2CF.sub.2CF.sub.2CF.sub.3 S(O)CF.sub.3 S(O)CH.sub.2CF.sub.3 S(O)CF.sub.2CF.sub.3 S(O)CH.sub.2CF.sub.2CF.sub.3 S(O)CF.sub.2CF.sub.2CF.sub.3 S(O)CH.sub.2CF.sub.2CF.sub.2CF.sub.3 S(O)CF.sub.2CF.sub.2CF.sub.2CF.sub.3 S(O).sub.2CF.sub.3 S(O).sub.2CH.sub.2CF.sub.3 S(O).sub.2CF.sub.2CF.sub.3 S(O).sub.2CH.sub.2CF.sub.2CF.sub.3 S(O).sub.2CF.sub.2CF.sub.2CF.sub.3 S(O).sub.2CH.sub.2CF.sub.2CF.sub.2CF.sub.3 S(O).sub.2CF.sub.2CF.sub.2CF.sub.2CF.sub.3
(78) TABLE-US-00003 TABLE 3A NHCH.sub.2CF.sub.3 NHCH.sub.2CF.sub.2CF.sub.3 NHCH.sub.2CF.sub.2CF.sub.2CF.sub.3 NMeCH.sub.2CF.sub.3 NMeCH.sub.2CF.sub.2CF.sub.3 NMeCH.sub.2CF.sub.2CF.sub.2CF.sub.3 NEtCH.sub.2CF.sub.3 NEtCH.sub.2CF.sub.2CF.sub.3 NEtCH.sub.2CF.sub.2CF.sub.2CF.sub.3 OS(O).sub.2CF.sub.3 OS(O).sub.2CF.sub.2CF.sub.3 OS(O).sub.2CF.sub.2CF.sub.2CF.sub.3 CH.sub.2OCF.sub.3 CH.sub.2OCH.sub.2CF.sub.3 CH.sub.2OCF.sub.2CF.sub.3 C(O)CF.sub.3 C(O)CF.sub.2CF.sub.3 C(O)CF.sub.2CF.sub.2CF.sub.3 C(O)NMeCH.sub.2CF.sub.3 NMeC(O)CF.sub.3 N═CEtCH.sub.2CF.sub.3
(79) TABLE-US-00004 TABLE 4A 3-CF.sub.3—Ph 4-CF.sub.3—Ph 3,5-(CF.sub.3).sub.2—Ph 3-SCF.sub.3—Ph 3-S(O)CF.sub.3—Ph 3-S(O).sub.2CF.sub.3—Ph 4-SCF.sub.3—Ph 4-S(O)CF.sub.3—Ph 4-S(O).sub.2CF.sub.3—Ph
(80) TABLE-US-00005 TABLE 5A 4-CF.sub.3—Py2 5-CF.sub.3—Py2 4-SCF.sub.3—Py2 4-S(O)CF.sub.3—Py2 4-S(O).sub.2CF.sub.3—Py2 5-SCF.sub.3—Py2 5-S(O)CF.sub.3—Py2 5-S(O).sub.2CF.sub.3—Py2 5-NMeCH.sub.2CF.sub.3—Py2
(81) TABLE-US-00006 TABLE 6A 5-CF.sub.3—Py3 6-CF.sub.3—Py3 5-SCF.sub.3—Py3 5-S(O)CF.sub.3—Py3 5-S(O).sub.2CF.sub.3—Py3 6-SCF.sub.3—Py3 6-S(O)CF.sub.3—Py3 6-S(O).sub.2CF.sub.3—Py3 6-NMeCH.sub.2CF.sub.3—Py3
(82) ##STR00085##
(83) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX2”).
(84) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX3”).
(85) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX4”).
(86) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX5”).
(87) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX6”).
(88) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX7”).
(89) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX8”).
(90) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX9”).
(91) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, and R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX10”).
(92) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX9”).
(93) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, and R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX12”).
(94) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, and R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX13”).
(95) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX14”).
(96) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX15”).
(97) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX16”).
(98) A present compound wherein A.sup.2 represents a nitrogen represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX17”).
(99) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX18”).
(100) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX19”).
(101) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX20”).
(102) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX21”).
(103) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX21”).
(104) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX22”).
(105) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX23”).
(106) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX24”).
(107) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX25”).
(108) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX26”).
(109) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX27”).
(110) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3, R.sup.5a and R.sup.5b represent a hydrogen atom and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX28”).
(111) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX29”).
(112) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX30”).
(113) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX31”).
(114) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX32”).
(115) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX33”).
(116) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX34”).
(117) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represent a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX35”).
(118) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represent a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX36”).
(119) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX37”).
(120) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX38”).
(121) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.51 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX39”).
(122) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX40”).
(123) A present compound wherein A.sup.2 represents a nitrogen represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX41”).
(124) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX42”).
(125) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX43”).
(126) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX44”).
(127) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX45”).
(128) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX46”).
(129) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX47”).
(130) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX48”).
(131) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 and R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX49”).
(132) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 and R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX50”).
(133) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 and R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX51”).
(134) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q13, R.sup.3 and R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX52”).
(135) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX53”).
(136) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX54”).
(137) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX55”).
(138) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q13, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX56”).
(139) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q14, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX57”).
(140) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q14, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX58”).
(141) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q14, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX59”).
(142) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q14, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX60”).
(143) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX61”).
(144) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX62”).
(145) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX63”).
(146) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX64”).
(147) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX65”).
(148) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX66”).
(149) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX67”).
(150) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX68”).
(151) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX69”).
(152) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX70”).
(153) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX71”).
(154) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, R.sup.5b represents a fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX72”).
(155) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX73”).
(156) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX74”).
(157) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX75”).
(158) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX76”).
(159) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX77”).
(160) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX78”).
(161) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX79”).
(162) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX80”).
(163) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX81”).
(164) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX82”).
(165) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX83”).
(166) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX84”).
(167) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX85”).
(168) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX86”).
(169) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX87”).
(170) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX88”).
(171) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX89”).
(172) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX90)).
(173) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX91”).
(174) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX92”).
(175) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX93”).
(176) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX94”).
(177) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represent a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX95”).
(178) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represent a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX96”).
(179) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX97”).
(180) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX98”).
(181) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX99”).
(182) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX100”).
(183) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX101”).
(184) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX102”).
(185) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by 17, R.sup.3 represents a methyl group, and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX103”).
(186) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX104”).
(187) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX105”).
(188) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX106”).
(189) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX107”).
(190) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX108”).
(191) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX109”).
(192) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a cyclopropyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX110”).
(193) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a 4-fluorophenyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX111”).
(194) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a hydrogen atom, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX112”).
(195) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a hydrogen atom, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX112”).
(196) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a cyclopropyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX113”).
(197) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a 4-fluorophenyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX114”).
(198) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a hydrogen atom, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX115”).
(199) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a cyclopropyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX116”).
(200) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q18, R.sup.3 represents a 4-fluorophenyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX117”).
(201) A present compound wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, R.sup.3 represents a hydrogen atom, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX118”).
(202) A present compound wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, R.sup.3 represents a cyclopropyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX119”).
(203) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, R.sup.3 represents a 4-fluorophenyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX120”).
(204) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q19, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX121”).
(205) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q19, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX122”).
(206) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q19, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX123”).
(207) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q19, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX124”).
(208) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 and R.sup.5a represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX125”).
(209) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a cyclopropyl group, R.sup.5a represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX126”).
(210) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a cyclopropyl group, R.sup.5a represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX127”).
(211) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 and R.sup.5a represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX128”).
(212) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a cyclopropyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX129”).
(213) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a 4-fluorophenyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX130”).
(214) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 and R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX131”).
(215) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a cyclopropyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX132”).
(216) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a 4-fluorophenyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX133”).
(217) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 and R.sup.5a represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX134”).
(218) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a cyclopropyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX135”).
(219) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a 4-fluorophenyl group, R.sup.5a represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX136”).
(220) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX137”).
(221) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a cyclopropyl group, and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX138”).
(222) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a 4-fluorophenyl group, and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX139”).
(223) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX140”).
(224) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a cyclopropyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX141”).
(225) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a 4-fluorophenyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX142”).
(226) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 and R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX143”).
(227) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a cyclopropyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX144”).
(228) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.3 represents a 4-fluorophenyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX145”).
(229) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.3 and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX146”).
(230) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.3 represents a cyclopropyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX147”).
(231) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.3 represents a 4-fluorophenyl group, R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX148”).
(232) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX149”).
(233) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX150”).
(234) A present compound wherein A.sup.2, A.sup.3, and A.sup.4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX151”).
(235) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX152”).
(236) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX153”).
(237) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX154”).
(238) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX155”).
(239) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX156”).
(240) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, R.sup.3 represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX157”).
(241) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.3 represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX158”).
(242) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.3 represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX159”).
(243) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.3 represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX160”).
(244) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5a and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX161”).
(245) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX162”).
(246) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX163”).
(247) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX164”).
(248) A present compound wherein A.sup.2 represents a nitrogen represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX165”).
(249) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX166”).
(250) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX167”).
(251) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX168”).
(252) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX169”).
(253) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represents CH, Q represents a group represented by Q23, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX170”).
(254) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX171”).
(255) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX172”).
(256) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX173”).
(257) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX174”).
(258) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX175”).
(259) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX176”).
(260) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A](hereinafter, referred to as “Compound class SX177”).
(261) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX178”).
(262) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX179”).
(263) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX180”).
(264) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX181”).
(265) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX182”).
(266) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX183”).
(267) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX184”).
(268) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.5c represents a hydrogen atom, R.sup.3, R.sup.5b and R.sup.5c represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX185”).
(269) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX186”).
(270) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX187”).
(271) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX188”).
(272) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX189”).
(273) A present compound wherein A.sup.2 represents a nitrogen represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX190”).
(274) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX191”).
(275) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX192”).
(276) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX193”).
(277) A present compound wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX194”).
(278) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX195”).
(279) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX196”).
(280) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX197”).
(281) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX198”).
(282) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX199”).
(283) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX200”).
(284) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX201”).
(285) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX202”).
(286) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX203”).
(287) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX204”).
(288) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX205”).
(289) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5b and R.sup.5c represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX206”).
(290) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX207”).
(291) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX208”).
(292) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX209”).
(293) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX210”).
(294) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX211”).
(295) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX212”).
(296) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX213”).
(297) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX214”).
(298) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX215”).
(299) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX216”).
(300) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX217”).
(301) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX218”).
(302) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX219”).
(303) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX220”).
(304) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX221”).
(305) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX222”).
(306) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX223”).
(307) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX224”).
(308) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX225”).
(309) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX226”).
(310) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX227”).
(311) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX228”).
(312) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX229”).
(313) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX230”).
(314) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX231”).
(315) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX232”).
(316) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX233”).
(317) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX234”).
(318) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX235”).
(319) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX236”).
(320) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX237”).
(321) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX238”).
(322) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 and R.sup.5b represent a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX239”).
(323) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX240”).
(324) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX241”).
(325) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 and R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX242”).
(326) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX243”).
(327) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX244”).
(328) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX245”).
(329) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX246”).
(330) A present compound wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX247”).
(331) A present compound wherein A.sup.2 represents a nitrogen represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX248”).
(332) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX249”).
(333) A present compound wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX250”).
(334) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX251”).
(335) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX252”).
(336) A present compound wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX253”).
(337) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a hydrogen atom, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX254”).
(338) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a cyclopropyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX255”).
(339) A present compound wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, R.sup.5b represents a 4-fluorophenyl group, and T represents any one substituent indicated in [Table 1A] to [Table 6A] (hereinafter, referred to as “Compound class SX256”).
(340) A compound represented by formula (L-1):
(341) ##STR00086##
(hereinafter, referred to as “Compound (L-1)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX257”).
[Table 3]
(342) TABLE-US-00007 TABLE 7A Et Pr i-Pr 1-CN-c-Pr C(O)Me C(O)OEt C(O)NHEt C(O)NHCH.sub.2CHMe.sub.2 C(O)NMe.sub.2 Ph 3-F—Ph 3-Cl—Ph 4-Cl—Ph 3-CF.sub.3—Ph 4-CF.sub.3—Ph 3-NMe.sub.2—Ph 4-NMe.sub.2—Ph 3-CN—Ph 4-CN—Ph 4-C(O)NMe.sub.2—Ph 4-NHC(O)Me—Ph 3,4-F.sub.2—Ph 3,5-F.sub.2—Ph 2,4-F.sub.2—Ph 3,4,5-F.sub.3—Ph
(343) TABLE-US-00008 TABLE 8A 3,4-Cl.sub.2—Ph 3,5-Cl.sub.2—Ph 3,5-Cl.sub.2-4-F—Ph 3,5-(CF.sub.3).sub.2—Ph Py2 4-F—Py2 5-F—Py2 4-Cl—Py2 5-Cl—Py2 4-CF.sub.3—Py2 5-CF.sub.3—Py2 3-Me—Py2 4-Me—Py2 5-Me—Py2 6-Me—Py2 5-CN—Py2 5-OCH.sub.2CF.sub.2CF.sub.3—Py2 3,5-F.sub.2—Py2 Py3 6-CF.sub.3—Py3 5-CF.sub.3—Py3 6-F—Py3 6-Cl—Py3 Py4
[Table 4]
(344) TABLE-US-00009 TABLE 9A
(345) TABLE-US-00010 TABLE 10
(346) TABLE-US-00011 TABLE 11A
[Table 5]
(347) TABLE-US-00012 TABLE 12A
(348) TABLE-US-00013 TABLE 13A
[Table 6]
(349) TABLE-US-00014 TABLE 14A F Cl Br Me CF.sub.3 OMe Et OPr Oi—Pr NH.sub.2 NHCH.sub.2CF.sub.3 CN NHC(O)c-Pr NMeC(O)c-Pr CH═N—OH CH═N—OMe OPh O-2-F—Ph OPy2 OPy3
(350) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX258”).
(351) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX259”).
(352) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX260”).
(353) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX261”).
(354) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX262”).
(355) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX263”).
(356) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX264”).
(357) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A](hereinafter, referred to as “Compound class SX265”).
(358) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX266”).
(359) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX267”).
(360) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX268”).
(361) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX269”).
(362) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX270”).
(363) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX271”).
(364) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX272”).
(365) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX273”).
(366) The compound (L-1) wherein A.sup.2 represents a nitrogen represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX274”).
(367) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX275”).
(368) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX276”).
(369) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX277”).
(370) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX278”).
(371) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX279”).
(372) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX280”).
(373) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX281”).
(374) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX282”).
(375) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX283”).
(376) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX284”).
(377) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX285”).
(378) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX286”).
(379) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX287”).
(380) The compound (L-1) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX288”).
(381) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX289”).
(382) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX290”).
(383) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX291”).
(384) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, 0 represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX292”).
(385) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX293”).
(386) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX294”).
(387) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX295”).
(388) The compound (L-1) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX296”).
(389) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX297”).
(390) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX298”).
(391) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX299”).
(392) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX300”).
(393) The compound (L-1) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX301”).
(394) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX302”).
(395) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX303”).
(396) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX304”).
(397) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX305”).
(398) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX306”).
(399) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX307”).
(400) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX308”).
(401) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX309”).
(402) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX310”).
(403) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX311”).
(404) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX312”).
(405) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX313”).
(406) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX314”).
(407) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX315”).
(408) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX316”).
(409) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX317”).
(410) The compound (L-1) wherein A.sup.2 represents a nitrogen represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX318”).
(411) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX319”).
(412) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX320”).
(413) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX321”).
(414) The compound (L-1) wherein A.sup.2 represents a nitrogen represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX322”).
(415) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX323”).
(416) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX324”).
(417) The compound (L-1) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX325”).
(418) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX326”).
(419) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX327”).
(420) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX328”).
(421) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX329”).
(422) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX330”).
(423) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX331”).
(424) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX332”).
(425) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX333”).
(426) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX334”).
(427) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX335”).
(428) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX336”).
(429) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX337”).
(430) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX338”).
(431) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX339”).
(432) The compound (L-1) wherein A.sup.2 represents a nitrogen represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX340”).
(433) The compound (L-1) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX341”).
(434) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX342”).
(435) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX343”).
(436) The compound (L-1) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX344”).
(437) A compound represented by formula (L-2):
(438) ##STR00135##
(hereinafter, referred to as “Compound (L-2)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX345”).
(439) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX346”).
(440) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5′ represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX347”).
(441) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX348”).
(442) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX349”).
(443) The compound (L-1) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX350”).
(444) The compound (L-1) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX351”).
(445) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX352”).
(446) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX353”).
(447) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.51 represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX354”).
(448) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX355”).
(449) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX356”).
(450) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX357”).
(451) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX358”).
(452) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX359”).
(453) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX360”).
(454) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX361”).
(455) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX362”).
(456) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX363”).
(457) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX364”).
(458) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX365”).
(459) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX366”).
(460) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX367”).
(461) The compound (L-2) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX368”).
(462) The compound (L-2) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX369”).
(463) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, 0 represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX370”).
(464) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX371”).
(465) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX372”).
(466) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX373”).
(467) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX374”).
(468) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX375”).
(469) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX376”).
(470) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX377”).
(471) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX378”).
(472) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX379).
(473) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX380”).
(474) The compound (L-2) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX381”).
(475) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX382”).
(476) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX383”).
(477) The compound (L-2) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX384”).
(478) The compound (L-2) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX385”).
(479) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX386”).
(480) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX387”).
(481) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX388”).
(482) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX389”).
(483) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX390”).
(484) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX391”).
(485) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5A represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX392”).
(486) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX393”).
(487) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX394”).
(488) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX395”).
(489) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX396”).
(490) The compound (L-2) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX397”).
(491) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX398”).
(492) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX399”).
(493) The compound (L-2) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX400”).
(494) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX401”).
(495) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX402”).
(496) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX403”).
(497) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX404”).
(498) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX405”).
(499) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX406”).
(500) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX407”).
(501) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX408”).
(502) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX409”).
(503) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX410”).
(504) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX411”).
(505) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX412”).
(506) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX413”).
(507) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX414”).
(508) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX415”).
(509) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX416”).
(510) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX417”).
(511) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX418”).
(512) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX419”).
(513) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX420”).
(514) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX421”).
(515) The compound (L-2) wherein A.sup.2 represents a nitrogen represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX422”).
(516) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX423”).
(517) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX424”).
(518) The compound (L-2) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX425”).
(519) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX426”).
(520) The compound (L-2) wherein A3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX427”).
(521) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX428”).
(522) The compound (L-2) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX429”).
(523) The compound (L-2) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX430”).
(524) The compound (L-2) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX431”).
(525) The compound (L-2) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX432”).
(526) A compound represented by formula (L-3):
(527) ##STR00136##
(hereinafter, referred to as “Compound (L-3)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX433”).
(528) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX434”).
(529) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX435”).
(530) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX436”).
(531) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX437”).
(532) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX438”).
(533) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX439”).
(534) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX440”).
(535) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX441”).
(536) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX442”).
(537) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX443”).
(538) The compound (L-2) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX444”).
(539) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX445”).
(540) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX446”).
(541) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX447”).
(542) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX448”).
(543) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX449”).
(544) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX450”).
(545) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX451”).
(546) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX452”).
(547) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX453”).
(548) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX454”).
(549) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX455”).
(550) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX456”).
(551) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX457”).
(552) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX458”).
(553) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX459”).
(554) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX460”).
(555) The compound (L-3) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX461”).
(556) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX462”).
(557) The compound (L-3) wherein A3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX463”).
(558) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX464”).
(559) The compound (L-3) wherein A.sup.2, A3 and A4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX465”).
(560) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX466”).
(561) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX467).
(562) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX468”).
(563) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX469”).
(564) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX470”).
(565) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX471”).
(566) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX472”).
(567) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX473”).
(568) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5 represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX474”).
(569) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5 represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX475”).
(570) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX476”).
(571) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX477”).
(572) The compound (L-3) wherein A.sup.2 represents a nitrogen represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX478”).
(573) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX479”).
(574) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX480”).
(575) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX481”).
(576) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX482”).
(577) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX483”).
(578) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX484”).
(579) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX485”).
(580) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX486”).
(581) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX487”).
(582) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX488”).
(583) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX489”).
(584) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX490”).
(585) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX491”).
(586) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX492”).
(587) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX493”).
(588) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX494”).
(589) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX495”).
(590) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX496”).
(591) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX497”).
(592) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX498”).
(593) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX499”).
(594) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX500”).
(595) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX501”).
(596) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX502”).
(597) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX503”).
(598) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX504”).
(599) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX505”).
(600) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX506”).
(601) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX507”).
(602) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, 0 represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX508”).
(603) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX509”).
(604) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX510”).
(605) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX511”).
(606) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX512”).
(607) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX513”).
(608) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX514”).
(609) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX515”).
(610) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX516”).
(611) The compound (L-3) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX517”).
(612) The compound (L-3) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX518”).
(613) The compound (L-3) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX519”).
(614) The compound (L-3) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX520”).
(615) A compound represented by formula (L-4):
(616) ##STR00137##
(hereinafter, referred to as “Compound (L-4)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX521”).
(617) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX522”).
(618) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX523”).
(619) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX524”).
(620) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX525”).
(621) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX526”).
(622) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX527”).
(623) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX528”).
(624) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX529”).
(625) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX530”).
(626) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX531”).
(627) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX532”).
(628) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX533”).
(629) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX534”).
(630) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX535”).
(631) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX536”).
(632) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX537”).
(633) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX538”).
(634) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX539”).
(635) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX540”).
(636) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX541”).
(637) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX542”).
(638) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX543”).
(639) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX544”).
(640) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX545”).
(641) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX546”).
(642) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX547”).
(643) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX548”).
(644) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX549”).
(645) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX550”).
(646) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX551”).
(647) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX552”).
(648) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX553”).
(649) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX554”).
(650) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX555).
(651) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX556”).
(652) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX557”).
(653) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX558”).
(654) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX559”).
(655) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX560”).
(656) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX561”).
(657) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX562”).
(658) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX563”).
(659) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX564”).
(660) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX565”).
(661) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX566”).
(662) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX567”).
(663) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX568”).
(664) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX569”).
(665) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX570”).
(666) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX571”).
(667) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX572”).
(668) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX573”).
(669) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX574”).
(670) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX575”).
(671) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX576”).
(672) The compound (L-4) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX577”).
(673) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX578”).
(674) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A2 and A4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX579”).
(675) The compound (L-4) wherein A4 represents a nitrogen atom, A2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX580”).
(676) The compound (L-4) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX581”).
(677) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX582”).
(678) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX583”).
(679) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX584”).
(680) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX585”).
(681) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX586”).
(682) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX587”).
(683) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX588”).
(684) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX589”).
(685) The compound (L-4) wherein A.sup.2 represents a nitrogen represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX590”).
(686) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX591”).
(687) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX592”).
(688) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX593”).
(689) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX594”).
(690) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX595”).
(691) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX596”).
(692) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX597”).
(693) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX598”).
(694) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX599”).
(695) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX600”).
(696) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX601”).
(697) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX602”).
(698) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX603”).
(699) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX604”).
(700) The compound (L-4) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX605”).
(701) The compound (L-4) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX606”).
(702) The compound (L-4) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX607”).
(703) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX608”).
(704) A compound represented by formula (L-5):
(705) ##STR00138##
(hereinafter, referred to as “Compound (L-5)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX609”).
(706) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX610”).
(707) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX611”).
(708) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX612”).
(709) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX613”).
(710) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX614”).
(711) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX615”).
(712) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX616”).
(713) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX617”).
(714) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX618”).
(715) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX619”).
(716) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX620”).
(717) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX621”).
(718) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX622”).
(719) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX623”).
(720) The compound (L-5) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX624”).
(721) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX625”).
(722) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX626”).
(723) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX627”).
(724) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX628”).
(725) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX629”).
(726) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX630”).
(727) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX631”).
(728) The compound (L-4) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX632”).
(729) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX633”).
(730) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX634”).
(731) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX635”).
(732) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX636”).
(733) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX637”).
(734) The compound (L-5) wherein A.sup.2 represents a nitrogen represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX638”).
(735) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX639”).
(736) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX640”).
(737) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX641”).
(738) The compound (L-5) wherein A.sup.2 represents a nitrogen represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX642”).
(739) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX643).
(740) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX644”).
(741) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX645”).
(742) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX646”).
(743) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX647”).
(744) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX648”).
(745) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX649”).
(746) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX650”).
(747) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX651”).
(748) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX652”).
(749) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX653”).
(750) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX654”).
(751) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX655”).
(752) The compound (L-5) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX656”).
(753) The compound (L-5) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX657”).
(754) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX658”).
(755) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX659”).
(756) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX660”).
(757) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX661”).
(758) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX662”).
(759) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX663”).
(760) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX664”).
(761) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX665”).
(762) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX666”).
(763) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX667”).
(764) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX668”).
(765) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX669”).
(766) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX670”).
(767) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX671”).
(768) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX672”).
(769) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX673”).
(770) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX674”).
(771) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX675”).
(772) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX676”).
(773) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX677”).
(774) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX678”).
(775) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX679”).
(776) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX680”).
(777) The compound (L-5) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX681”).
(778) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX682”).
(779) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX683”).
(780) The compound (L-5) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table-14A] (hereinafter, referred to as “Compound class SX684”).
(781) The compound (L-5) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX685”).
(782) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX686”).
(783) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX687”).
(784) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX688”).
(785) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX689”).
(786) The compound (L-5) wherein A.sup.2 represents a nitrogen represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX690”).
(787) The compound (L-5) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX691”).
(788) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX692”).
(789) The compound (L-5) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX693”).
(790) The compound (L-5) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX694”).
(791) The compound (L-5) wherein A3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX695”).
(792) The compound (L-5) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX696”).
(793) A compound represented by formula (L-6):
(794) ##STR00139##
(hereinafter, referred to as “Compound (L-6)”) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX697”).
(795) The compound (L-6) wherein A.sup.2 represents a nitrogen represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX698”).
(796) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX699”).
(797) The compound (L-6) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX700”).
(798) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX701”).
(799) The compound (L-6) wherein A.sup.2 represents a nitrogen represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX702”).
(800) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX703”).
(801) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX704”).
(802) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX705”).
(803) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX706”).
(804) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX707”).
(805) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX708”).
(806) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX709”).
(807) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX710”).
(808) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX711”).
(809) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX712”).
(810) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX713”).
(811) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX714”).
(812) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX715”).
(813) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX716”).
(814) The compound (L-6) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX717”).
(815) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX718”).
(816) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX719”).
(817) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX720”).
(818) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX721”).
(819) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX722”).
(820) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX723”).
(821) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX724”).
(822) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX725”).
(823) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX726”).
(824) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX727”).
(825) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX728”).
(826) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX729”).
(827) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX730”).
(828) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX731).
(829) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX732”).
(830) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX733”).
(831) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX734”).
(832) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX735”).
(833) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX736”).
(834) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5 represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX737”).
(835) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX738”).
(836) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX739”).
(837) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX740”).
(838) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX741”).
(839) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX742”).
(840) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX743”).
(841) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX744”).
(842) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX745”).
(843) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX746”).
(844) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX747”).
(845) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX748”).
(846) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX749”).
(847) The compound (L-6) wherein A.sup.2 represents a nitrogen represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX750”).
(848) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX751”).
(849) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX752”).
(850) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX753”).
(851) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX754”).
(852) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX755”).
(853) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX756”).
(854) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX757”).
(855) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX758”).
(856) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX759”).
(857) The compound (L-6) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX760”).
(858) The compound (L-6) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX761”).
(859) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX762”).
(860) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX763”).
(861) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX764”).
(862) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX765”).
(863) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX766”).
(864) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX767”).
(865) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX768”).
(866) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX769”).
(867) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX770”).
(868) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX771”).
(869) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX772”).
(870) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX773”).
(871) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX774”).
(872) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX775”).
(873) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX776”).
(874) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX777”).
(875) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX778”).
(876) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX779”).
(877) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX780”).
(878) The compound (L-6) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX781”).
(879) The compound (L-6) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX782”).
(880) The compound (L-6) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX783”).
(881) The compound (L-6) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX784”).
(882) A compound represented by formula (L-7):
(883) ##STR00140##
(hereinafter, referred to as “Compound (L-7)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX785”).
(884) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX786”).
(885) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX787”).
(886) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX788”).
(887) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX789”).
(888) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX790”).
(889) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX791”).
(890) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX792”).
(891) The compound (L-7) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX793”).
(892) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX794”).
(893) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX795”).
(894) The compound (L-7) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX796”).
(895) The compound (L-7) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX797”).
(896) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX798”).
(897) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX799”).
(898) The compound (L-7) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX800”).
(899) The compound (L-7) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX801”).
(900) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX802”).
(901) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX803”).
(902) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX804”).
(903) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX805”).
(904) The compound (L-7) wherein A.sup.2 represents a nitrogen represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX806”).
(905) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX807”).
(906) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX808”).
(907) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX809”).
(908) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX810”).
(909) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX811”).
(910) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX812”).
(911) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX813”).
(912) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX813”).
(913) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX815”).
(914) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX816”).
(915) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX817”).
(916) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX818”).
(917) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX819).
(918) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX820”).
(919) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX821”).
(920) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX822”).
(921) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX823”).
(922) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX824”).
(923) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX825”).
(924) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX826”).
(925) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX827”).
(926) The compound (L-7) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX828”).
(927) The compound (L-7) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX829”).
(928) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX830”).
(929) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX831”).
(930) The compound (L-7) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX832”).
(931) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX833”).
(932) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX834”).
(933) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX835”).
(934) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX836”).
(935) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX837”).
(936) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX838”).
(937) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX839”).
(938) The compound (L-7) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX840”).
(939) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX841”).
(940) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX842”).
(941) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX843”).
(942) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX844”).
(943) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX845”).
(944) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX846”).
(945) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX847”).
(946) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX848”).
(947) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX849”).
(948) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX850”).
(949) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX851”).
(950) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX852”).
(951) The compound (L-7) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX853”).
(952) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX854”).
(953) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX855”).
(954) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX856”).
(955) The compound (L-7) wherein A.sup.2, A3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX857”).
(956) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX858”).
(957) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX859”).
(958) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX860”).
(959) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX861”).
(960) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX862”).
(961) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX863”).
(962) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX864”).
(963) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX865”).
(964) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX866”).
(965) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX867”).
(966) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX868”).
(967) The compound (L-7) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX869”).
(968) The compound (L-7) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX870”).
(969) The compound (L-7) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX871”).
(970) The compound (L-7) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX872”).
(971) A compound represented by formula (L-8):
(972) ##STR00141##
(hereinafter, referred to as “Compound (L-8)”) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX873”).
(973) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX874”).
(974) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX875”).
(975) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q10, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX876”).
(976) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.54 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX877”).
(977) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX878”).
(978) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX879”).
(979) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q11, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX880”).
(980) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX881”).
(981) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX882”).
(982) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX883”).
(983) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 and R.sup.5a represent a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX884”).
(984) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX885”).
(985) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX886”).
(986) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX887”).
(987) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q12, R.sup.3 represents a methyl group, R.sup.5a represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX888”).
(988) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX889”).
(989) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX890”).
(990) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX891”).
(991) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A3 represent CH, Q represents a group represented by Q15, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX892”).
(992) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX893”).
(993) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX894”).
(994) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX895”).
(995) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q16, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX896”).
(996) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX897”).
(997) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX898”).
(998) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX899”).
(999) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a hydrogen atom, R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX900”).
(1000) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX901”).
(1001) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX902”).
(1002) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX903”).
(1003) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q17, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX904”).
(1004) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX905”).
(1005) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX906”).
(1006) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX907).
(1007) The compound (L-8) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q18, and R.sup.5a and R.sup.5c represent a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX908”).
(1008) The compound (L-8) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX909”).
(1009) The compound (L-8) wherein A.sup.2 represents a nitrogen represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX910”).
(1010) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX911”).
(1011) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a hydrogen atom, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX912”).
(1012) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX913”).
(1013) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX914”).
(1014) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX915”).
(1015) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.3 represents a methyl group, and R.sup.5a represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX916”).
(1016) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX917”).
(1017) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX918”).
(1018) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX919”).
(1019) The compound (L-8) wherein A4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q20, R.sup.5a represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX920”).
(1020) The compound (L-8) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX921”).
(1021) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX922”).
(1022) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX923”).
(1023) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q21, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX924”).
(1024) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX925”).
(1025) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX926”).
(1026) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q22, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX927”).
(1027) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q22, R.sup.5c represents a hydrogen atom, and R.sup.3 represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX928”).
(1028) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX929”).
(1029) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX930”).
(1030) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX931”).
(1031) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q23, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX932”).
(1032) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX933”).
(1033) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX934”).
(1034) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX935”).
(1035) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q24, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX936”).
(1036) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 9A] (hereinafter, referred to as “Compound class SX937”).
(1037) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX938”).
(1038) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX939”).
(1039) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 and R.sup.5c represent a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX940”).
(1040) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX941”).
(1041) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX942”).
(1042) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX943”).
(1043) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q25, R.sup.3 represents a methyl group, R.sup.5c represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX944”).
(1044) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX945”).
(1045) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX946”).
(1046) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX947”).
(1047) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q26, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX948”).
(1048) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX949”).
(1049) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX950”).
(1050) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX951”).
(1051) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q27, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX952”).
(1052) The compound (L-8) wherein A.sup.2, A.sup.3 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX953”).
(1053) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX954”).
(1054) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX955”).
(1055) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a hydrogen atom, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX956”).
(1056) The compound (L-8) wherein A.sup.2, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX957”).
(1057) The compound (L-8) wherein A.sup.2 represents a nitrogen atom, A.sup.3 and A4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX958”).
(1058) The compound (L-8) wherein A.sup.3 represents a nitrogen atom, A.sup.2 and A.sup.4 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX959”).
(1059) The compound (L-8) wherein A.sup.4 represents a nitrogen atom, A.sup.2 and A.sup.3 represent CH, Q represents a group represented by Q28, R.sup.3 represents a methyl group, and R.sup.5b represents any one substituent indicated in [Table 7A] to [Table 14A] (hereinafter, referred to as “Compound class SX960”).
(1060) Next, the Formulation examples of the present compound are shown below. The “parts” represents “part by weight”. Further, the present compound S represents the compounds described as the compound groups SX1 to SX960.
Formulation Example 1
(1061) Into a mixture of 10 parts of any one of the present compounds S, 35 parts of xylene, and 35 parts of DMF, and then 14 parts of polyoxyethylene styryl phenyl ether and 6 parts of calcium dodecylbenzene sulfonate are added, followed by mixing them to obtain each formulation.
Formulation Example 2
(1062) Four (4) parts of sodium lauryl sulfate, 2 parts of calcium lignin sulfonate, 20 parts of wet process silica, and 54 parts of diatomaceous earth are mixed, and further 20 parts of any one of the present compounds S is added thereto, followed by mixing them to obtain each formulation.
Formulation Example 3
(1063) To 2 parts of any one of the present compounds S, 1 part of wet process silica, 2 parts of calcium lignin sulfonate, 30 parts of bentonite, and 65 parts of kaolin clay are added, followed by mixing them. To the mixtures is then added an appropriate amount of water, and the mixtures are further stirred, granulated with a granulator, and forced-air dried to obtain each formulation.
Formulation Example 4
(1064) Into an appropriate amount of acetone, 1 part of any one of the present compounds S is mixed, and then 5 parts of wet process silica, 0.3 parts of isopropyl acid phosphate, and 93.7 parts of kaolin clay are added, following by mixing them with stirring thoroughly and removal of acetone from the mixture by evaporation to obtain each formulation.
Formulation Example 5
(1065) A mixture of 35 parts of polyoxyethylene alkyl ether sulfate ammonium salt and wet process silica (weight ratio of 1:1), 20 parts of any one of the present compounds S, and 45 parts of water are enough mixed to obtain each formulation.
Formulation Example 6
(1066) Into a mixture of 5 parts of xylene and 5 parts of trichloroethane, 0.1 parts of any one of the present compounds S are mixed, and the resulting mixture is then mixed with 89.9 parts of kerosene to obtain each solution.
Formulation Example 7
(1067) Into 0.5 ml of acetone, 10 mg of any one of the present compounds S is mixed, and the solution is added dropwise to 5 g of a solid feed powder for an animal (solid feed powder for rearing and breeding CE-2, manufactured by CLEA Japan, Inc.), followed by mixing the resulting mixtures uniformly, and then by drying them by evaporation of acetone to obtain each poison bait.
Formulation Example 8
(1068) Into an aerosol can, 0.1 parts of any one of the present compounds S and 49.9 parts of Neothiozole (manufactured by Chuo Kasei Co., Ltd.) are placed. After mounting an aerosol valve, 25 parts of dimethyl ether and 25 parts of LPG are filled, followed by shaking and further mounting an actuator to obtain each oily aerosol.
Formulation Example 9
(1069) A mixture of 0.6 parts of any one of the present compounds S, 0.01 parts of 2,6-di-tert-butyl-4-methylphenol, 5 parts of xylene, 3.39 parts of kerosene, and 1 part of Rheodol (registered trademark) MO-60, and 50 parts of distilled water are filled into an aerosol container, and a valve part of the container is attached. Then, 40 parts of LPG is filled therein through the valve under pressure to obtain each aqueous aerosol.
Formulation Example 10
(1070) Zero point one (0.1) g of any one of the present compounds S is mixed into 2 ml of propylene glycol, and the resulting solution is impregnated into a ceramic plate having a size of 4.0 cm×4.0 cm and a thickness of 1.2 cm to obtain each thermal fumigant.
Formulation Example 11
(1071) Five (5) parts of any one of the present compounds S, and 95 parts of ethylene-methyl methacrylate copolymer (the ratio of the methyl methacrylate in the copolymer: 10 weight %) are melted and kneaded, and the resulting kneaded product is extruded from an extrusion molding machine to obtain each rod-shaped molded product having a length of 15 cm and a diameter of 3 mm.
Formulation Example 12
(1072) Five (5) parts of any one of the present compounds S, and 95 parts of plasticized polyvinyl chloride resin are melted and kneaded, and the resulting kneaded product is extruded from an extrusion molding machine to obtain each rod-shaped molded product having a length of 15 cm and a diameter of 3 mm.
Formulation Example 13
(1073) One-hundred (100) mg of any one of the present compounds S, 68.75 mg of lactose, 237.5 mg of corn starch, 43.75 mg of microcrystalline cellulose, 18.75 mg of polyvinylpyrrolidone, 28.75 mg of sodium carboxymethyl starch, and 2.5 mg of magnesium stearate are mixed, and the resulting mixtures are compressed to an appropriate size to obtain each tablet.
Formulation Example 14
(1074) Twenty-five (25) mg of any one of the present compounds S, 60 mg of lactose, 25 mg of corn starch, 6 mg of carmellose calcium, and an appropriate amount of 5% aqueous hydroxypropyl methylcellulose solution are mixed, and the resulting mixtures are filled into a hard shell gelatin capsule or a hydroxypropyl methylcellulose capsule to obtain each capsule.
Formulation Example 15
(1075) To 100 mg of any one of the present compounds S, 500 mg of fumaric acid, 2000 mg of sodium chloride, 150 mg of methyl paraben, 50 mg of propyl paraben, 25,000 mg of granulated sugar, 13,000 mg of sorbitol (70% solution), 100 mg of Veegum (registered trademark) K (manufactured by Vanderbilt Co.), 35 mg of a perfume, and 500 mg of a coloring agent, distilled water is added so that a final volume is set to be 100 mL, followed by mixing the mixtures
Formulation Example 16
(1076) Into a mixture of 5 parts of an emulsifier, 3 parts of benzyl alcohol and 30 parts of propylene glycol, 5 parts of any one of the present compounds S is mixed, and phosphate buffer is added thereto so that a pH of the solution is set to be 6.0 to 6.5, and water is added as the rest parts to obtain each solution for oral administration.
Formulation Example 17
(1077) To a mixture of 57 parts of fractional distillated palm oil and 3 parts of polysorbate 85, 5 parts of aluminium distearate is added, and heated to disperse it. The resulting mixture is cooled to room temperature, and 25 parts of saccharin is dispersed in an oil vehicle. Ten (10) parts of any one of the present compounds S is divided thereto to obtain each paste for oral administration.
Formulation Example 18
(1078) Five (5) parts of any one of the present compounds S is mixed with 95 parts of limestone filler, followed by a wet-granulation of the resulting mixture to obtain each granule for oral administration.
Formulation Example 19
(1079) Into 80 parts of diethylene glycol monoethyl ether, 5 parts of any one of the present compounds S is mixed, and 15 parts of propylene carbonate is added thereto, and the resulting mixture is mixed to obtain each spot-on solution.
Formulation Example 20
(1080) Into 70 parts of diethylene glycol monoethyl ether, 10 parts of any one of the present compounds S is mixed, and 20 parts of 2-octyldodecanol is added thereto, and the resulting mixture is mixed to obtain each pour-on solution.
Formulation Example 21
(1081) To 0.1 parts of any one of the present compounds S, 40 parts of sodium polyoxyethylene lauryl ether sulfate (25% aqueous solution), 5 parts of lauramidopropyl betaine, 5 parts of coconut fatty acid monoethanolamide, 0.5 parts of carboxy vinyl polymer, and 49.4 parts of purified water are added, and the resulting mixture is enough mixed to obtain each shampoo formulation.
Formulation Example 22
(1082) Zero point fifteen (0.15) parts of any one of the present compounds S, 95 parts of animal feed, as well as 4.85 parts of a mixture of dibasic calcium phosphate, diatomaceous earth, Aerosil (registered trademark), and carbonate (or chalk) are enough mixed to obtain each premix for animal feed.
Formulation Example 23
(1083) Seven point two (7.2) g of any one of the present compounds S, and 92.8 g of Hosco (registered trademark)S-55 are mixed at 100° C., and the resulting mixture is poured into a suppository mold, followed by performing a cooling solidification to obtain each suppository.
(1084) Next, an efficacy of the present compound on controlling harmful arthropods is shown by Test examples. The following tests were conducted at 25° C.
(1085) Test Method 1
(1086) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.
(1087) Cucumber (cucumber sativus) seedling (on the developmental stage of the second true leaf) is planted in a cup, and approximately 30 cotton aphids (Aphis gossypii) (all stages of life) are released onto the seedling. After one day, the diluted solutions are sprayed into the seedling at a ratio of 10 mL/seedling. After 5 days, the number of the surviving insects is examined and the controlling value is calculated by the following equation.
Controlling value (%)=(1−(Cb×Tai)/(Cai×Tb))×100
wherein the symbols in the equation represent the following descriptions.
(1088) Cb: Number of the test insects in untreated group;
(1089) Cai: Number of the surviving insects at the time of the examination in untreated group;
(1090) Tb: Number of the test insects in treated group;
(1091) Tai: Number of the surviving insects at the time of the examination in treated group;
(1092) Here the “untreated group” represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.
Test Example 1
(1093) The test was conducted according to the Test method 1 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value. Present compound Nos: 12 and 13
(1094) Test Method 2
(1095) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.
(1096) Cucumber (cucumber sativus) seedling (on the developmental stage of the second true leaf) is planted in a cup, and the diluted solutions are drenched to the foot of the seedling at a ratio of 5 mL/seedling. After 7 days, approximately 30 cotton aphids (Aphis gossypii) (all stages of life) are released onto the leaf of the seedling. After 6 days, the number of the surviving insects is examined and the controlling value is calculated by the following equation.
Controlling value (%)={1−(Cb×Tai)/(Cai×Tb)}×100
wherein the symbols in the equation represent the following descriptions.
(1097) Cb: Number of the test insects in untreated group;
(1098) Cai: Number of the surviving insects at the time of the examination in untreated group;
(1099) Tb: Number of the test insects in treated group;
(1100) Tai: Number of the surviving insects at the time of the examination in treated group;
(1101) Here the “untreated group” represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.
(1102) Test Method 3
(1103) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.
(1104) Cabbage (Brassicae oleracea) seedling (on the developmental stage of the second to third true leaf) is planted in a cup, and the diluted solutions are sprayed into the seedling at a ratio of 20 mL/seedling. Thereafter, the stem and leaf thereof is cut out and then is installed into a cup that is covered with filter paper on the bed of the cup. Five (5) tobacco cutworms (Spodoptera litura) at the second instar larval stage are released into the cup. After 5 days, the number of the surviving insects is counted, and the mortality of insects is calculated by the following equation.
Mortality (%)=(1−Number of surviving insects/5)×100
Test Example 3-1
(1105) The test was conducted according to the Test method 3 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality of insects. Present compound Nos: 11 and 15
Test Example 3-2
(1106) The test was conducted according to the Test method 3 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality of insects. Present compound Nos: 2 and 11
(1107) Test Method 4
(1108) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.
(1109) Cabbage (Brassicae oleracea) seedling (on the developmental stage of the second to third true leaf) is planted in a cup, and the diluted solutions are sprayed into the seedling at a ratio of 20 mL/seedling. Thereafter, the stem and leaf thereof is cut out and then is installed into a cup that is covered with filter paper on the bed of the cup. Five (5) diamondback moth (Plutella xylostella) at the second instar larval stage are released into the cup. After 5 days, the number of the surviving insects is counted, and the mortality of insects is calculated by the following equation.
Mortality (%)=(1−Number of surviving insects/5)×100
Test Example 4-1
(1110) The test was conducted according to the Test method 4 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality of insects. Present compound Nos: 5, 15, and 16
Test Example 4-2
(1111) The test was conducted according to the Test method 4 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality of insects. Present compound Nos: 2, 5, and 16
(1112) Test Method 5
(1113) Each 1 mg of the test compounds is dissolved into 50 L of a mixed solution of polyoxyethylene sorbitan mono-cocoate and acetone (polyoxyethylene sorbitan mono-cocoate:acetone=5:95 (v/v ratio)). Thereto is added water containing 0.03% by volume of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.
(1114) A young entire seedling of Corns (Zea mays) is immersed into the diluted solution for 30 seconds. Thereafter, each two grains of the seedlings are installed in a plastic petri dish (90 mm radius), and 10 Western corn rootworms (Diabrotica virgifera virgifera) at the second instar larval stage are released into the dish. After 5 days, the number of the dead insects is counted, and the mortality of insects is calculated by the following equation.
Mortality (%)=(Number of dead insects/10)×100
Test Example 5
(1115) The test was conducted according to the Test method 5 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality of insects. Present compound Nos: 13 and 15
(1116) Test Method 6
(1117) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.
(1118) A filter paper having a diameter of 5.5 cm in diameter is spread on the bottom of the cup, and then 0.7 ml of the diluted solutions are added dropwise to the filter paper and 30 mg of sucrose is uniformly placed on the filter paper as a bait. Ten (10) housefly (Musca domestica) female adults are released into the cup, and the cup is then covered with the lid. After 24 hours, the number of the dead insects is counted, and the mortality of insects is calculated by the following equation.
Mortality (%)=(Number of dead insects/Number of tested insects)×100
Test Method 7
(1119) Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.
(1120) A filter paper having a diameter of 5.5 cm is spread on the bottom of the cup, and then 0.7 ml of the diluted solutions are added dropwise to the filter paper and 30 mg of sucrose is uniformly placed on the filter paper as a bait. Two (2) German cockroach (Blattella germanica) male adults are released into the cup, and the cup is covered with the lid. After 6 days, the number of the dead insects is counted, and the mortality of insects is calculated by the following equation.
Mortality (%)=(Number of dead insects/Number of tested insects)×100
Test Method 8
(1121) Each 1 mg of the present compounds is dissolved into 10 μL of a mixed solution of xylene, DMF, and a surfactant (xylene:DMF:surfactant=4:4:1 (v/v ratio)). Thereto is added water containing 0.02% by volume of a spreader to prepare diluted solution A containing a prescribed concentration of the present compound.
(1122) Each 1 mg of the present ingredients is dissolved into 10 μL of a mixed solution of xylene, DMF, and a surfactant (xylene:DMF:surfactant=4:4:1 (v/v ratio)). Thereto is added water containing 0.02% by volume of a spreader to prepare diluted solution B containing a prescribed concentration of the present ingredient?
(1123) The diluted solution A is mixed with the diluted solution B to prepare diluted solution C.
(1124) Leaf discs of Cucumber (cucumber sativus) cotyledon (length 1.5 cm) are placed in each well of 24-well microplate. Two (2) apterous adults and 8 larvae of cotton aphids (Aphis gossypii) per one well are released and the diluted solution C is sprayed at 20 μL per one well. The group is defined as “treated group”. A well that is sprayed with 20 μL of water containing 0.02% by volume of a spreader instead of the diluted solution C is defined as “untreated group”.
(1125) After drying the diluted solution C, the upper microplate is covered with a film sheet. After 5 days, the number of the surviving insects in each well is examined.
(1126) The controlling value is calculated by the following equation.
Controlling value (%)={1−(Tai)/(Cai)}×100
wherein the symbols in the equation represent the following descriptions.
(1127) Cai: Number of the surviving insects at the time of the examination in untreated group;
(1128) Tai: Number of the surviving insects at the time of the examination in treated group.
(1129) Specific diluted solutions C, which can confirm their effect according to the Test method 8, are described in the following 1) to 5).
(1130) 1) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 200 ppm and a concentration of the present ingredient is 2000 ppm. In List A, Comp X represents any compound selected from the present compounds 1 to 16.
List A:
Comp X+Clothianidin; Comp X+thiamethoxam; Comp X+imidacloprid; Comp X+thiacloprid; Comp x+flupyradifurone; Comp X+sulfoxaflor; Comp X+triflumezopyrim; Comp X+dicloromezotiaz; Comp X+beta-cyfluthrin; Comp X+tefluthrin; Comp X+fipronil; Comp X+chlorantraniliprole; Comp X+cyantraniliprole; Comp X+tetraniliprole; Comp X+thiodicarb; Comp X+carbofuran; Comp X+fluxametamide; Comp X+afoxolaner; Comp X+fluralaner; Comp X+broflanilide; Comp X+abamectin; Comp X+fluopyram; Comp X+fluensulfone; Comp X+fluazaindolizine; Comp X+tioxazafen; Comp X+flupyrimin; Comp X+Mycorrhizal Fungi; Comp X+Bradyrhizobium japonicum TA-11; Comp X+Bacillus firmus; Comp X+Bacillus firmus I-1582; Comp X+Bacillus amyloliquefaciens; Comp X+Bacillus amyloliquefaciens FZB42; Comp X+Pasteuria nishizawae; Comp X+Pasteuria nishizawae Pn1; Comp X+Pasteuria penetrans; Comp X+tebuconazole; Comp X+prothioconazole; Comp X+metconazole; Comp X+ipconazole; Comp X+triticonazole; Comp X+difenoconazole; Comp X+imazalil; Comp X+triadimenol; Comp X+tetraconazole; Comp X+flutriafol; Comp X+mandestrobin; Comp X+azoxystrobin; Comp X+pyraclostrobin; Comp X+trifloxystrobin; Comp X+fluoxastrobin; Comp X+picoxystrobin; Comp X+fenamidone; Comp X+metalaxyl; Comp X+metalaxyl-M; Comp X+fludioxonil; Comp X+sedaxane; Comp X+penflufen; Comp X+fluxapyroxad; Comp X+benzovindiflupyr; Comp X+boscalid; Comp X+carboxin; Comp X+penthiopyrad; Comp X+flutolanil; Comp X+captan; Comp X+thiram; Comp X+tolclofos-methyl; Comp X+thiabendazole; Comp X+ethaboxam; Comp X+mancozeb; Comp X+picarbutrazox; Comp X+oxathiapiprolin; Comp X+silthiofam; Comp X+inpyrfluxam.
2) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 200 ppm, and a concentration of the present ingredient is 200 ppm.
3) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 50 ppm.
4) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 5 ppm.
5) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 0.5 ppm.
INDUSTRIAL APPLICABILITY
(1131) The present compound shows an excellent control effect against a harmful arthropod.