METHOD FOR PROVIDING INFORMATION ON THERAPEUTIC REACTION OF CANCER IMMUNOTHERAPY AND KIT USING SAME
20210325394 · 2021-10-21
Assignee
- INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (Seoul, KR)
- REPUBLIC OF KOREA (MINISTER OF FOOD AND DRUG SAFETY) (Chungcheongbuk-Do, KR)
Inventors
- Sang Jun HA (Seoul, KR)
- Hye Ryun KIM (Seoul, KR)
- Hyo Sup SHIM (Seoul, KR)
- Bo Ryeong LEE (Seoul, KR)
- Jung Yeon YI (Sejong, KR)
- Dae Hee HWANG (Daegu, KR)
Cpc classification
G01N33/74
PHYSICS
International classification
Abstract
Provided in the present disclosure are a method for providing information on a therapeutic reaction of cancer immunotherapy and a kit using same for providing information, the method comprising the steps of: measuring respective expression levels of PD-L1 and PVR in a biological sample isolated from a subject; and evaluating the therapeutic reaction of cancer immunotherapy for the subject on the basis of the measured expression levels of PD-L1 and PVR.
Claims
1. A method for providing information on a therapeutic response to a cancer immunotherapy, the method comprising: measuring expression levels of PD-L1 and PVR, respectively, for a biological sample isolated from a subject; and evaluating the therapeutic response to the cancer immunotherapy for the subject, based on the measured expression levels of PD-L1 and PVR.
2. The method of claim 1, wherein the subject is a subject suspected of non-small lung cancer, wherein the biological sample includes at least one selected from a group consisting of tumor tissue, blood, serum, and plasma, and is isolated from the subject before or after the cancer immunotherapy is performed.
3. The method of claim 1, wherein the evaluating of the therapeutic response to the cancer immunotherapy includes: when the measured expression level of each of the PD-L1 and PVR is greater than or equal to a predetermined level, determining each of expressions of PD-L1 and PVR as positive and when the measured expression level of each of the PD-L1 and PVR is lower than the predetermined level, determining each of expressions of PD-L1 and PVR as negative; and evaluating the therapeutic response to the cancer immunotherapy, based on whether the expressions of PD-L1 and PVR are negative or positive, wherein the cancer immunotherapy includes one therapy selected from a group consisting of anti-PD-1 therapy, anti-TIGIT therapy, and anti-PD-1/anti-TIGIT combination therapy.
4. The method of claim 3, wherein the evaluating of the therapeutic response to the cancer immunotherapy includes: evaluating that a subject having the PD-L1 expression positive and the PVR expression negative has the therapeutic response to the anti-PD-1 therapy higher than the therapeutic response to the anti-PD-1 therapy of one of a subject having the PD-L1 expression positive and the PVR expression positive, a subject having the PD-L1 expression negative and the PVR expression negative, and a subject having the PD-L1 expression negative and the PVR expression positive.
5. The method of claim 3, wherein the evaluating of the therapeutic response to the cancer immunotherapy includes: evaluating that a subject having the PD-L1 expression negative and the PVR expression positive has the therapeutic response to the anti-TIGIT therapy or the anti-PD-1/anti-TIGIT combination therapy higher than the therapeutic response to the anti-PD-1 therapy.
6. The method of claim 3, wherein the predetermined levels for the PD-L1 and the PVR are TPS (Tumor Proportion Score) 10% and TPS 60%, respectively.
7. The method of claim 1, wherein the cancer immunotherapy includes at least one therapy selected from a group consisting of anti-CTLA-4 therapy, anti-PD-1 therapy, anti-CD28 therapy, anti-KIR therapy, anti-TCR therapy, anti-LAG-3 therapy, anti-TIM-3 therapy, anti-TIGIT therapy, anti-A2aR therapy, anti-ICOS therapy, anti-OX40 therapy, anti-4-1BB therapy and anti-GITR therapy.
8. A method for providing information on a therapeutic response to a cancer immunotherapy, the method comprising: a first step of respectively measuring expression levels of PVR for biological samples isolated from a subject before and after the cancer immunotherapy is performed; and a second step of evaluating the therapeutic response to the cancer immunotherapy for the subject, based on the expression levels of PVR.
9. The method of claim 8, wherein the cancer immunotherapy is anti-PD-1 therapy, wherein the evaluating of the therapeutic response to the cancer immunotherapy for the subject includes: evaluating, that a subject whose expression level of PVR after the anti-PD-1 is performed is higher than a level thereof before the anti-PD-1 is performed, has the therapeutic response to the anti-PD-1 therapy lower than the therapeutic response to the anti-PD-1 therapy of a subject whose expression level of PVR after the anti-PD-1 is performed is lower than or equal to a level thereof before the anti-PD-1 is performed.
10. A kit for providing information on a therapeutic response to a cancer immunotherapy, the kit containing formulations configured to measure expression levels of PD-L1 and PVR, respectively, for a biological sample isolated from a subject.
11. The kit of claim 10, wherein the kit is configured to present a positive or negative therapeutic response to the cancer immunotherapy based on a predetermined expression level of each of the PD-L1 and PVR, wherein the cancer immunotherapy includes one selected from a group consisting of anti-PD-1 therapy, anti-TIGIT therapy, and anti-PD-1; anti-TIGIT combination therapy.
12. The kit of claim 11, wherein the kit is further configured to present the positive therapeutic response to the anti-PD-1 therapy when the subject has the expression level of PD-L1 higher than or equal to the predetermined expression level and the expression level of PVR lower than the predetermined expression level.
13. The kit of claim 11, wherein the kit is further configured to present the negative therapeutic response to the anti-PD-1 therapy, or the positive therapeutic response to the anti-TIGIT therapy or the anti-PD-1/anti-TIGIT combination therapy when the subject has the expression level of PD-L1 lower than the predetermined expression level and the expression level of PVR greater than or equal to the predetermined expression level.
14. The kit of claim 11, wherein the predetermined expression level is in a range of an expression rate of 1% to 10% for each of the PD-L1 and PVR.
15. The kit of claim 10, wherein the subject is a subject suspected of non-small lung cancer, wherein the biological sample includes at least one selected from a group consisting of tumor tissue, blood, serum, and plasma and is isolated from the subject before or after the cancer immunotherapy is performed.
16. The kit of claim 10, wherein the cancer immunotherapy includes at least one therapy selected from a group consisting of anti-CTLA-4 therapy, anti-PD-1 therapy, anti-CD28 therapy, anti-KIR therapy, anti-TCR therapy, anti-LAG-3 therapy, anti-TIM-3 therapy, anti-TIGIT therapy, anti-A2aR therapy, anti-ICOS therapy, anti-OX40 therapy, anti-4-1BB therapy and anti-GITR therapy.
Description
BRIEF DESCRIPTION OF THE DRAWINGS
[0042]
[0043]
[0044]
[0045]
[0046]
BEST MODES FOR CARRYING OUT THE INVENTION
[0047] Advantages and features of the present disclosure, and a method of achieving them will become apparent with reference to the embodiments described later in detail together with the accompanying drawings. However, the present disclosure is not limited to the embodiments disclosed below, but will be implemented in various different forms. Only these embodiments make the disclosure of the present disclosure complete and are provided to completely inform the scope of the disclosure to those with ordinary knowledge in the technical field to which the present disclosure belongs. The present disclosure is only defined by the scope of the claims.
[0048] Hereinafter, a procedure of a method for providing information on a therapeutic response to cancer immunotherapy according to an embodiment of the present disclosure will be described in detail with reference to
[0049]
[0050] Referring to
[0051] According to an embodiment of the present disclosure, in the step of measuring the expression level (S110), the expression levels of PD-L1 and PVR are measured for biological samples such as tumor tissue, blood, serum, or plasma isolated from a subject suspected of the non-small lung cancer.
[0052] According to an embodiment of the present disclosure, the step of evaluating the therapeutic response to cancer immunotherapy (S120) can include: when the measured expression level of each of the PD-L1 and PVR is greater than or equal to a predetermined level, determining each of expressions of PD-L1 and PVR as positive; when the measured expression level of each of the PD-L1 and PVR is lower to the predetermined level, determining each of expressions of PD-L1 and PVR as negative; and evaluating the therapeutic response to the cancer immunotherapy, based on whether the expressions of PD-L1 and PVR are negative or positive.
[0053] In this connection, the cancer immunotherapy includes one therapy selected from a group consisting of anti-PD-1 therapy, anti-TIGIT therapy, and anti-PD-1/anti-TIGIT combination therapy. However, the disclosure is not limited thereto. For example, the cancer immunotherapy can include at least one therapy selected from the group consisting of anti-CTLA-4 therapy, anti-CD28 therapy, anti-KIR therapy, anti-TCR therapy, anti-LAG-3 therapy, anti-TIM-3 therapy, anti-A2aR therapy, anti-ICOS therapy, anti-OX40 therapy, anti-4-1BB therapy, and anti-GITR therapy.
[0054] According to another embodiment of the present disclosure, the step of evaluating the therapeutic response to cancer immunotherapy (S120) can include evaluating that a subject having the PD-L1 expression positive and the PVR expression negative has the therapeutic response to anti-PD-1 therapy higher than the therapeutic response to anti-PD-1 therapy of one of a subject having the PD-L1 expression positive and the PVR expression positive, a subject having the PD-L1 expression negative and the PVR expression negative, and a subject having the PD-L1 expression negative and the PVR expression positive.
[0055] According to the above procedure, the method tier providing information on a therapeutic response according to an embodiment of the present disclosure can measure the levels of various markers, and thus can provide information to allow a therapeutic response to the cancer immunotherapy for a subject, particularly, a therapeutic response to anti-PD-1 to be early predicted.
EXAMPLE 1
Biomarker Setup for Early Prediction of Therapeutic Response to PD-1 Blockade
[0056] Hereinafter, with reference to
[0057]
[0058] Referring to
[0059] Referring to (a), (b), and (c) in
[0060] Based on a result of Example 1 above, PVR, or PD-L1 and PVR can be used as biomarkers for prediction of a therapeutic response in a method for providing information about a therapeutic response according to various embodiments of the present disclosure.
EXAMPLE 2
Early Prediction of Therapeutic Response to PD-1 Blockade Based on PD-L1 and PVR Expression Patterns for Non-Small Lung Cancer Patients
[0061] Hereinafter, an evaluation result of the therapeutic response prediction to the anti-PD-1 therapy according to the expression patterns of PD-L1 and PVR in the tumor tissue of anon-small lung cancer patient will be described with reference to
[0062]
[0063] In the following experiment, 119 patients having recurrent/metastatic non-small lung cancer over the age of 20 as confirmed, for which previous platinum-based chemotherapy failed, and who underwent the PD-1 blockage at least once were set as the experimental group. In this connection, treatment efficacy was evaluated based on clinical responses defined as CR (complete response), PR (partial response) and SD (stable disease) using contrast-enhanced CT approximately 8 weeks after the first injection of nivolumab. A responder (R) was defined as a patient with a PR or SD of greater than or equal to 6 months and a non-responder (NR) was defined as a patient having a PD or SD of smaller than 6 months.
[0064] Referring to (a) and (b) in
[0065] Referring to
[0066] Referring to (a) and (b) in
[0067] Based on a result of Example 2 above, PD-L1 and PVR can be used as markers for response prediction to cancer immunotherapy, and the response to PD-1 therapy can be evaluated according to the expression pattern for two biomarkers. For example, a patient group with positive PD-L1 expression and negative PVR expression can be evaluated as having a higher response to the PD-1 blockade therapy. Furthermore, the patient group with PD-L1 expression negative and PVR expression positive can be evaluated as having a lower response to the PD-1 blockade therapy. For this patient group, immune checkpoint blockade strategy different from PD-1 blockade strategy, for example, TIGIT blockade strategy in which TIGIT is a receptor for PVR can be proposed, or a combination therapy of PD-1 blockade strategy and TIGIT blockade strategy can be proposed.
EXAMPLE 3
Early Prediction of Therapeutic Response to PD-1 Blockades Based on the Expression Patterns of PD-L1 and PVR in Mouse Model
[0068] Hereinafter, the evaluation results of the therapeutic response prediction to the anti-PD-1 therapy according to the expression patterns of PD-L1 and PVR in the tumor tissue of a mouse model will be described with reference to
[0069]
[0070] Referring to
[0071] Referring to
[0072] Referring to (a) and (b) in
[0073] Referring to (a) to (d) in
[0074] Based on a result of Example 3 above, the therapeutic response to the anti-PD-1 therapy can vary based on the expression patterns of PD-L1 and PVR in the tumor tissue obtained from the mouse model, and more specifically, the expression patterns of PD-L1 and PVR of the transplanted tumor cell line and the host. Accordingly, a method for providing information on a prediction response for a therapeutic response according to various embodiments of the present disclosure and a kit using the same can predict the therapeutic response to cancer immunotherapy based on the expression patterns of PD-L1 and PVR, and then propose customized cancer immunotherapy in consideration of the patient's tumor microenvironment.
EXAMPLE 4
Setting Up Cancer Immunotherapy having High Therapeutic Response Based on the Expression Patterns of PD-L1 and PVR
[0075] Hereinafter, a method of setting an alternative treatment therapy to PD-1 based on the expression patterns of PD-L1 and PVR will be described in detail with reference to
[0076]
[0077] Referring to (a) and (b) in
[0078] Referring to (a) and (b) in
[0079] Referring to
[0080] Furthermore, in the non-small lung cancer patient 2 (patient no. 2), B7-1 and B7-2, and PVR were expressed along with PD-L1. In other words, even when a PD-1 blockade that inhibits the reaction of PD-L1 and PD-1 was administered theret the patient 2 can have lower response to anti-PD-1 therapy due to reaction of B7-1 and B7-2 of the tumor tissue and CTLA-4 of T-cells, or due to the reaction of PVR of the tumor tissue and TIGIT of T-cells. Thus, the patient 2 can be expected to have a higher anticancer treatment effect when anti-PD-1 therapy was combined with anti-CTL-4 therapy or/and anti-TIGIT therapy than when anti-PD-1 therapy was conducted alone.
[0081] Based on a result of Example 4 above, it is confirmed that anti-TIGIT therapy or combination therapy of anti-PD-1/anti-TIGIT can effectively act as an alternative treatment to the PD-L1−/PVR+ patient group evaluated to have a low response to anti-PD-1 therapy according to the method for providing information on the therapeutic response to cancer immunotherapy in the present disclosure. Accordingly, the present disclosure predicts the early therapeutic response of the subject to the cancer immunotherapy, especially, PD-1 blockage at high sensitivity, and thus can provide information to quickly determine whether to further proceed with anti-PD-1 therapy or whether the anti-PD-1 therapy is to be combined with other immunotherapies.
[0082] The results of Examples 1 to 4 indicate that responses to the first treatment of patients with non-small lung cancer can be predicted early based on the expression patterns of PD-L1 and PVR. That is, PD-L1 and PVR, or PVR can act as practical indicators for prediction of the therapeutic response to immunotherapies of non-small lung cancer.
[0083] However, the present disclosure is not limited to the above, and can be used to provide information for the prediction of a therapeutic response to a variety of immunotherapy methods. For example, the present disclosure can be configured to provide information for prediction of the therapeutic response to at least one therapy selected from the group consisting of anti-CTLA-4 therapy, anti-PD-1 therapy, anti-CD28 therapy, anti-KIR therapy, anti-TCR therapy, anti-LAG-3 therapy, anti-TIM-3 therapy, anti-TIGIT therapy, anti-A2aR therapy, anti-ICOS therapy, anti-OX40 therapy, anti-4-1BB therapy, and anti-GITR therapy.
[0084] Furthermore, the present disclosure can further provide an information providing kit configured to predict a therapeutic response to cancer immunotherapy as the kit contains a formulation configured to measure the expression levels of PD-L1 and PVR, respectively, for a biological sample isolated from a subject.
[0085] The features of the various embodiments of the present disclosure can be partially or entirely coupled or combined with each other. As those skilled in the art can fully understand, various technical associations and operations therebetween can be realized. The embodiments may be implemented independently of each other and may be implemented together in a combined relationship.
[0086] Although the embodiments of the present disclosure have been described in more detail with reference to the accompanying drawings, the present disclosure is not necessarily limited to these embodiments. Various modifications can be made within the scope of the technical idea of the present disclosure. Therefore, the embodiments disclosed in the present disclosure are not intended to limit the technical idea of the present disclosure thereto. The scope of the technical idea of the present disclosure is not limited to the embodiments. Therefore, it should be understood that the embodiments described above are illustrative in all respects and not limiting. The scope of protection of the present disclosure should be construed by the claims below. All technical ideas within the scope of the equivalents thereto should be construed as being included in the scope of the present disclosure.
[0087] National R&D project 1 that supported the present disclosure, Project Identification Number: 2017R1A5A1014560, Ministry Name: Ministry of Science and Technology Information and Communication, Research Management Organization: Korea Research Foundation, Research Project Name: Leading Research Center Business Science (SRC), Research Project Title: Center for Immune Research on Non-lymphoid Organ, Contribution Percentage: 1/5, Host Institution: Yonsei University Industry-Academic Cooperation Foundation, Research Period: 20170601 to 20240228
[0088] National R&D project 2 that supported the present disclosure, Project Identification Number: 2018M3A91-13024850, Ministry Name: Ministry of Science and Technology Information and Communication, Research Management Organization: Korea Research Foundation, Research Project Name: Biomedical Technology Development Project-Grand Challenge, Research Project Title: Developing a precision immunotherapy method based on engineered bacteria, Contribution Percentage: 1/5, Host Institution: Yonsei University Industry-Academic Cooperation Foundation, Research Period: 20180401 to 20261231,
[0089] National R&D project 3 that supported the present disclosure, Project identification Number: 2015R1A2A1A10056084, Ministry Name: Food and Drug Safety Evaluation Institute, Research Management Organization: Food and Drug Safety Evaluation Institute, Research Project Name: Safety Evaluation Technology Development Research Project (Personalized Drug Evaluation Base Research), Research Project Title: Research on development of immune anticancer drug response prediction/evaluation method, Contribution Percentage: 1/5, Host Institution: Yonsei University Industry-Academic Cooperation Foundation, Research Period: 20180516 to 20201130,
[0090] National R&D project 4 that supported the present disclosure, Project Identification Number: NRF-2017M3A9E9072669, Ministry Name: Ministry of Science and Technology Information and Communication, Research Management Organization: Korea Research Foundation, Research Project Name: Biomedical Technology Development Project, Research Project Title: High-precision preclinical model using patient-derived circulating tumor cells, identification of the mechanism of acquired resistance to anticancer drugs through construction and presentation of treatment strategies, Contribution Percentage: 1/5, Host Institution: Yonsei University Industry-Academic Cooperation Foundation, Research Period: 20170901 to 20220531
[0091] National R&D project 5 that supported the present disclosure, Project identification Number: NRF-2017R1D1A1B03029874, Ministry Name: Ministry of Science and Technology information and Communication, Research Management Organization: Korea Research Foundation, Research Project Name: individual basic research in science and engineering (basic, regional), Research Project Title: Immuno-anticancer drugs using immune markers in peripheral blood of lung cancer patients, establishment of effective immuno-cancer treatment strategies through identification of treatment predictors. Contribution Percentage: 1/5, Host institution: Yonsei University Industry-Academic Cooperation Foundation, Research Period: 20170601 to 20200531