HETEROCYCLIC COMPOUND AND HARMFUL-ARTHROPOD-CONTROLLING COMPOSITION CONTAINING SAME

Abstract

The present invention provides a compound that has an excellent control effect on harmful arthropods, and is represented by formula (I) [wherein Z.sup.1 and Z.sup.2 represent an oxygen atom, etc., G.sup.1 represents CR.sup.1a, etc., G.sup.2 represents CR.sup.1c, etc., G.sup.3 represents CR.sup.1d, etc., Q represents a C6-C10 aryl group, etc., R.sup.1b represents a C1-C6 chain hydrocarbon group, etc., and R.sup.1a, R.sup.1c and R.sup.1d represent a C1-C6 chain hydrocarbon group, etc.]

or its N-oxide, or salts thereof.

##STR00001##

Claims

1. A compound represented by formula (I): ##STR00119## [wherein Z.sup.1 and Z.sup.2 are identical or different from each other and each represents an oxygen atom or a sulfur atom, a combination of G.sup.1, G.sup.2, and G.sup.3 represents a combination wherein G.sup.1 represents a nitrogen atom, G.sup.2 represents CR.sup.1c, and G.sup.3 represents CR.sup.1d; a combination wherein G.sup.1 represents CR.sup.1a, G.sup.2 represents a nitrogen atom or CR.sup.1c, G.sup.3 represents CR.sup.1d; or a combination wherein G.sup.1 represents CR.sup.1a, G.sup.2 represents CR.sup.1c, and G.sup.3 represents a nitrogen atom, R.sup.1b represents a C1-C6 chain hydrocarbon group, a C1-C6 alkoxy group {the C1-C6 chain hydrocarbon group and the C1-C6 alkoxy group may be optionally substituted with one or more substituents selected from Group A}, a C3-C7 cycloalkyl group, a C1-C6 alkylsulfanyl group, a C1-C6 alkylsulfinyl group, a C1-C6 alkylsulfonyl group {the C3-C7 cycloalkyl group, the C1-C6 alkylsulfanyl group, the C1-C6 alkylsulfinyl group and the C1-C6 alkylsulfonyl group may be optionally substituted with one or more substituents selected from Group B}, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more substituents selected from Group C, a phenyl group, a three- to seven-membered nonaromatic heterocyclic group {the phenyl group and the three- to seven-membered nonaromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group D, a nitro group, NR.sup.2R.sup.3, or a halogen atom, R.sup.1c represents a C1-C6 chain hydrocarbon group, a C1-C6 alkoxy group {the C1-C6 chain hydrocarbon group and the C1-C6 alkoxy group may be optionally substituted with one or more substituents selected from Group A}, a C3-C7 cycloalkyl group, a C1-C6 alkylsulfanyl group, a C1-C6 alkylsulfinyl group, a C1-C6 alkylsulfonyl group {the C3-C7 cycloalkyl group, the C1-C6 alkylsulfanyl group, the C1-C6 alkylsulfinyl group and the C1-C6 alkylsulfonyl group may be optionally substituted with one or more substituents selected from Group B}, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more substituents selected from Group C, a phenyl group, a three- to seven-membered nonaromatic heterocyclic group {the phenyl group and the three- to seven-membered nonaromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group D}, a nitro group, NR.sup.2R.sup.3, a halogen atom, or a hydrogen atom, R.sup.1a and R.sup.1d are identical or different from each other and each represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a halogen atom, or a hydrogen atom, Q represents a C6-C10 aryl group which may be optionally substituted with one or more substituents selected from Group H, or a five- to ten-membered aromatic heterocyclic group which may be optionally substituted with one or more substituents selected from Group 1, R.sup.2, R.sup.2a and R.sup.5 are identical or different from each other and each represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, or a hydrogen atom, R.sup.3 and R.sup.3a are identical or different from each other and each represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more substituents selected from Group E, a C3-C7 cycloalkyl group, a C3-C7 cycloalkenyl group {the C3-C7 cycloalkyl group and the C3-C7 cycloalkenyl group may be optionally substituted with one or more substituents selected from Group C}, a phenyl group, a five- or six-membered aromatic heterocyclic group {the phenyl group and the five- or six-membered aromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group F}, S(O).sub.2R.sup.13, or a hydrogen atom, R.sup.13 represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, or a phenyl group which may be optionally substituted with one or more substituents selected from Group F. Group A is a group consisting of a C1-C6 alkoxy group, a C3-C6 alkenyloxy group, a C3-C6 alkynyloxy group, a C1-C6 alkylsulfanyl group, a C1-C6 alkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C3-C6 cycloalkyl group {the C1-C6 alkoxy group, the C3-C6 alkenyloxy group, the C3-C6 alkynyloxy group, the C1-C6 alkylsulfanyl group, the C1-C6 alkylsulfinyl group, the C1-C6 alkylsulfonyl group and the C3-C6 cycloalkyl group may be optionally substituted with one or more halogen atoms}, a hydroxy group, a cyano group and a halogen atom. Group B is a group consisting of a C1-C6 chain hydrocarbon group, a C1-C6 alkoxy group, a C3-C6 alkenyloxy group, a C3-C6 alkynyloxy group {the C1-C6 chain hydrocarbon group, the C1-C6 alkoxy group, the C3-C6 alkenyloxy group and the C3-C6 alkynyloxy group may be optionally substituted with one or more halogen atoms}, a hydroxy group, a cyano group, a nitro group and a halogen atom. Group C is a group consisting of a C1-C6 alkyl group which may be optionally substituted with one or more halogen atoms, a cyano group and a halogen atom. Group D is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a five- or six-membered aromatic heterocyclic group which may be optionally substituted with one or more substituents selected from Group F, OR.sup.17, NR.sup.16R.sup.17, C(O)R.sup.17, C(O)NR.sup.16R.sup.17, OC(O)R.sup.16, OC(O)OR.sup.16a, NR.sup.17C(O)R.sup.16a, NR.sup.17C(O)OR.sup.16a, C(O)OR.sup.17, a cyano group, a nitro group and a halogen atom. R.sup.16a represents a C1-C6 alkyl group, or a C3-C6 cycloalkyl group {the C1-C6 alkyl group and the C3-C6 cycloalkyl group may be optionally substituted with one or more halogen atoms}, R.sup.16 and R.sup.17 are identical or different from each other and each represents a C1-C6 alkyl group, a C3-C6 cycloalkyl group {the C1-C6 alkyl group and the C3-C6 cycloalkyl group may be optionally substituted with one or more halogen atoms}, or a hydrogen atom. Group E is a group consisting of a C1-C6 alkoxy group, a C3-C7 cycloalkyl group {the C1-C6 alkoxy group and the C3-C7 cycloalkyl group may be optionally substituted one or more halogen atoms}, a phenyl group, a five- or six-membered aromatic heterocyclic group {the phenyl group and the five- or six-membered aromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group F}, a three- to seven-membered nonaromatic heterocyclic group which may be optionally substituted with one or more substituents selected from Group G, NHR.sup.14, NR.sup.14R.sup.15, an amino group, a cyano group and a halogen atom. R.sup.14 and R.sup.15 are identical or different from each other, and each represents a C1-C6 alkyl group which may be optionally substituted with one or more halogen atoms. Group F is a group consisting of a C1-C6 chain hydrocarbon group, a C1-C6 alkoxy group, a C3-C6 alkenyloxy group, a C3-C6 alkynyloxy group, a C1-C6 alkylsulfanyl group, a C1-C6 alkylsulfinyl group, a C1-C6 alkylsulfonyl group {the C1-C6 chain hydrocarbon group, the C1-C6 alkoxy group, the C3-C6 alkenyloxy group, the C3-C6 alkynyloxy group, the C1-C6 alkylsulfanyl group, the C1-C6 alkylsulfinyl group and the C1-C6 alkylsulfonyl group may be optionally substituted with one or more halogen atoms}, NHR.sup.14, NR.sup.14R.sup.15, C(O)R.sup.14, OC(O)R.sup.14, C(O)OR.sup.14, a hydroxy group, a sulfanyl group, an amino group, a cyano group, a nitro group and a halogen atom. Group G is a group consisting of a C1-C6 chain hydrocarbon group, a C1-C6 alkoxy group, a C3-C6 alkenyloxy group, a C3-C6 alkynyloxy group {the C1-C6 chain hydrocarbon group, the C1-C6 alkoxy group, the C3-C6 alkenyloxy group and the C3-C6 alkynyloxy group may be optionally substituted with one or more halogen atoms}, and a halogen atom. Group H is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more substituents selected from Group A, a C3-C7 cycloalkyl group which may be optionally substituted with one or more substituents selected from Group B, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more substituents selected from Group C, a phenyl group which may be optionally substituted with one or more substituents selected from Group D, a five- or six-membered aromatic heterocyclic group which may be optionally substituted with one or more substituents selected from Group D, OR.sup.3a, NR.sup.2aR.sup.3a NR.sup.2bR.sup.3b, NR.sup.5NR.sup.2aR.sup.3a NR.sup.5OR.sup.2a, NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)OR.sup.7, NR.sup.2aC(O)NR.sup.8R.sup.9, NR.sup.5NR.sup.2aC(O)NR.sup.10R.sup.11, N?CHNR.sup.10R.sup.11, N?S(O).sub.pR.sup.8R.sup.9, C(O)R.sup.12, C(O)NR.sup.10R.sup.11, C(O)NR.sup.2aS(O).sub.2R.sup.13, CR.sup.5?NOR.sup.12, NR.sup.2aCR.sup.5?NOR.sup.12, S(O).sub.mR.sup.13, a cyano group, a nitro group and a halogen atom. p is 0 or 1, m is 0, 1 or 2, R.sup.2b and R.sup.3b combine together with a nitrogen atom to which they are bounded to form a three- to seven-membered nonaromatic heterocyclic group which may be optionally substituted with one or more substituents selected from Group B, R.sup.6 represents a C1-C6 chain hydrocarbon group, a C3-C7 cycloalkyl group, a (C3-C6 cycloalkyl)C1-C3 alkyl group {the C1-C6 chain hydrocarbon group, the C3-C7 cycloalkyl group and the (C3-C6 cycloalkyl)C1-C3 alkyl group may be optionally substituted with one or more halogen atoms}, a phenyl group, a five- or six-membered aromatic heterocyclic group {the phenyl group and the five- or six-membered aromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group F}, or a hydrogen atom. R.sup.6a represents a C1-C6 chain hydrocarbon group, a C3-C7 cycloalkyl group, a (C3-C6 cycloalkyl)C1-C3 alkyl group {the C1-C6 chain hydrocarbon group, the C3-C7 cycloalkyl group and the (C3-C6 cycloalkyl)C1-C3 alkyl group may be optionally substituted with one or more halogen atoms}, a phenyl group, or a five- or six-membered aromatic heterocyclic group {the phenyl group and the five- or six-membered aromatic heterocyclic group may be optionally substituted with one or more substituents selected from Group F}, R.sup.7 represents a C1-C6 chain hydrocarbon group, a C3-C7 cycloalkyl group, a (C3-C6 cycloalkyl)C1-C3 alkyl group {the C1-C6 chain hydrocarbon group, the C3-C7 cycloalkyl group and the (C3-C6 cycloalkyl)C1-C3 alkyl group may be optionally substituted with one or more halogen atoms}, or a phenyl C1-C3 alkyl group {the phenyl moiety in the phenyl C1-C3 alkyl group may be optionally substituted with one or more substituents selected from Group F}, R.sup.8 and R.sup.9 are identical or different from each other and each represents a C1-C6 alkyl group which may be optionally substituted with one or more halogen atoms, R.sup.10 represents a C1-C6 alkyl group which may be optionally substituted with one or more halogen atoms, or a hydrogen atom, R.sup.11 represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more substituents selected from Group B, or a C3-C7 cycloalkyl group which may be optionally substituted with one or more substituents selected from Group G, S(O).sub.2R.sup.6a, or a hydrogen atom, R.sup.12 represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more substituents selected from Group F, or a hydrogen atom. Group I is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more substituents selected from Group A, a C3-C7 cycloalkyl group which may be optionally substituted with one or more substituents selected from Group B, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more substituents selected from Group C, OR.sup.3a, NR.sup.2aR.sup.3a, NR.sup.2bR.sup.3b, NR.sup.5NR.sup.2aR.sup.3a, NR.sup.5OR.sup.2a, NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)OR.sup.7, NR.sup.2aC(O)NR.sup.8R.sup.9, NR.sup.5NR.sup.2aC(O)NR.sup.10R.sup.11, N?CHNR.sup.10R.sup.11, N?S(O).sub.pR.sup.8R.sup.9, C(O)R.sup.12, C(O)NR.sup.10R.sup.11, C(O)NR.sup.2aS(O).sub.2R.sup.13, CR.sup.5?NOR.sup.12, NR.sup.2aCR.sup.5?NOR.sup.12, S(O).sub.mR.sup.13, a cyano group, a nitro group and a halogen atom.], or its N-oxide or a salt thereof.

2. The compound according to claim 1 wherein Z.sup.2 represents an oxygen atom, Q represents a phenyl group, a naphthyl group {the phenyl group and the naphthyl group may be optionally substituted with one or more substituents selected from Group J}, a furanyl group, a thienyl group, a pyrazolyl group, an imidazolyl group, an oxazolyl group, a thiazolyl group, an isoxazolyl group, a pyridyl group, a pyridazinyl group, a pyrimidinyl group, a pyrazinyl group, a quinolyl group, an imidazopyridyl group, a benzofuranyl group, or a benzothiophenyl group {the furanyl group, the thienyl group, the pyrazolyl group, the imidazolyl group, the oxazolyl group, the thiazolyl group, the isoxazolyl group, the pyridyl group, the pyridazinyl group, the pyrimidinyl group, the pyrazinyl group, the quinolyl group, the imidazopyridyl group, the benzofuranyl group and the benzothiophenyl group may be optionally substituted with one or more substituents selected from Group K}, Group J is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more halogen atoms, a five- or six-membered aromatic heterocyclic group which may be optionally substituted with one or more halogen atoms, OR.sup.3a, NR.sup.2aR.sup.3a, NR.sup.2bR.sup.3b, NR.sup.5NR.sup.2aR.sup.3a, NR.sup.5OR.sup.2a, NR.sup.2aC(O)R.sup.6a, NR.sup.5NR.sup.2aC(O)R.sup.6a, NR.sup.5NR.sup.2aC(O)OR.sup.7, NR.sup.2aC(O)NR.sup.8R.sup.9, NR.sup.5NR.sup.2aC(O)NR.sup.10R.sup.11, N?CHNR.sup.10R.sup.11, N?S(O).sub.pR.sup.8R.sup.9, C(O)R.sup.12, C(O)NR.sup.10R.sup.11, C(O)NR.sup.2aS(O).sub.2R.sup.13, CR.sup.5?NOR.sup.12, NR.sup.2aCR.sup.5?NOR.sup.12, S(O).sub.mR.sup.13, a cyano group, a nitro group and a halogen atom. Group K is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkenyl group which may be optionally substituted with one or more halogen atoms, OR.sup.3a, NR.sup.2aR.sup.3a NR.sup.2bR.sup.3bNR.sup.5NR.sup.2aR.sup.3a NR.sup.5OR.sup.2a, NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)R.sup.6a NR.sup.5NR.sup.2aC(O)OR.sup.7, NR.sup.2aC(O)NR.sup.8R.sup.9, NR.sup.5NR.sup.2aC(O)NR.sup.10R.sup.11, N?CHNR.sup.10R.sup.11, N?S(O).sub.mR.sup.8R.sup.9, C(O)R.sup.12, C(O)NR.sup.10R.sup.11, C(O)NR.sup.2aS(O).sub.2R.sup.13, CR.sup.5?NOR.sup.12, NR.sup.2aCR.sup.5?NOR.sup.12, S(O).sub.mR.sup.13, a cyano group, a nitro group and a halogen atom, or its N-oxide or a salt thereof.

3. The compound according to claim 1 wherein G.sup.1 represents CR.sup.1a, G.sup.2 represents a nitrogen atom or CR.sup.1c, and G.sup.3 represents CR.sup.1d or its N-oxide or a salt thereof.

4. The compound according to claim 1 wherein R.sup.1b represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, or a halogen atom, and R.sup.1c represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a halogen atom, or a hydrogen atom, or its N-oxide or a salt thereof.

5. The compound according to claim 1 wherein Q represents a phenyl group, a naphthyl group {the phenyl group and the naphthyl group may be optionally substituted with one or more substituents selected from Group L}, a pyridyl group, or a quinolyl group {the pyridyl group and the quinolyl group may be optionally substituted with one or more substituents selected from Group M}, Group L is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more halogen atoms, OR.sup.19, S(O).sub.mR.sup.19, and a halogen atom, Group M is a group consisting of a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, OR.sup.19, S(O).sub.mR.sup.19, and a halogen atom, R.sup.19 represents a C1-C3 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, or its N-oxide or a salt thereof.

6. The compound according to claim 1 wherein Q represents a group represented by Q1: ##STR00120## [wherein, R.sup.18a, R.sup.18b, and R.sup.18c are identical or different from each other and each represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more halogen atoms, OR.sup.19, S(O).sub.mR.sup.19, a halogen atom, or a hydrogen atom, and R.sup.19 represents a C1-C3 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms], its N-oxide or a salt thereof.

7. The compound according to claim 1 wherein Z.sup.1 and Z.sup.2 represent an oxygen atom, or its N-oxide or a salt thereof.

8. A composition for controlling harmful arthropod comprising the compound of claim 1, or its N-oxide or a salt thereof.

9. A composition which comprises one or more ingredients selected from the group consisting of Group (a), Group (b), Group (c) and Group (d), as well as the compound of claim 1, or its N-oxide or a salt thereof: Group (a): a group consisting of an insecticidal ingredient, a miticidal ingredient, and a nematicidal ingredient; Group (b): a fungicidal ingredient; Group (c): a plant growth modulating ingredient; and Group (d): a repellent ingredient.

10. A method for controlling a harmful arthropod which comprises applying an effective amount of the compound of claim 1, or its N-oxide or a salt thereof, to a harmful arthropod or a habitat where a harmful arthropod lives.

11. A seed or vegetative reproductive organ carrying an effective amount of the compound of claim 1, or its N-oxide or a salt thereof.

12. A compound represented by formula (II): ##STR00121## [wherein, G.sup.4 represents CR.sup.1f or a nitrogen atom, R.sup.1e represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, or a halogen atom, R.sup.1f represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a halogen atom, or a hydrogen atom, R.sup.18d and R.sup.18e are identical or different from each other and each represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more halogen atoms, OR.sup.19a, S(O).sub.nR.sup.19a, a halogen atom, or a hydrogen atom, R.sup.18f represents a C1-C6 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, a C3-C7 cycloalkyl group which may be optionally substituted with one or more halogen atoms, a phenyl group which may be optionally substituted with one or more halogen atoms, OR.sup.19, S(O).sub.nR.sup.19a, or a halogen atom, R.sup.19a represents a C1-C3 chain hydrocarbon group which may be optionally substituted with one or more halogen atoms, and n is 0, 1 or 2.

13. A method for controlling a harmful arthropod which comprises applying an effective amount of the composition of claim 9 to a harmful arthropod or a habitat where a harmful arthropod lives.

14. A seed or vegetative reproductive organ carrying an effective amount of the composition of claim 9.

Description

EXAMPLES

[0361] Hereinafter, the present invention is explained in more detail by Preparation Examples, Reference Preparation Examples, Formulation Examples, and Test Examples, however, the present invention should not be limited to these Examples.

[0362] As used herein, Me represents methyl group, Et represents ethyl group, Pr represents propyl group, i-Pr represents isopropyl group, t-Bu represents tert-butyl group, c-Pr represents cyclopropyl group, c-Bu represents cyclobutyl group, c-Pen represents cyclopentyl group, c-Hex represents cyclohexyl group, Ph represents phenyl group, Py2 represents 2-pyridyl group, Py3 represents 3-pyridyl group, and Py4 represents 4-pyridyl group, and Bn represents benzyl group. When c-Pr, c-Bu, c-Pen, c-Hex, Ph, Py2, Py3, and Py4 has any substituent(s), the substituent(s) is described together with a substitution position before the symbol. For example, 1-CN-c-Pr represents 1-cyanocyclopropyl group, 3,4-F.sub.2-Ph represents 3,4-difluorophenyl group, 4-CF.sub.3-Py2 represents 4-(trifluoromethyl)-2-pyridyl group, and 5-OCH.sub.2CF.sub.2CF.sub.3-Py2 represents 5-(2,2,3,3,3-pentafluoropropoxy)-2-pyridyl group.

[0363] Firstly, Preparation examples of the compound of the present invention are described.

[0364] When a physical property of a compound is measured by a liquid chromatography/mass spectrometry analysis (hereinafter, referred to as LCMS), a measured molecular ion value [M+H].sup.+ or [M?H].sup.? and a retention time (hereinafter, referred to as RT) is described. The measured condition for liquid chromatography (hereinafter, referred to as LC) is described below.

[LC Condition]

[0365] Column: L-column2 ODS, inner diameter 4.6 mm, length 30 mm, particle size 3 ?m

(Chemicals Evaluation and Research Institute, Japan)

[0366] UV measurement wavelength: 254 nm
Mobile phase: A solution: 0.1% aqueous formic acid solution,
B solution: 0.1% formic acid in acetonitrile
Flow Rate: 2.0 mL/min
Pump: LC-20AD (manufacturer SHIMADZU) 2 umps (high pressure gradient)
Gradient condition: The following concentration gradient shown in [Table LC1] is liquid-transferred.

TABLE-US-00001 TABLE LC1 Time (min) A solution (%) B solution (%) 0.01 90 10 2.00 0 100 4.00 0 100 4.01 90 10

[Ms Condition]

[0367] Detector: LCMS-2020 (manufacturer SHIMADZU)
Ionization method: DUIS

Reference Preparation Example 1

[0368] Hydrazine monohydrate 48 g was added to a mixture of 3,4,5-trichloropyridine 73 g, potassium carbonate 69 g, and THF 200 mL at 55? C. over 30 minutes, and the resulting mixture was stirred for 3 hours. Water was added to the resulting mixture, and the mixture was extracted with methyl isobutyl ketone. The resulting organic layer was washed with saturated brine, and dried over anhydrous sodium sulfate, and concentrated under reduced pressure to obtain an intermediate compound 1 represented by the following formula 61 g.

##STR00013##

[0369] Intermediate compound 1: .sup.1H-NMR (CDCl.sub.3) ?: 8.22 (2H, s), 6.09 (1H, s), 4.15 (2H, s).

Reference Preparation Example 1-1

[0370] The compounds which were prepared according to the Reference Preparation Example 1 and their physical property value are shown below.

[0371] A compound represented by formula (A-1):

##STR00014##

wherein a combination of G.sup.1, R.sup.1b, G.sup.2 and G.sup.3 represents any combinations described in [Table A-1]. Here, in working examples, IM represents an intermediate compound.

TABLE-US-00002 TABLE A-1 IM G.sup.1 R.sup.1b G.sup.2 G.sup.3 2 CH C1 CH CH 3 CH Br CH CH 4 CH NO.sub.2 CH CH 5 CH CF.sub.3 CH CH 6 CCl Cl CCl CCl 7 CCl [00015] embedded image N CH 8 CH Br CBr CH

[0372] Intermediate compound 2: .sup.1H-NMR (CDCl.sub.3) ?: 8.24-8.23 (2H, m), 7.03 (1H, d), 6.08 (1H, s), 3.67 (2H, s).

[0373] Intermediate compound 3: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (1H, s), 8.24 (1H, d), 7.01 (1H, d), 6.09 (1H, s), 3.69 (2H, s).

[0374] Intermediate compound 4: .sup.1H-NMR (CDCl.sub.3) ?: 9.19 (1H, s), 9.06 (1H, s), 8.36 (1H, dd), 7.52 (1H, d), 3.86 (2H, s).

[0375] Intermediate compound 5: .sup.1H-NMR (CDCl.sub.3) ?: 8.46 (1H, s), 8.43 (1H, d), 7.24 (1H, d), 6.18 (1H, s), 3.70 (2H, s).

[0376] Intermediate compound 6: LCMS: 248 [M+H].sup.+, RT=1.73 min.

[0377] Intermediate compound 7: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (1H, s), 7.84 (1H, s), 5.96 (1H, s), 4.28-4.24 (2H, m), 4.06-4.05 (2H, m), 4.01-3.97 (2H, m), 2.27-2.21 (1H, m), 1.53-1.50 (1H, m).

[0378] Intermediate compound 8: .sup.1H-NMR (CDCl.sub.3) ?: 8.38 (2H, s), 6.10 (1H, s), 4.12 (2H, s).

Reference Preparation Example 2

[0379] Triethylamine 0.9 mL was added to a mixture of the intermediate compound 1.89 g, 2-methyl-benzoic acid 0.68 mL, DMF 5 mL and BOP 2.75 g, and the mixture was stirred at room temperature for 1 hour. Aqueous saturated sodium hydrocarbonate solution was added to the resulting mixture, and the mixture was filtered. The filtered materials were washed with water and mixed solvent (ethyl acetate:hexane=25:75) successively. The obtained solid was dried under reduced pressure to obtain an intermediate compound 9 represented by the following formula 1.10 g.

##STR00016##

[0380] Intermediate compound 9: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 7.86 (1H, d), 7.50 (1H, d), 7.41-7.39 (1H, m), 7.28-7.28 (2H, m), 7.09 (1H, d), 2.45 (3H, s).

Reference Preparation Example 2-1

[0381] The compounds which were prepared according to the Preparation Example 2 and their physical property value are shown below.

[0382] A compound represented by formula (A-2):

##STR00017##

wherein a combination of A.sup.1, A.sup.2, A.sup.3, A.sup.4 and A.sup.5 represents any combinations described in [Table A-2A], [Table A-2B], and [Table A-2C].

TABLE-US-00003 TABLE A-2A IM A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 10 CF CH CH CH CH 11 CCl CH CH CH CH 12 CBr CH CH CH CH 13 CCF.sub.3 CH CH CH CH 14 COCF.sub.3 CH CH CH CH 15 CH CF CF CH CH 16 CH CF CH CH CH 17 CH CCl CH CH CH 18 CH CBr CH CH CH 19 CH CI CH CH CH 20 CH CCF.sub.3 CH CH CH 21 CH COCF.sub.3 CH CH CH 22 CH CCH.sub.3 CH CH CH 23 CH CH CF CH CH 24 CH CH CCl CH CH 25 CH CH CBr CH CH 26 CH CH CI CH CH 27 CH CH CCF.sub.3 CH CH 28 CH CH COCF.sub.3 CH CH 29 CH CH CCH.sub.3 CH CH 30 COMe CH CH CH CH 31 CH COMe CH CH CH 32 CH CH COMe CH CH 33 CH CH C-iPr CH CH 34 CH CH C-tBu CH CH 35 C-iPr CH CH CH CH 36 CH C-iPr CH CH CH 37 CH COCF.sub.2CHF.sub.2 CH CH CH 38 CH CCN CH CH CH 39 CH CCF.sub.3 CH N CH 40 CH CNO.sub.2 CH CH CH 41 CH CH CNO.sub.2 CH CH 42 CH [00018] embedded image CH CH

TABLE-US-00004 TABLE A-2B IM A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 43 CH CBr CH CC1 CH 44 CH CC1 CH CH N 45 CH CC1 N CH CH 46 CH CC1 CCl CH CH 47 CF CH CF CH CH 48 CF CH CF CH CF 49 CH CF CF CH CF 50 CH CF CH CF CH 51 CH CSCF.sub.3 CH CH CH 52 CH CH CSCF.sub.3 CH CH 53 CH CH N CH N 54 CH N CH CH N 55 CH CCl CH CF CH 56 CH CC1 CF CH CH 57 CH CCF.sub.3 CF CH CH 58 CH COCF.sub.3 CF CH CH 59 CH CH COCH.sub.2CF.sub.2CF.sub.3 CH N 61 N [00019] embedded image CH CH 62 CH [00020] N CH 63 CH CCF.sub.3 CH CF CH 64 CH CF CF CF CH 65 CH COCH.sub.2CF.sub.3 CH CH N 66 CH COCF.sub.3 CH CF CH 67 CH CCF.sub.3 CH CCF.sub.3 CH 68 CH CS (O) CF.sub.3 CH CH CH 69 CH CS (O) .sub.2CF.sub.3 CH CH CH 70 CH CCHF.sub.2 CH CH CH 61 CH CCF.sub.2CF.sub.3 CH CH CH 71 CH COPh CH CH CH 72 CH CBr N CH CH 73 CH CCF.sub.3 CH CCl CH 75 CH CBr CH CF CH 75 CH CBr CF CH CH 76 CH CF CCl CF CH 77 CH CBr CH CBr CH 78 CH COMe CH COMe CH 79 CH CI CMe CH CH 80 CH COCF.sub.3 CH CCl CH

TABLE-US-00005 TABLE A-2C IM A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 81 CH CCF.sub.3 CH CBr CH 82 CH CF CMe CH CH 83 CH CMe CMe CH CH 84 CH CCF.sub.3 CH CMe CH 85 CH CBr CH CMe CH 86 CH CF CMe CF CH 87 CF CCF.sub.3 CH CH CH 88 CH CCF.sub.3 CH CH CF 89 CH CF CF CCl CH 90 CH CBr CF CH CF 91 CH CH CH CH CH 108 CH CH COPh CH CH 109 CH CCF.sub.3 CH CH N 110 CH CCF.sub.3 N CH CH 111 N CCF.sub.3 CH CH CH 112 CH COCHF.sub.2 CH CH CH

[0383] Intermediate compound 10: .sup.1HR-NMR (CDCl.sub.3) ?: 8.89 (1H, d), 8.34 (2H, s), 8.10-8.08 (1H, in), 7.58-7.53 (1H, m), 7.31-7.29 (1H, m), 7.21-7.14 (2H, m).

[0384] Intermediate compound 11: .sup.1H-NMR (CDCl.sub.3) ?: 8.43-8.42 (1H, in), 8.36 (2H, s), 7.75 (1H, d), 7.46-7.45 (2H, m), 7.39-7.37 (1R, at), 7.13-7.13 (1H, m).

[0385] Intermediate compound 12: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.15 (1H, s), 7.65 (1H, d), 7.60 (1H, d), 7.38-7.35 (2H, in), 7.11 (1H, d).

[0386] Intermediate compound 13: .sup.1H-NMR (CDCl.sub.3) ?: 8.38 (2H, s), 7.89 (1H, d), 7.77-7.76 (1H, m), 7.66-7.61 (3H, m), 7.07 (1H, d).

[0387] Intermediate compound 14: .sup.1H-NMR (CDCl.sub.3) ?: 8.74 (1H, d), 8.35 (2H, s), 8.06 (1H, dd), 7.60-7.58 (1H, m), 7.43-7.41 (1H, m), 7.37 (1H, d), 7.14 (1H, d).

[0388] Intermediate compound 15: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.15 (1H, d), 7.70-7.65 (1H, m), 7.59-7.57 (1H, m), 7.30-7.28 (1H, m), 7.06 (1H, d).

[0389] Intermediate compound 16: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.17 (1H, s), 7.58 (1H, d), 7.53-7.45 (2H, m), 7.30-7.28 (1H, m), 7.07 (1H, d).

[0390] Intermediate compound 17: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.18 (1H, d), 7.79-7.79 (1H, m), 7.69-7.67 (1H, m), 7.57-7.55 (1H, m), 7.44-7.42 (1H, m), 7.06 (1H, d).

[0391] Intermediate compound 18: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.15 (1H, d), 7.95-7.94 (1H, m), 7.74-7.70 (2H, m), 7.38-7.36 (1H, m), 7.05 (1H, d).

[0392] Intermediate compound 19: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.26 (1H, s), 8.15 (1H, d), 7.92-7.90 (1H, m), 7.77-7.75 (1H, m), 7.23-7.21 (1H, m), 7.04 (1H, d).

[0393] Intermediate compound 20: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.24 (1H, d), 8.08 (1H, s), 7.99 (1H, d), 7.85 (1H, d), 7.65 (1H, d), 7.08 (1H, d).

[0394] Intermediate compound 21: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.23 (1H, s), 7.72-7.70 (2H, m), 7.55-7.53 (1H, m), 7.43 (1H, d), 7.08 (1H, s).

[0395] Intermediate compound 22: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.17 (1H, d), 7.61-7.59 (2H, m), 7.39-7.38 (2H, m), 7.08 (1H, d), 2.42 (3H, s).

[0396] Intermediate compound 23: LCMS: 300 [M+H].sup.+, RT=1.43 min.

[0397] Intermediate compound 24: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.16 (1H, d), 7.75 (2H, d), 7.47 (2H, d), 7.07 (1H, d).

[0398] Intermediate compound 25: LCMS: 362 [M+H].sup.+, RT=1.66 min.

[0399] Intermediate compound 26: LCMS: 408 [M+H].sup.+, RT=1.70 min.

[0400] Intermediate compound 27: LCMS: 350 [M+H].sup.+, RT=1.71 min.

[0401] Intermediate compound 28: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.17 (1H, d), 7.87 (2H, d), 7.33 (2H, d), 7.08 (1H, d).

[0402] Intermediate compound 29: .sup.1H-NMR (CDCl.sub.3) ?: 8.33 (2H, s), 8.14 (1H, d), 7.71 (2H, d), 7.29 (2H, d), 7.08 (1H, d), 2.42 (3H, s).

[0403] Intermediate compound 30: .sup.1H-NMR (CDCl.sub.3) ?: 10.02 (1H, d), 8.32 (2H, s), 8.18-8.16 (1H, m), 7.54-7.49 (1H, m), 7.24 (1H, d), 7.11-7.09 (1H, m), 7.04 (1H, d), 4.06 (3H, s).

[0404] Intermediate compound 31: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.18 (1H, d), 7.41-7.32 (3H, m), 7.12-7.07 (2H, m), 3.85 (3H, s).

[0405] Intermediate compound 32: .sup.1H-NMR (CDCl.sub.3) ?: 8.33 (2H, s), 8.10-8.09 (1H, m), 7.79-7.77 (2H, m), 7.09-7.08 (1H, m), 6.97-6.96 (2H, m), 3.87 (3H, s).

[0406] Intermediate compound 33: LCMS: 324 [M+H].sup.+, RT=1.76 min

[0407] Intermediate compound 34: .sup.1H-NMR (CDCl.sub.3) ?: 8.33 (2H, s), 8.16 (1H, d), 7.75 (2H, d), 7.50 (2H, d), 7.08 (1H, d), 1.34 (9H, s).

[0408] Intermediate compound 35: LCMS: 324 [M+H].sup.+, RT=2.71 min.

[0409] Intermediate compound 36: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.18-8.17 (1H, m), 7.70 (1H, s), 7.59 (1H, d), 7.43-7.40 (2H, m), 7.09 (1H, s), 3.00-2.94 (1H, m), 1.27 (6H, d).

[0410] Intermediate compound 37: LCMS: 398 [M+H].sup.+, RT=1.72 min.

[0411] Intermediate compound 38: .sup.1H-NMR (CDCl.sub.3) ?: 8.40 (1H, s), 8.36 (2H, s), 8.11 (1H, d), 8.05 (1H, dd), 7.87 (1H, dd), 7.65-7.63 (1H, m), 7.07 (1H, s).

[0412] Intermediate compound 39: LCMS: 351 [M+H].sup.+, RT=1.46 min.

[0413] Intermediate compound 40: .sup.1H-NMR (CDCl.sub.3) ?: 8.67-8.65 (1H, m), 8.46-8.44 (1H, m), 8.37 (2H, s), 8.33 (1H, d), 8.16 (1H, d), 7.73-7.71 (1H, m), 7.08 (1H, d).

[0414] Intermediate compound 41: .sup.1H-NMR (CDCl.sub.3) ?: 8.38 (2H, s), 8.35 (2H, d), 8.27 (1H, d), 7.99 (2H, d), 7.09 (1H, d).

[0415] Intermediate compound 42: .sup.1H-NMR (CDCl.sub.3) ?: 8.37-8.33 (4H, m), 7.96-7.94 (2H, m), 7.91 (1H, d), 7.84 (1H, d), 7.64-7.58 (2H, m), 7.16 (1H, s).

[0416] Intermediate compound 43: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.15 (1H, d), 7.81-7.81 (1H, m), 7.72-7.71 (2H, m), 7.02 (1H, d).

[0417] Intermediate compound 44: .sup.1H-NMR (CDCl.sub.3) ?: 9.81 (1H, s), 8.52 (1H, d), 8.33 (2H, s), 8.12 (1H, d), 7.51 (1H, dd), 6.97 (1H, d).

[0418] Intermediate compound 45: .sup.1H-NMR (CDCl.sub.3) ?: 8.57 (1H, d), 8.36 (2H, s), 8.01 (1H, s), 7.71 (1H, s), 7.58 (1H, d), 7.03 (1H, s).

[0419] Intermediate compound 46: LCMS: 352 [M+H].sup.+, RT=1.77 min.

[0420] Intermediate compound 47: .sup.1H-NMR (CDCl.sub.3) ?: 8.78 (1H, d), 8.34 (2H, s), 8.12 (1H, dd), 7.11 (1H, s), 7.03 (1H, dd), 6.95 (1H, dd).

[0421] Intermediate compound 48: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.13 (1H, s), 7.07 (1H, d), 6.80-6.77 (2H, m).

[0422] Intermediate compound 49: .sup.1H-NMR (CDCl.sub.3) ?: 8.80 (1H, d), 8.35 (2H, s), 7.93 (1H, d), 7.10-7.07 (2H, m).

[0423] Intermediate compound 50: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.18 (1H, d), 7.34-7.30 (2H, m), 7.07-7.00 (2H, m).

[0424] Intermediate compound 51: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.24 (1H, d), 8.10 (1H, s), 7.93 (1H, d), 7.87 (1H, d), 7.58-7.56 (1H, m), 7.08 (1H, d).

[0425] Intermediate compound 52: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.21 (1H, d), 7.85 (2H, d), 7.77 (2H, d), 7.08 (1H, d).

[0426] Intermediate compound 53: .sup.1H-NMR (CDCl.sub.3) ?: 9.86 (1H, s), 9.31 (1H, s), 9.02 (1H, d), 8.35 (2H, s), 8.05 (1H, d), 6.99 (1H, s).

[0427] Intermediate compound 54: .sup.1H-NMR (CDCl.sub.3) ?: 9.68 (1H, d), 9.34 (1H, d), 8.83 (1H, d), 8.60 (1H, dd), 8.34 (2H, s), 6.99 (1H, d).

[0428] Intermediate compound 55: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.29 (1H, s), 7.58 (1H, s), 7.42 (1H, d), 7.30 (1H, d), 7.04 (1H, s).

[0429] Intermediate compound 56: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.13 (1H, s), 7.90-7.88 (1H, m), 7.72-7.71 (1H, m), 7.18-7.16 (1H, m), 7.05 (1H, s).

[0430] Intermediate compound 57: LCMS: 368 [M+H].sup.+, RT=1.76 min.

[0431] Intermediate compound 58: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.22 (1H, d), 7.83 (1H, d), 7.77-7.74 (1H, m), 7.34-7.32 (1H, m), 7.05 (1H, d).

[0432] Intermediate compound 59: .sup.1H-NMR (CDCl.sub.3) ?: 9.70 (1H, s), 8.34-8.32 (3H, m), 8.13 (1H, d), 7.37 (1H, d), 6.96 (1H, d), 4.56-4.53 (2H, m).

[0433] Intermediate compound 60: .sup.1H-NMR (CDCl.sub.3) ?: 10.10 (1H, d), 8.35-8.34 (3H, m), 8.21-8.17 (2H, m), 7.91 (1H, d), 7.84-7.80 (1H, m), 7.69-7.65 (1H, m), 7.03 (1H, d).

[0434] Intermediate compound 61: .sup.1H-NMR (CDCl.sub.3) ?: 9.30 (1H, d), 8.64 (1H, d), 8.41 (1H, d), 8.38 (2H, s), 8.18 (1H, d), 7.95 (1H, d), 7.89-7.85 (1H, m), 7.68-7.66 (1H, m), 7.15 (1H, d).

[0435] Intermediate compound 62: LCMS: 368[M+H].sup.+, RT=1.78 min.

[0436] Intermediate compound 63: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.12 (1H, d), 7.47-7.46 (2H, m), 7.03 (1H, d).

[0437] Intermediate compound 64: .sup.1H-NMR (CDCl.sub.3) ?: 9.70 (1H, d), 8.35 (1H, d), 8.32 (2H, s), 8.12 (1H, d), 7.36 (1H, dd), 6.95 (1H, d), 4.48 (2H, q).

[0438] Intermediate compound 65: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.28 (1H, s), 7.48-7.45 (2H, m), 7.18 (1H, d), 7.05 (1H, s).

[0439] Intermediate compound 66: .sup.1H-NMR (CDCl.sub.3) ?: 8.46 (1H, d), 8.38 (2H, s), 8.27 (2H, s), 8.09 (1H, s), 7.06 (1H, d).

[0440] Intermediate compound 67: LCMS: 398 [M+H].sup.+, RT=1.71 min.

[0441] Intermediate compound 68: LCMS: 414 [M+H].sup.+, RT=2.21 min.

[0442] Intermediate compound 69: LCMS: 332 [M+H].sup.+, RT=1.74 min.

[0443] Intermediate compound 70: LCMS: 400 [M+H].sup.+, RT=1.45 min.

[0444] Intermediate compound 71: LCMS: 372 [M?H].sup.?, RT=1.44 min.

[0445] Intermediate compound 72: LCMS: 363 [M+H].sup.+, RT=1.02 min.

[0446] Intermediate compound 73: LCMS: 384 [M+H].sup.+, RT=1.44 min.

[0447] Intermediate compound 74: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.23 (1H, d), 7.72 (1H, s), 7.47-7.45 (2H, m), 7.03 (1H, d).

[0448] Intermediate compound 75: LCMS: 380 [M+H].sup.+, RT=1.28 min.

[0449] Intermediate compound 76: LCMS: 352 [M+H].sup.+, RT=1.35 min.

[0450] Intermediate compound 77: LCMS: 440 [M+H].sup.+, RT=1.49 min.

[0451] Intermediate compound 78: +H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.13 (1H, d), 7.05 (1H, d), 6.92 (2H, s), 6.63 (1H, s), 3.83 (6H, s).

[0452] Intermediate compound 79: +H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.24 (1H, d), 8.12 (1H, d), 7.67 (1H, dd), 7.33 (1H, d), 7.04 (1H, d), 2.49 (3H, s).

[0453] Intermediate compound 80: LCMS: 400 [M+H].sup.+, RT=1.93 min.

[0454] Intermediate compound 81: .sup.1H-NMR (CDCl.sub.3) ?: 8.37 (2H, s), 8.25 (1H, d), 8.11 (1H, s), 7.99-7.97 (2H, m), 7.04 (1H, d).

[0455] Intermediate compound 82: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.13 (1H, d), 7.48-7.46 (2H, m), 7.32-7.30 (1H, m), 7.06 (1H, d), 2.34 (3H, s).

[0456] Intermediate compound 83: .sup.1H-NMR (CDCl.sub.3) ?: 8.33 (2H, s), 8.13 (1H, d), 7.58 (1H, s), 7.52 (1H, d), 7.22 (1H, d), 7.07 (1H, d), 2.32 (6H, s).

[0457] Intermediate compound 84: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.21 (1H, d), 7.85 (1H, s), 7.79 (1H, s), 7.64 (1H, s), 7.06 (1H, d), 2.49 (3H, s).

[0458] Intermediate compound 85: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.12 (1H, d), 7.71 (1H, s), 7.53-7.52 (2H, m), 7.03 (1H, d), 2.40 (3H, s).

[0459] Intermediate compound 86: .sup.1H-NMR (CDCl.sub.3) ?: 8.35 (2H, s), 8.11 (1H, d), 7.30-7.29 (2H, m), 7.04 (1H, d), 2.26 (3H, s).

[0460] Intermediate compound 87: .sup.1H-NMR (CDCl.sub.3) ?: 8.82 (1H, dd), 8.36 (2H, s), 8.29-8.27 (1H, m), 7.85-7.83 (1H, m), 7.44-7.42 (1H, m), 7.13 (1H, d).

[0461] Intermediate compound 88: .sup.1H-NMR (CDCl.sub.3) ?: 8.89 (1H, dd), 8.42 (1H, dd), 8.36 (2H, s), 7.85-7.81 (1H, m), 7.35 (1H, dd), 7.13 (1H, d).

[0462] Intermediate compound 89: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (2H, s), 8.16 (1H, d), 7.66-7.65 (1H, m), 7.59-7.55 (1H, m), 7.02 (1H, d).

[0463] Intermediate compound 90: LCMS: 398 [M+H].sup.+, RT=1.71 min.

[0464] Intermediate compound 91: .sup.1H-NMR (CDCl.sub.3) ?: 8.34 (2H, s), 8.28 (1H, d), 7.81 (2H, d), 7.60-7.56 (1H, m), 7.52-7.45 (2H, m), 7.09 (1H, d).

[0465] Intermediate compound 108: .sup.1H-NMR (CDCl.sub.3) ?: 8.33 (2H, s), 8.11 (1H, d), 7.79-7.77 (2H, m), 7.41-7.39 (2H, m), 7.19 (1H, d), 7.06-7.03 (5H, m).

[0466] Intermediate compound 109: .sup.1H-NMR (CDCl.sub.3) ?: 9.85 (1H, d), 8.82 (1H, d), 8.37 (1H, s), 8.34 (2H, s), 7.74 (1H, d), 7.00 (1H, d).

[0467] Intermediate compound 110: LCMS: 351 [M+H].sup.+, RT=1.51 min.

[0468] Intermediate compound 111: .sup.1H-NMR (CDCl.sub.3) ?: 9.82 (1H, d), 8.34-8.32 (3H, m), 8.12-8.09 (1H, m), 7.90 (1H, d), 6.99 (1H, d).

[0469] Intermediate compound 112: LCMS: 348 [M+H].sup.+, RT=1.62 min.

Reference Preparation Example 2-2

[0470] The compounds which were prepared according to the Preparation Example 2 and their physical property value are shown below.

[0471] A compound represented by formula (A-3):

##STR00021##

wherein Q represents any substituents described in [Table A-3A] and [Table A-3B].

TABLE-US-00006 TABLE A-3A IM Q 92 [00022] embedded image 94 [00023] 96 [00024] 98 [00025]

TABLE-US-00007 TABLE A-3B IM O 93 [00026] embedded image 95 [00027] 97 [00028]

[0472] Intermediate compound 92: LCMS: 288 [M+H].sup.+, RT=1.26 min.

[0473] Intermediate compound 93: LCMS: 272 [M+H].sup.+, RT=1.06 min.

[0474] Intermediate compound 94: LCMS: 356 [M+H].sup.+, RT=1.74 min.

[0475] Intermediate compound 95: LCMS: 322 [M+H].sup.+, RT=1.55 min.

[0476] Intermediate compound 96: +H-NMR (CDCl.sub.3) ?: 8.83 (1H, d), 8.32 (2H, s), 8.11 (1H, s), 6.90 (1H, d), 2.51 (3H, s).

[0477] Intermediate compound 97: LCMS: 286 [M+H].sup.+, RT=0.67 min.

[0478] Intermediate compound 98: LCMS: 286 [M+H].sup.+, RT=1.04 min.

[0479] A compound represented by formula (A-4):

##STR00029##

wherein a combination of G.sup.1, G.sup.4, R.sup.1e, R.sup.18d, R.sup.18e, and R.sup.18f represents any combinations described in [Table A-4].

TABLE-US-00008 TABLE A-4 IM G.sup.1 G.sup.4 R.sup.1e R.sup.18d R.sup.18e R.sup.18f 99 CCl N [00030] embedded image CF.sub.3 H H 100 CH CH Cl CF.sub.3 H H 101 CH CH Cl OCF.sub.3 H H 102 CH CH Br CF.sub.3 H H 103 CH CH NO.sub.2 CF.sub.3 H H 104 CH CH CF.sub.3 CF.sub.3 H H 105 CH CBr Br H H H 106 CH CBr Br CF.sub.3 H H 107 CH CBr Br OCF.sub.3 H H 114 CH CBr Br F F H 115 CH CBr Br H F H 116 CH CBr Br f Br H 117 CH CF Cl CF.sub.3 H H 118 CH CF Cl F F H

[0480] Intermediate compound 99: .sup.1H-NMR (CDCl.sub.3) ?: 9.73 (1H, s), 9.22 (1H, s), 8.38 (1H, s), 8.15 (1H, s), 8.05-8.03 (1H, m), 7.84 (1H, d), 7.66-7.64 (1H, m), 6.02 (1H, s), 4.38-4.36 (2H, m), 4.06-4.03 (2H, m), 1.32-1.31 (1H, m), 1.27-1.25 (1H, m).

[0481] Intermediate compound 100: LCMS: 314 [M?H]?, RT=1.08 min.

[0482] Intermediate compound 101: LCMS: 330 [M?H]?, RT=1.16 min.

[0483] Intermediate compound 102: .sup.1H-NMR (CDCl.sub.3) ?: 8.51 (1H, s), 8.28 (1H, d), 8.14 (1H, s), 8.09-8.07 (2H, m), 7.88 (1H, d), 7.69-7.67 (1H, m), 6.81-6.80 (2H, m).

[0484] Intermediate compound 103: LCMS: 327 [M+H].sup.+, RT=1.40 min.

[0485] Intermediate compound 104: LCMS: 350 [M+H].sup.+, RT=1.19 min.

[0486] Intermediate compound 105: LCMS: 370 [M?H].sup.?, RT=1.40 min.

[0487] Intermediate compound 106: LCMS: 440 [M+H].sup.+, RT=1.74 min.

[0488] Intermediate compound 107: LCMS: 454 [M?H].sup.?, RT=1.78 min.

[0489] Intermediate compound 114: .sup.1H-NMR (CDCl.sub.3) ?: 8.49 (2H, s), 8.28-8.24 (1H, m), 7.73-7.66 (1H, m), 7.62-7.58 (1H, m), 7.33-7.24 (1H, m), 7.07-7.02 (1H, m).

[0490] Intermediate compound 115: .sup.1H-NMR (CDCl.sub.3) ?: 8.50 (2H, s), 8.21 (1H, d), 7.89-7.85 (2H, m), 7.20-7.16 (2H, m), 7.08 (1H, d).

[0491] Intermediate compound 116: .sup.1H-NMR (CDCl.sub.3) ?: 8.51 (2H, s), 8.24 (1H, d), 7.74-7.68 (1H, m), 7.62-7.59 (1H, m), 7.51-7.49 (1H, m), 7.06 (1H, d).

[0492] Intermediate compound 117: .sup.1H-NMR (CDCl.sub.3) ?: 8.36 (1H, s), 8.29 (1H, s), 8.26-8.23 (1H, m), 8.07 (1H, s), 8.00 (1H, d), 7.85 (1H, d), 7.68-7.62 (1H, m), 6.89 (1H, s).

[0493] Intermediate compound 118: .sup.1H-NMR (CDCl.sub.3) ?: 8.29 (1H, s), 8.24 (1H, d), 8.19-8.16 (1H, m), 7.70-7.65 (1H, m), 7.60-7.55 (1H, m), 7.34-7.28 (1H, m), 6.87-6.84 (1H, m).

Preparation Example 1

[0494] Triethylamine 1.75 mL was added to a mixture of the intermediate compound 9 1.10 g, THF 25 mL and triphosgene 1.04 g, and the resulting mixture was stirred at room temperature for 1 hour. Aqueous saturated sodium hydrogencarbonate solution 20 mL was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting mixture was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain a present compound 1 represented by the following formula 0.38 g.

##STR00031##

[0495] Present compound 1: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.88 (1H, d), 7.47-7.45 (1H, m), 7.37-7.35 (2H, m), 2.63 (3H, s).

Preparation Example 1-1

[0496] The compounds which were prepared according to the Preparation Example 1 and their physical property value are shown below.

[0497] A compound represented by formula (B-1):

##STR00032##

wherein a combination of A.sup.1, A.sup.2, A.sup.3, A.sup.4 and A.sup.5 represents any combinations described in [Table B-1A], [Table B-1B] and [Table B-1C]. Here in the working examples, Comp represents present compound.

TABLE-US-00009 TABLE B-1A Comp A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 2 CH CH CH CH CH 3 CCl CH CH CH CH 4 CBr CH CH CH CH 5 CCF.sub.3 CH CH CH CH 6 COCF.sub.3 CH CH CH CH 7 CH CF CH CH CH 8 CH CCl CH CH CH 9 CH CBr CH CH CH 10 CH CI CH CH CH 11 CH CCF.sub.3 CH CH CH 12 CH COCF.sub.3 CH CH CH 13 CH CCH.sub.3 CH CH CH 14 CH CH CF CH CH 15 CH CH CCl CH CH 16 CH CH CBr CH CH 17 CH CH CI CH CH 18 CH CH CCF.sub.3 CH CH 19 CH CH COCF.sub.3 CH CH 20 CH CH CCH.sub.3 CH CH 21 COMe CH CH CH CH 22 CH COMe CH CH CH 23 CH CH COMe CH CH 24 CH CH C-iPr CH CH 25 CH CH C-tBu CH CH 26 C-iPr CH CH CH CH 27 CH C-iPr CH CH CH 28 CH COCF.sub.2CHF.sub.2 CH CH CH 29 CF CH CH CH CH 30 CH CF CH C-F CH 31 CH CNO.sub.2 CH CH CH 32 CH CH CNO.sub.2 CH CH 33 CH [00033] embedded image CH CH 34 CH CBr CH CCl CH 35 CH CC1 CH CH N 36 CH CCl N CH CH 37 CH CCl CCl CH CH 38 CF CH CF CH CH 39 CF CH CF CH CF 40 CH CF CF CH CF 41 CH CF CF CH CH

TABLE-US-00010 TABLE B-1B Comp A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 42 CH CSCF.sub.3 CH CH CH 43 CH CH CSCF.sub.3 CH CH 44 CH CH N CH N 45 CH N CH CH N 46 CH CCl CH CF CH 47 CH CCl CF CH CH 48 CH CCF.sub.3 CF CH CH 49 CH COCF.sub.3 CF CH CH 50 CH CH COCH.sub.2CF.sub.2CF.sub.3 CH N 51 N [00034] embedded image CH CH 52 CH [00035] N CH 53 CH CCF.sub.3 CH CF CH 54 CH CF CF CF CH 55 CH COCH.sub.2CF.sub.3 CH CH N 56 CH COCF.sub.3 CH CF CH 57 CH CCF.sub.3 CH CCF.sub.3 CH 58 CH CS(O)CF.sub.3 CH CH CH 59 CH CS(O).sub.2CF.sub.3 CH CH CH 60 CH CCHF.sub.2 CH CH CH 61 CH CCF.sub.2CF.sub.3 CH CH CH 62 CH COPh CH CH CH 63 CH CBr N CH CH 64 CH CCF.sub.3 CH CCl CH 65 CH CBr CH CF CH 66 CH CBr C-F CH CH 67 CH CCN CH CH CH 68 CH CBr CH CBr CH 69 CH COMe CH COMe CH 70 CH CI CMe CH CH 71 CH COCF.sub.3 CH CCl CH 72 CH CCF.sub.3 CH CBr CH 73 CH CF CMe CH CH 74 CH CMe CMe CH CH 75 CH CCF.sub.3 CH CMe CH 76 CH CBr CH CMe CH 77 CH CCF.sub.3 CH N CH 78 C-F CCF.sub.3 CH CH CH 79 CH CCF.sub.3 CH CH CF 80 CH CF CF CCl CH 81 CH CBr CF CH CF

TABLE-US-00011 TABLE B-1C Comp A.sup.1 A.sup.2 A.sup.3 A.sup.4 A.sup.5 137 CH CH COPh CH CH 138 CH CCF.sub.3 CH CH N 139 CH CCF.sub.3 N CH CH 140 N CCF.sub.3 CH CH CH 145 CH COCHF.sub.2 CH CH CH

[0498] Present compound 2: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.94-7.91 (2H, m), 7.59-7.53 (3H, m).

[0499] Present compound 3: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.90 (1H, dd), 7.58-7.56 (1N, in), 7.53-7.49 (1N, in), 7.45-7.43 (1N, in).

[0500] Present compound 4: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.86 (1H, d), 7.77 (1N, d), 7.51-7.47 (1N, in), 7.44-7.40 (1N, m).

[0501] Present compound 5: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.94-7.88 (2H, m), 7.75-7.74 (2H, m).

[0502] Present compound 6: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.96 (1H, dd), 7.65-7.62 (1H, m), 7.49-7.46 (2H, m).

[0503] Present compound 7: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.72 (1H, dd), 7.62 (1H, dd), 7.53-7.50 (1H, m), 7.31-7.29 (1H, m).

[0504] Present compound 8: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.92 (1H, s), 7.81 (1H, d), 7.56 (1H, d), 7.48-7.46 (1H, m).

[0505] Present compound 9: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.08 (1H, s), 7.85 (1H, d), 7.71 (1H, d), 7.42-7.40 (1H, m).

[0506] Present compound 10: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.27 (1H, d), 7.91-7.88 (2H, m), 7.26-7.24 (1H, m).

[0507] Present compound 11: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.20 (1H, s), 8.12-8.10 (1H, m), 7.85-7.83 (1H, m), 7.71-7.67 (1H, m).

[0508] Present compound 12: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.86 (1H, d), 7.77 (1H, s), 7.59-7.57 (1H, m), 7.44 (1H, d).

[0509] Present compound 13: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.74-7.71 (2H, m), 7.41-7.40 (2H, m), 2.44 (3H, s).

[0510] Present compound 14: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.95-7.91 (2H, m), 7.23-7.21 (2H, m).

[0511] Present compound 15: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.86 (2H, d), 7.51 (2H, d).

[0512] Present compound 16: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.78 (2H, d), 7.67 (2H, d).

[0513] Present compound 17: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.89 (2H, d), 7.63 (2H, d)).

[0514] Present compound 18: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.05 (2H, d), 7.80 (2H, d).

[0515] Present compound 19: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.97 (2H, d), 7.37 (2H, d).

[0516] Present compound 20: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.80 (2H, d), 7.32 (2H, d), 2.44 (3H, s).

[0517] Present compound 21: .sup.1H-NMR (CDCl.sub.3) ?: 8.69 (2H, s), 7.82 (1H, dd), 7.55-7.53 (1H, m), 7.10-7.06 (2H, m), 3.96 (3H, s).

[0518] Present compound 22: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.51 (1H, dd), 7.45-7.41 (2H, m), 7.13-7.10 (1H, m), 3.87 (3H, s).

[0519] Present compound 23: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.85 (2H, d), 7.01 (2H, d), 3.89 (3H, s).

[0520] Present compound 24: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.89 (1H, d), 7.84 (1H, d), 7.38 (1H, d), 7.16 (1H, d), 3.02-2.95 (1H, m), 1.29 (6H, d).

[0521] Present compound 25: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.85 (2H, d), 7.54 (2H, d), 1.36 (9H, s).

[0522] Present compound 26: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.81 (1H, d), 7.53-7.51 (2H, m), 7.35-7.33 (1H, m), 3.85-3.78 (1H, m), 1.28 (6H, d).

[0523] Present compound 27: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.77 (1H, d), 7.75-7.72 (1H, m), 7.45-7.44 (2H, m), 3.02-2.95 (1H, m), 1.29 (6H, d).

[0524] Present compound 28: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.85 (1H, d), 7.78 (1H, s), 7.58-7.56 (1H, m), 7.44 (1H, d), 5.95 (1H, t).

[0525] Present compound 29: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, d), 7.90-7.88 (1H, m), 7.60-7.56 (1H, m), 7.35-7.29 (2H, m).

[0526] Present compound 30: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.46-7.45 (2H, m), 7.05-7.03 (1H, m).

[0527] Present compound 31: .sup.1H-NMR (CDCl.sub.3) ?: 8.79 (1H, s), 8.74 (2H, s), 8.44 (1H, d), 8.24 (1H, d), 7.77-7.75 (1H, m).

[0528] Present compound 32: .sup.1H-NMR (CDCl.sub.3) ?: 8.74 (2H, s), 8.40 (2H, d), 8.12 (2H, d).

[0529] Present compound 33: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.43 (1H, s), 7.97-7.94 (3H, m), 7.91 (1H, d), 7.65-7.58 (2H, m).

[0530] Present compound 34: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.96-7.95 (1H, m), 7.85-7.84 (1H, m), 7.72-7.71 (1H, m).

[0531] Present compound 35: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.69 (1H, dd), 7.98 (1H, dd), 7.51 (1H, dd).

[0532] Present compound 36: .sup.1H-NMR (CDCl.sub.3) ?: 8.74 (2H, s), 8.61 (1H, d), 7.82 (1H, d), 7.70 (1H, dd).

[0533] Present compound 37: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.02 (1H, d), 7.75 (1H, dd), 7.62 (1H, d).

[0534] Present compound 38: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.91-7.88 (1H, m), 7.09-7.00 (2H, m).

[0535] Present compound 39: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 6.91-6.85 (2H, m).

[0536] Present compound 40: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.74-7.71 (1H, m), 7.17-7.14 (1H, m).

[0537] Present compound 41: .sup.1H-NMR (CDCl.sub.3) ?: 8.76 (2H, s), 7.82-7.77 (1H, m), 7.76-7.72 (1H, m), 7.41-7.34 (1H, m).

[0538] Present compound 42: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.22 (1H, s), 8.05-8.04 (1H, m), 7.87-7.87 (1H, m), 7.63-7.59 (1H, m).

[0539] Present compound 43: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.97 (2H, d), 7.81 (2H, d).

[0540] Present compound 44: .sup.1H-NMR (CDCl.sub.3) ?: 9.44 (1H, d), 9.03 (1H, d), 8.73 (2H, s), 7.91 (1H, d).

[0541] Present compound 45: .sup.1H-NMR (CDCl.sub.3) ?: 9.23-9.22 (1H, m), 8.80-8.79 (1H, m), 8.78-8.77 (1H, m), 8.73 (2H, s).

[0542] Present compound 46: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.73 (1H, s), 7.54-7.52 (1H, m), 7.32-7.30 (1H, m).

[0543] Present compound 47: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.00 (1H, dd), 7.83-7.81 (1H, m), 7.32-7.29 (1H, m).

[0544] Present compound 48: .sup.1H-NMR (CDCl.sub.3) ?: 8.74 (2H, s), 8.21-8.19 (1H, m), 8.14-8.10 (1H, m), 7.41-7.38 (1H, m).

[0545] Present compound 49: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 7.89-7.88 (2H, m), 7.40-7.38 (1H, m).

[0546] Present compound 50: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.52-8.52 (1H, m), 7.97-7.95 (1H, m), 7.43-7.41 (1H, m), 4.59-4.56 (2H, m).

[0547] Present compound 51: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.36 (1H, d), 8.29 (1H, d), 8.05 (1H, d), 7.92 (1H, d), 7.85-7.83 (1H, m), 7.70-7.68 (1H, m).

[0548] Present compound 52: .sup.1H-NMR (CDCl.sub.3) ?: 9.40 (1H, d), 8.74 (2H, s), 8.69 (1H, d), 8.20 (1H, d), 7.97 (1H, d), 7.89-7.87 (1H, m), 7.70-7.68 (1H, m).

[0549] Present compound 53: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, d), 8.00 (1H, s), 7.81 (1H, d), 7.55 (1H, d).

[0550] Present compound 54: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.59-7.56 (2H, m).

[0551] Present compound 55: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.53 (1H, d), 7.96-7.95 (1H, m), 7.43-7.41 (1H, m), 4.51 (2H, q).

[0552] Present compound 56: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, d), 7.59-7.58 (2H, m), 7.18 (1H, d).

[0553] Present compound 57: .sup.1H-NMR (CDCl.sub.3) ?: 8.75 (2H, s), 8.37 (2H, s), 8.08 (1H, s).

[0554] Present compound 58: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, d), 8.33 (1H, s), 8.21 (1H, d), 8.01 (1H, d), 7.83-7.81 (1H, m).

[0555] Present compound 59: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, d), 8.58 (1H, s), 8.38-8.36 (1H, m), 8.24 (1H, d), 7.90-7.88 (1H, m).

[0556] Present compound 60: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.08 (1H, s), 8.04 (1H, d), 7.73 (1H, d), 7.66-7.64 (1H, m), 6.72 (1H, t).

[0557] Present compound 61: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.15-8.13 (2H, m), 7.82 (1H, d), 7.72-7.70 (1H, m).

[0558] Present compound 62: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.65-7.63 (1H, m), 7.51-7.51 (1H, m), 7.48-7.46 (1H, m), 7.40-7.38 (2H, m), 7.20-7.18 (2H, m), 7.07-7.04 (2H, m) Present compound 63: .sup.1H-NMR (CDCl.sub.3) ?: 8.74 (2H, s), 8.59 (1H, d), 7.98 (1H, s), 7.73 (1H, d)).

[0559] Present compound 64: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.09 (1H, s), 8.07 (1H, s), 7.81 (1H, s).

[0560] Present compound 65: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.88 (1H, s), 7.58-7.56 (1H, m), 7.47-7.45 (1H, m).

[0561] Present compound 66: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.16-8.15 (1H, m), 7.87-7.85 (1H, m), 7.30-7.29 (1H, m).

[0562] Present compound 67: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.22 (1H, s), 8.15 (1H, d), 7.87 (1H, d), 7.69 (1H, t).

[0563] Present compound 68: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.00 (2H, s), 7.87 (1H, s).

[0564] Present compound 69: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.05 (2H, d), 6.65-6.64 (1H, m), 3.85 (6H, s).

[0565] Present compound 70: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.35 (1H, d), 7.78 (1H, dd), 7.37 (1H, d), 2.52 (3H, s).

[0566] Present compound 71: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 7.87 (1H, s), 7.67 (1H, s), 7.44 (1H, s).

[0567] Present compound 72: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, s), 8.25 (1H, s), 8.11 (1H, s), 7.96 (1H, s).

[0568] Present compound 73: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.60 (1H, dd), 7.55 (1H, dd), 7.35-7.33 (1H, m), 2.37 (3H, d)).

[0569] Present compound 74: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.68 (1H, s), 7.64 (1H, d), 7.29-7.28 (1H, m), 2.35 (3H, s), 2.33 (3H, s).

[0570] Present compound 75: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.99 (1H, s), 7.91 (1H, s), 7.64 (1H, s), 2.52 (3H, s).

[0571] Present compound 76: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.87 (1H, s), 7.66 (1H, s), 7.54 (1H, s), 2.42 (3H, s).

[0572] Present compound 77: .sup.1H-NMR (CDCl.sub.3) ?: 9.34 (1H, s), 9.08 (1H, s), 8.74 (2H, s), 8.43 (1H, s).

[0573] Present compound 78: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.11-8.09 (1H, m), 7.86-7.84 (1H, m), 7.47-7.45 (1H, m).

[0574] Present compound 79: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.19 (1H, dd), 7.87-7.83 (1H, m), 7.42-7.40 (1H, m).

[0575] Present compound 80: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.80-7.78 (1H, m), 7.69-7.64 (1H, m).

[0576] Present compound 81: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.12-8.11 (1H, m), 7.12-7.09 (1H, m).

[0577] Present compound 137: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.87 (2H, d), 7.42 (2H, d), 7.22 (1H, t), 7.11-7.06 (4H, m).

[0578] Present compound 138: .sup.1H-NMR (CDCl.sub.3) ?: 9.00 (1H, d), 8.73 (2H, d), 8.19 (1H, s), 7.73 (1H, d).

[0579] Present compound 139: .sup.1H-NMR (CDCl.sub.3) ?: 8.97 (1H, d), 8.75 (2H, s), 8.17 (1H, s), 7.97 (1H, d).

[0580] Present compound 140: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.18-8.09 (2H, m), 7.89 (1H, d).

[0581] Present compound 145: .sup.1H-NMR (CDCl.sub.3) ?: 8.73 (2H, d), 7.79 (1H, d), 7.69 (1H, s), 7.58-7.52 (1H, m), 7.36 (1H, d), 6.59 (1H, t).

Preparation Example 1-2

[0582] The compounds which were prepared according to the Preparation Example 1 and their physical property value are shown below.

[0583] A compound represented by formula (B-2):

##STR00036##

wherein Q represents any substituents described in [Table B-2A] and [Table B-2B].

TABLE-US-00012 TABLE B-2A Comp Q 82 [00037] embedded image 84 [00038] 86 [00039] 88 [00040]

TABLE-US-00013 TABLE B-2B Comp Q 83 [00041] embedded image 85 [00042] 87 [00043]

[0584] Present compound 82: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.72 (1H, dd), 7.60 (1H, dd), 7.19 (1H, dd).

[0585] Present compound 83: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.66 (1H, dd), 7.13 (1H, dd), 6.62 (1H, dd).

[0586] Present compound 84: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.67-7.66 (1H, m), 7.52-7.50 (1H, m).

[0587] Present compound 85: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.72 (1H, d), 7.60 (1H, d), 7.49-7.47 (2H, m), 7.38-7.34 (1H, m).

[0588] Present compound 86: .sup.1H-NMR (CDCl.sub.3) ?: 8.69 (2H, s), 8.13 (1H, s), 2.57 (3H, s).

[0589] Present compound 87: .sup.1H-NMR (CDCl.sub.3) ?: 8.69 (2H, s), 7.49 (1H, d), 6.78 (1H, d), 4.03 (3H, s)

[0590] Present compound 88: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.28 (1H, s), 7.12 (1H, s), 3.98 (3H, s).

[0591] A compound represented by formula (B-3):

##STR00044##

wherein a combination of G.sup.1, G.sup.2, R.sup.1b, R.sup.18a, R.sup.18b, and R.sup.18c represents any combinations described in [Table B-3A].

TABLE-US-00014 TABLE B-3A Comp G.sup.1 G.sup.2 R.sup.1b R.sup.18a R.sup.18b R.sup.18c 89 CCl N [00045] embedded image CF.sub.3 H H 90 CH CH Cl CF.sub.3 H H 91 CH CH Cl OCF.sub.3 H H 92 CH CH Br CF.sub.3 H H 93 CH CH NO.sub.2 CF.sub.3 H H 94 CH CH CF.sub.3 CF.sub.3 H H 95 CH CBr Br H H H 96 CH CB Br CF.sub.3 H H 97 CH CB Br OCF.sub.3 H H 143 CH CB Br F F H 146 CH CB Br H F H 147 CH CB Br F Br H 148 CH CF Cl CF.sub.3 H H 149 CH CF Cl F F H

[0592] Present compound 89: .sup.1H-NMR (CDCl.sub.3) ?: 9.00 (1H, s), 8.24 (1H, s), 8.14 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 5.92 (1H, s), 4.25-4.23 (2H, m), 3.94-3.91 (2H, m), 2.17-2.14 (1H, m), 1.41 (1H, m).

[0593] Present compound 90: .sup.1H-NMR (CDCl.sub.3) ?: 8.81 (1H, s), 8.66 (1H, d), 8.20 (1H, s), 8.12 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 7.58 (1H, d).

[0594] Present compound 91: .sup.1H-NMR (CDCl.sub.3) (?: 8.80 (1H, s), 8.65 (1H, d), 7.90-7.85 (1H, m), 7.79 (1H, s), 7.62-7.56 (2H, m), 7.47-7.42 (1H, m).

[0595] Present compound 92: .sup.1H-NMR (CDCl.sub.3) ?: 8.94 (1H, s), 8.69 (1H, d), 8.20 (1H, s), 8.12 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 7.56 (1H, d).

[0596] Present compound 93: .sup.1H-NMR (CDCl.sub.3) ?: 9.17 (1H, d), 8.93 (1H, dd), 8.18 (1H, s), 8.11 (1H, d), 7.92 (1H, dd), 7.88 (1H, d), 7.72-7.70 (1H, m).

[0597] Present compound 94: .sup.1H-NMR (CDCl.sub.3) ?: 9.11 (1H, s), 8.96 (1H, d), 8.17 (1H, s), 8.11 (1H, d), 7.85 (1H, d), 7.79 (1H, d), 7.70-7.68 (1H, m).

[0598] Present compound 95: .sup.1H-NMR (CDCl.sub.3) ?: 8.84 (2H, s), 7.93 (2H, d), 7.59-7.51 (3H, m).

[0599] Present compound 96: .sup.1H-NMR (CDCl.sub.3) ?: 8.86 (2H, s), 8.20 (1H, s), 8.11 (1H, d), 7.84 (1H, d), 7.69 (1H, t).

[0600] Present compound 97: .sup.1H-NMR (CDCl.sub.3) ?: 8.85 (2H, s), 7.87 (1H, d), 7.78 (1H, s), 7.58 (1H, t), 7.44 (1H, d).

[0601] Present compound 143: .sup.1H-NMR (CDCl.sub.3) ?: 8.85 (2H, s), 7.79-7.69 (2H, m), 7.38-7.30 (1H, m).

[0602] Present compound 146: .sup.1H-NMR (CDCl.sub.3) ?: 8.85 (2H, s), 7.96-7.92 (2H, m), 7.25-7.21 (2H, m).

[0603] Present compound 147: .sup.1H-NMR (CDCl.sub.3) ?: 8.86 (2H, s), 7.77-7.73 (1H, m), 7.69-7.66 (1H, m), 7.62-7.59 (1H, m).

[0604] Present compound 148: .sup.1H-NMR (CDCl.sub.3) ?: 8.68 (1H, s), 8.64 (1H, s), 8.20 (1H, s), 8.11 (1H, d), 7.86 (1H, d), 7.73-7.67 (1H, m).

[0605] Present compound 149: .sup.1H-NMR (CDCl.sub.3) ?: 8.67 (1H, s), 8.63 (1H, s), 7.78-7.68 (2H, m), 7.39-7.31 (1H, m).

Preparation Example 2

[0606] A mixture of the present compound 10 193 mg, 4-fluorophenyl boronic acid 80 mg, and potassium carbonate 212 mg, tris(dibenzylideneacetone)dipalladium (0) 46 mg, 2-dicyclohexylphoshino-2,6-dimethoxy biphenyl 41 mg, toluene 3 mL, and water 1 mL was stirred at 65? C. for 4 hours. Water was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain the present compound 98 represented by the following formula 90 mg.

##STR00046##

[0607] Present compound 98: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.09 (1H, s), 7.89 (1H, d), 7.75 (1H, d), 7.62-7.57 (3H, m), 7.18-7.15 (2H, m).

Preparation Example 2-1

[0608] The compounds which were prepared according to the Preparation Example 2 and their physical property value are shown below.

[0609] A compound represented by formula (B-3):

##STR00047##

wherein a combination of G.sup.5, R.sup.18a, R.sup.13b and R.sup.18c represents any combinations described in [Table B-3B].

TABLE-US-00015 TABLE B-3B Comp G.sup.5 R.sup.18a R.sup.18b R.sup.18c 99 CH H H [00048] embedded image 100 CH H H C-Pr

[0610] Present compound 99: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 8.21 (1H, s), 8.00 (1H, s), 7.89-7.85 (2H, m), 7.69 (1H, s), 7.66-7.64 (1H, m).

[0611] Present compound 100: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, d), 7.69 (1H, d), 7.60 (1H, s), 7.41-7.39 (1H, m), 7.29-7.27 (1H, m), 1.97-1.95 (1H, m), 1.05-1.04 (2H, m), 0.77-0.75 (2H, m).

Preparation Example 3

[0612] A mixture of the present compound 9 387 mg, bis(pinacolato)diboron 508 mg, potassium acetate 294 mg, dichloro(1,1-bis(diphenylphoshino)ferrocene palladium (II) 36 mg, and toluene 3 mL was stirred at 80? C. for 6 hours. Water was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. Sodium acetate 615 mg, water 5 mL and THF 5 mL were added to the resulting mixture successively. The resulting mixture was cooled to 0? C., and 30% aqueous hydrogen peroxide solution 0.11 mL was added thereto, and the mixture was stirred at room temperature for 9 hours. Aqueous sodium thiosulfate solution was added to the resulting mixture, and the mixture was extracted with chloroform. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure to obtain the present compound 101 150 mg as a crude product.

##STR00049##

[0613] Present compound 101: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.52-7.49 (1H, m), 7.40-7.38 (2H, m), 7.06-7.04 (1H, m), 5.20 (1H, s).

Preparation Example 3-1

[0614] The compounds which were prepared according to the Preparation Example 3 and their physical property value are shown below.

[0615] A compound represented by formula (B-3):

##STR00050##

wherein a combination of G.sup.5, R.sup.18a, R.sup.18b and R.sup.18c represents any combinations described in [Table B-4A].

TABLE-US-00016 TABLE B-4A Comp G.sup.5 R.sup.18a R.sup.18b R.sup.18c 102 CH H OH H 103 CH OH H F 104 CH OH H Cl 105 CF H F OH

[0616] Present compound 102: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.82 (2H, d), 6.96 (2H, d), 5.44 (1H, s).

[0617] Present compound 103: LCMS: 340 [M?H].sup.?, RT=1.86 min.

[0618] Present compound 104: LCMS: 356 [M?H].sup.?, RT=1.97 min.

[0619] Present compound 105: LCMS: 358 [M?H].sup.?, RT=1.66 min.

Preparation Example 4

[0620] A mixture of the present compound 101 (which was obtained in the Preparation Example 3) as crude product 100 mg cesium carbonate 163 mg, DMF 2 mL and iodomethane 0.04 mL was stirred at room temperature for 1 hour. Water was added to the resulting mixture, and the mixture was extracted with 2-methoxy-2-methylpropane. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain the present compound 106 represented by the following formula 60 mg.

##STR00051##

[0621] Present compound 106: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.49 (1H, d), 7.41-7.39 (2H, m), 7.11-7.09 (1H, m), 4.09 (2H, q), 1.45 (3H, t).

Preparation Example 4-1

[0622] The compounds which were prepared according to the reparation Example 4 and their physical property value are shown below.

[0623] A compound represented by formula (B-3):

##STR00052##

wherein a combination of G.sup.5, R.sup.18a, R.sup.18b and R.sup.18c represents any combinations described in [Table B-5A].

TABLE-US-00017 TABLE B-5A Comp G.sup.5 R.sup.18a R.sup.18b R.sup.18c 107 CH H OEt H 108 CH OCH.sub.2CF.sub.3 H H 109 CH OCH.sub.2CF.sub.2CF.sub.3 H H 110 CH OCH.sub.2CF.sub.3 H F 111 CH OCH.sub.2CF.sub.3 H Cl 112 CF H F OCH.sub.2CF.sub.3

[0624] Present compound 107: .sup.1H-NMR (CDCl.sub.3) ?: 8.69 (2H, s), 7.84 (2H, d), 6.99 (2H, d), 4.11 (2H, q), 1.46 (3H, t).

[0625] Present compound 108: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.62 (1H, d), 7.52-7.46 (2H, m), 7.18 (1H, dd), 4.42 (2H, t).

[0626] Present compound 109: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.63 (1H, d), 7.52-7.46 (2H, m), 7.18 (1H, dd), 4.49 (2H, t).

[0627] Present compound 110: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.35-7.33 (1H, m), 7.28-7.27 (1H, m), 6.91-6.89 (1H, m), 4.42 (2H, q).

[0628] Present compound 111: .sup.1H-NMR (CDCl.sub.3) ?: 8.72 (2H, s), 7.62-7.61 (1H, m), 7.36-7.35 (1H, m), 7.18-7.17 (1H, m), 4.42 (2H, q).

[0629] Present compound 112: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.55-7.53 (1H, m), 7.13-7.10 (1H, m), 4.46 (2H, q).

Preparation Example 5

[0630] The present compound 31 700 mg was added to a mixture of iron powder 990 mg, ethanol 5 mL and acetic acid 0.29 mL at 90? C., and the mixture was stirred at 90? C. for 5 hours. The resulting mixture was filtered through Celite (registered trademark), and aqueous saturated sodium hydrocarbonate solution was added to the filtrates, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure to obtain the present compound 113 represented by the following formula 170 mg.

##STR00053##

[0631] Present compound 113: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.29-7.28 (2H, m), 7.19-7.19 (1H, m), 6.86-6.86 (1H, m), 3.87 (2H, s).

Preparation Example 5-1

[0632] The compounds which were prepared according to the Preparation Example 5 and their physical property value are shown below.

##STR00054##

[0633] Present compound 114: .sup.1H-NMR (CDCl.sub.3) ?: 8.68 (2H, s), 7.70 (2H, d), 6.73 (2H, d), 4.12 (2H, d).

Preparation Example 6

[0634] Acetyl chloride 0.03 mL was added to a mixture of the present compound 113 120 mg, triethylamine 0.06 mL, and chloroform 1 mL at 0? C., and the mixture was stirred at room temperature for 3 hours. Water was added to the resulting mixture, and the mixture was extracted with chloroform. The resulting organic layer was dried over anhydrous sodium sulfate and concentrated under reduced pressure to obtain the present compound 115 represented by the following formula 120 mg.

##STR00055##

[0635] Present compound 115: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 8.01 (1H, s), 7.80 (1H, d), 7.66 (1H, d), 7.49-7.47 (1H, m), 7.26 (1H, s), 2.22 (3H, s).

Preparation Example 6-1

[0636] The compounds which were prepared according to the Preparation Example 6 and their physical property value are shown below.

##STR00056##

[0637] Present compound 116: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (2H, s), 7.87 (2H, d), 7.69 (2H, d), 7.30 (1H, s), 2.24 (3H, s).

Preparation Example 7

[0638] A mixture or the present compound 92 386 mg, 2-(propen-2-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 300 mg, tripotassium phosphate 424 mg, tris(dibenzylideneacetone)dipalladium (0) 45 mg, toluene 10 mL, and water 1 mL was stirred at 60? C. for 6 hours. Water was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate, and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain the present compound 117 represented by the following formula 35 mg.

##STR00057##

[0639] Present compound 117: .sup.1H-NMR (CDCl.sub.3) ?: 8.65-8.65 (2H, m), 8.16 (1H, s), 8.08 (1H, d), 7.83 (1H, d), 7.69-7.67 (1H, m), 7.56 (1H, d), 5.26 (1H, s), 5.00 (1H, s), 2.13 (3H, s).

Preparation Example 7-1

[0640] The compounds which were prepared according to the Preparation Example 7 and their physical property value are shown below.

[0641] A compound represented by formula (B-4):

##STR00058##

wherein a combination of G.sup.1, R.sup.1b, G.sup.2, G.sup.3, G.sup.5, R.sup.18a, R.sup.18b and R.sup.18c represents any combinations described in [Table B-4B].

TABLE-US-00018 TABLE B-4B Comp G.sup.1 R.sup.1b G.sup.2 G.sup.3 G.sup.5 R.sup.18a R.sup.18b R.sup.18c 118 CH CH?CH.sub.2 CH CH CH H H CF.sub.3 119 CH Me CH CH CH H H CF.sub.3 120 CH CPr CH CH CH H H CF.sub.3 121 CH Ph CH CH CH H H CF.sub.3 122 CH [00059] embedded image CH CH CH H H CF.sub.3 123 CH [00060] CH CH CH H H CF.sub.3 124 CH CH?CH.sub.2 CCH?CH.sub.2 CH CH H H CF.sub.3 125 CH Me CMe CH CH H H CF.sub.3 126 CH CMe?CH.sub.2 CCMe?CH.sub.2 CH CH H H OCF.sub.3 127 CH [00061] [00062] CH CH H H OCF.sub.3 128 CH Me CMe CH CH H H OCF.sub.3

[0642] Present compound 118: .sup.1H-NMR (CDCl.sub.3) ?: 8.92 (1H, s), 8.65 (1H, d), 8.19 (1H, s), 8.11 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 7.53 (1H, d), 6.97 (1H, dd), 5.87 (1H, d), 5.53 (1H, d).

[0643] Present compound 119: .sup.1H-NMR (CDCl.sub.3) ?: 8.63 (1H, s), 8.59 (1H, d), 8.19 (1H, s), 8.11 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 7.50 (1H, d), 2.47 (3H, s).

[0644] Present compound 120: .sup.1H-NMR (CDCl.sub.3) ?: 8.58 (1H, d), 8.55 (1H, s), 8.20 (1H, s), 8.11 (1H, d), 7.83 (1H, d), 7.71-7.69 (1H, m), 7.44 (1H, d), 2.19-2.16 (1H, m), 1.02-1.00 (2H, m), 0.75-0.72 (2H, m).

[0645] Present compound 121: .sup.1H-NMR (CDCl.sub.3) ?: 8.76-8.75 (2H, m), 7.93 (1H, s), 7.87 (1H, d), 7.78 (1H, d), 7.66 (1H, d), 7.62-7.60 (1H, m), 7.46-7.34 (5H, m).

[0646] Present compound 122: .sup.1H-NMR (CDCl.sub.3) ?: 8.76 (1H, d), 8.64 (1H, s), 7.78-7.75 (4H, m), 7.58-7.56 (1H, m), 7.33-7.28 (2H, m), 7.22 (1H, dd), 7.16-7.14 (1H, m), 2.14 (3H, s).

[0647] Present compound 123: .sup.1H-NMR (CDCl.sub.3) ?: 8.70 (1H, d), 8.61 (1H, d), 8.17 (1H, s), 8.08 (1H, d), 7.83 (1H, dd), 7.69-7.67 (1H, m), 7.49-7.49 (1H, m), 5.94-5.91 (1H, m), 2.64-2.59 (2H, m), 2.53-2.48 (2H, m), 2.02-2.00 (2H, m).

[0648] Present compound 124: .sup.1H-NMR (CDCl.sub.3) ?: 8.83 (2H, s), 8.19 (1H, s), 8.10 (1H, d), 7.83 (1H, d), 7.69-7.67 (1H, m), 6.66 (2H, dd), 5.89 (2H, d), 5.52 (2H, d).

[0649] Present compound 125: .sup.1H-NMR (CDCl.sub.3) ?: 8.49 (2H, s), 8.18 (1H, s), 8.10 (1H, d), 7.83 (1H, d), 7.68 (1H, t), 2.31 (6H, s).

[0650] Present compound 126: .sup.1H-NMR (CDCl.sub.3) ?: 8.71 (2H, s), 7.88 (1H, d), 7.79 (1H, s), 7.58 (1H, t), 7.43 (1H, d), 6.45-6.19 (4H, m), 1.89 (6H, dd).

[0651] Present compound 127: LCMS: 404 [M+H].sup.+, RT=2.22 min.

[0652] Present compound 128: .sup.1H-NMR (CDCl.sub.3) ?: 8.49 (2H, s), 7.86 (1H, d), 7.77 (1H, s), 7.58 (1H, t), 7.43 (1H, d), 2.31 (6H, s).

Preparation Example 8

[0653] A mixture of the present compound 118 100 mg, ethanol 5 mL, and palladium carbon 5 mg was stirred at room temperature under hydrogen atmosphere for 6 hours. The resulting mixture was filtered, and the filtrates were concentrated under reduced pressure to obtain the present compound 130 represented by the following formula 100 mg.

##STR00063##

[0654] Present compound 130: .sup.1H-NMR (CDCl.sub.3) ?: 8.67 (1H, s), 8.60 (1H, d), 8.18 (1H, s), 8.10 (1H, d), 7.84 (1H, d), 7.70-7.68 (1H, m), 7.48 (1H, d), 2.87 (2H, q), 1.30 (3H, t).

Preparation Example 8-1

[0655] The compounds which were prepared according to the Preparation Example 8 and their physical property value are shown below.

[0656] A compound represented by formula (B-5):

##STR00064##

wherein a combination of G.sup.1, R.sup.1b, G.sup.2, G.sup.3, G.sup.5, R.sup.18a, R.sup.18b and R.sup.18c represents any combinations described in [Table B-5B].

TABLE-US-00019 TABLE B-5B Comp G.sup.1 R.sup.1b G.sup.2 G.sup.3 G.sup.5 R.sup.18a R.sup.18b R.sup.18c 131 CH Et CEt CH CH H H CF.sub.3 132 CH Et CEt CH CH H H OCF.sub.3 133 CH iPr CiPr CH CH H H OCF.sub.3 134 CH Pr Pr CH CH H H OCF.sub.3

[0657] Present compound 131: .sup.1H-NMR (CDCl.sub.3) ?: 8.54 (2H, s), 8.19 (1H, s), 8.10 (1H, d), 7.83 (1H, d), 7.69 (1H, d), 2.66 (4H, q), 1.25 (6H, t).

[0658] Present compound 132: .sup.1H-NMR (CDCl.sub.3) ?: 8.54 (2H, s), 7.86 (1H, d), 7.77 (1H, s), 7.58 (1H, t), 7.43 (1H, d), 2.65 (4H, q), 1.24 (6H, t).

[0659] Present compound 133: .sup.1H-NMR (CDCl.sub.3) ?: 8.61 (2H, s), 7.85 (1H, d), 7.76 (1H, s), 7.57 (1H, t), 7.42 (1H, d), 2.93-2.86 (2H, m), 1.34-1.29 (12H, m).

[0660] Present compound 134: .sup.1H-NMR (CDCl.sub.3) ?: 8.50 (2H, s), 7.86 (1H, d), 7.77 (1H, s), 7.58 (1H, t), 7.43 (1H, d), 2.65-2.53 (4H, m), 1.68-1.57 (4H, m), 0.92 (6H, t).

Preparation Example 9

[0661] A mixture of the present compound 12 392 mg, chloroform 5 mL, and m-chloroperoxybenzoic acid 246 mg was stirred at room temperature for 6 hours. The resulting mixture was washed with aqueous sodium thiosulfate solution and aqueous sodium hydrocarbonate solution successively. The resulting organic layer was dried over anhydrous sodium sulfate and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain the present compound 135 represented by the following formula 240 mg.

##STR00065##

[0662] Present compound 135: .sup.1H-NMR (CDCl.sub.3) ?: 8.29 (2H, s), 7.85 (1H, d), 7.76 (1H, s), 7.59 (1H, t), 7.44 (1H, d).

Preparation Example 10

[0663] Thiophosgene 0.15 mL was added to a mixture of the intermediate compound 20 348 mg, triethylamine 0.4 mL, and THF 5 mL, and the mixture was stirred at room temperature for 6 hours. Aqueous saturated sodium hydrocarbonate solution was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was dried over anhydrous sodium sulfate and concentrated under reduced pressure. The resulting residue was subjected to a silica gel column chromatography (ethyl acetate:hexane=30:70) to obtain the present compound 136 represented by the following formula 150 mg.

##STR00066##

[0664] Present compound 136: .sup.1H-NMR (CDCl.sub.3) ?: 8.76 (2H, s), 8.26 (1H, s), 8.18 (1H, d), 7.88 (1H, d), 7.71 (1H, t).

[0665] Next, examples of the present compounds which are prepared according to any one of the Preparation Examples described in Working Examples and the Processes described herein are indicated below.

[0666] A compound represented by formula (L-1):

##STR00067##

(hereinafter, referred to as compound (L-1)) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, and A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any substituents described in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX1).

TABLE-US-00020 TABLE L1 CCF.sub.3 CCHF.sub.2 CCH.sub.2CF.sub.3 CCF.sub.2CF.sub.3 CCH.sub.2CF.sub.2CF.sub.3 CCF.sub.2CF.sub.2CF.sub.3 CCF.sub.2CF.sub.2CF.sub.2CF.sub.3 CCF.sub.2CF.sub.2CF.sub.2CF.sub.2CF.sub.3 COCF.sub.3 COCHF.sub.2 COCH.sub.2CF.sub.3 COCH.sub.2CHF.sub.2 COCF.sub.2CF.sub.3 COCH(CH.sub.3)CF.sub.3 COCH.sub.2CF.sub.2CHF.sub.2 COCH.sub.2CF.sub.2CF.sub.3 COCF.sub.2CF.sub.2CF.sub.3 COCF.sub.2CHF.sub.2 COCH.sub.2CF.sub.2CHFCF.sub.3 COCH.sub.2CF.sub.2CF.sub.2CF.sub.3 COCF.sub.2CF.sub.2CF.sub.2CF.sub.3 COCH.sub.2(2,2-F.sub.2cPr) COCH.sub.2(1-CF.sub.3cPr) COS(O).sub.2CF.sub.3 COS(O).sub.2CF.sub.2CF.sub.3 COS(O).sub.2CF.sub.2CF.sub.2CF.sub.3

TABLE-US-00021 TABLE L2 CSCF.sub.3 CSCH.sub.2CF.sub.3 CSCF.sub.2CF.sub.3 CSCH.sub.2CF.sub.2CF.sub.3 CSCF.sub.2CF.sub.2CF.sub.3 CSCH.sub.2CF.sub.2CF.sub.2CF.sub.3 CSCF.sub.2CF.sub.2CF.sub.2CF.sub.3 CS(O)CF.sub.3 CS(O)CH.sub.2CF.sub.3 CS(O)CF.sub.2CF.sub.3 CS(O)CH.sub.2CF.sub.2CF.sub.3 CS(O)CF.sub.2CF.sub.2CF.sub.3 CS(O)CH.sub.2CF.sub.2CF.sub.2CF.sub.3 CS(O)CF.sub.2CF.sub.2CF.sub.2CF.sub.3 CS(O).sub.2CF.sub.3 CS(O).sub.2CH.sub.2CF.sub.3 CS(O).sub.2CF.sub.2CF.sub.3 CS(O).sub.2CH.sub.2CF.sub.2CF.sub.3 CS(O).sub.2CF.sub.2CF.sub.2CF.sub.3 CF CCl CBr CI COCH.sub.3 COCH.sub.2CH.sub.3 COCH(CH.sub.3).sub.2

TABLE-US-00022 TABLE L3 COCH.sub.2CH.sub.2CH.sub.3 COCH.sub.2CH.sub.2CH.sub.2CH.sub.3 COCH.sub.2C(CH.sub.3).sub.2 CCH.sub.3 CCH.sub.2CH.sub.3 CC(CH.sub.3).sub.2 CCH.sub.2CH.sub.2CH.sub.3 CCH.sub.2CH.sub.2CH.sub.2CH.sub.3 CC(CH.sub.3).sub.3 CCH?CH.sub.2 [00068] embedded image [00069] CCCH.sub.3?CH.sub.2 C-2-FPh C-3-FPh C-4-FPh C-2-ClPh C-3-ClPh C-4-ClPh C-2,6-F.sub.2Ph C-3,5-F.sub.2Ph C-2,4-F.sub.2Ph C-2,4,6-F.sub.3Ph C-2,6-Cl.sub.2Ph C-3,5-Cl.sub.2Ph C-2,4-Cl.sub.2Ph

[0667] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CR, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX2).

[0668] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CR, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX3).

[0669] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX4)

[0670] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX5).

[0671] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX6)

[0672] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX7).

[0673] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX8)

[0674] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX9).

[0675] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX10).

[0676] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX11).

[0677] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX12).

[0678] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX13).

[0679] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX14).

[0680] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX15).

[0681] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX16).

[0682] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX17).

[0683] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX18).

[0684] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1crepresents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX19).

[0685] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX20).

[0686] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX21).

[0687] A present compound (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX22).

[0688] A present compound (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX23).

[0689] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX24).

[0690] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX25).

[0691] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX26).

[0692] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX27).

[0693] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX28).

[0694] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX29).

[0695] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX30).

[0696] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX31).

[0697] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX32).

[0698] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX33).

[0699] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2, A, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX34).

[0700] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX35).

[0701] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX36).

[0702] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX37).

[0703] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX38).

[0704] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX39).

[0705] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX40).

[0706] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX41).

[0707] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX42).

[0708] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX43).

[0709] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX44).

[0710] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX45).

[0711] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX46).

[0712] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX47).

[0713] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX48).

[0714] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX49).

[0715] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX50).

[0716] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX51).

[0717] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX52).

[0718] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX53).

[0719] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX54).

[0720] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX55).

[0721] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX56).

[0722] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX57).

[0723] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX58).

[0724] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX59).

[0725] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX60).

[0726] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX61).

[0727] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX62).

[0728] A present compound (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX63).

[0729] A present compound (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX64).

[0730] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX65).

[0731] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX66).

[0732] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX67).

[0733] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX68).

[0734] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX69).

[0735] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX70).

[0736] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX71).

[0737] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX72).

[0738] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX73).

[0739] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX74).

[0740] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX75).

[0741] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX76).

[0742] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX77).

[0743] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX78).

[0744] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX79).

[0745] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX80).

[0746] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX81).

[0747] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX82).

[0748] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX83).

[0749] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX84).

[0750] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX85).

[0751] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX86).

[0752] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX87).

[0753] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX88).

[0754] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX89).

[0755] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX90).

[0756] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX91).

[0757] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX92).

[0758] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX93).

[0759] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX94).

[0760] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX95).

[0761] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX96).

[0762] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX97).

[0763] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX98).

[0764] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX99).

[0765] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX100).

[0766] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX101).

[0767] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX102).

[0768] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX103).

[0769] A present compound (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX104).

[0770] A present compound (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX105).

[0771] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX106).

[0772] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX107).

[0773] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX108).

[0774] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX109).

[0775] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX110).

[0776] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX111).

[0777] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX112).

[0778] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX113).

[0779] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX114).

[0780] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX115).

[0781] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX116).

[0782] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX117).

[0783] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX118).

[0784] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX119).

[0785] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX120).

[0786] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX121).

[0787] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX122).

[0788] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX123).

[0789] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.5, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX124).

[0790] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX125).

[0791] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX126).

[0792] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX127).

[0793] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX128).

[0794] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX129).

[0795] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX130).

[0796] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX131).

[0797] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3](hereinafter, referred to as Compound class SX132).

[0798] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX133).

[0799] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX134).

[0800] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX135).

[0801] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX136).

[0802] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX137).

[0803] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX138).

[0804] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX139).

[0805] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX140).

[0806] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX141).

[0807] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX142).

[0808] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX143).

[0809] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX144).

[0810] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX145).

[0811] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX146).

[0812] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX147).

[0813] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX148).

[0814] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX149).

[0815] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX150).

[0816] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX151).

[0817] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX152).

[0818] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX153).

[0819] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX154).

[0820] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX155).

[0821] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX156).

[0822] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX157).

[0823] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX158).

[0824] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX159).

[0825] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX160).

[0826] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX161).

[0827] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX162).

[0828] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX163).

[0829] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX164).

[0830] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX165).

[0831] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX166).

[0832] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX167).

[0833] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX168).

[0834] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX169).

[0835] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX170).

[0836] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX171).

[0837] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX172).

[0838] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX173).

[0839] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX174).

[0840] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX175).

[0841] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX176).

[0842] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX177).

[0843] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX178).

[0844] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX179).

[0845] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX180).

[0846] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX181).

[0847] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX182).

[0848] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX183).

[0849] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX184).

[0850] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX185).

[0851] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX186).

[0852] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX187).

[0853] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX188).

[0854] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX189).

[0855] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX190).

[0856] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX191).

[0857] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.1, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX192).

[0858] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX193).

[0859] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX194).

[0860] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX195).

[0861] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX196).

[0862] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX197).

[0863] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX198).

[0864] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX199).

[0865] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX200).

[0866] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX201).

[0867] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX202).

[0868] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX203).

[0869] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX204).

[0870] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX205).

[0871] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX206).

[0872] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX207).

[0873] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX208).

[0874] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX209).

[0875] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX210).

[0876] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX211).

[0877] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX212).

[0878] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX213).

[0879] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX214).

[0880] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX215).

[0881] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX216).

[0882] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX217).

[0883] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX218).

[0884] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX219).

[0885] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX220).

[0886] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX221).

[0887] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX222).

[0888] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX223).

[0889] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX224).

[0890] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX225).

[0891] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX226).

[0892] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX227).

[0893] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX228).

[0894] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX229).

[0895] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX230).

[0896] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX231).

[0897] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX232).

[0898] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX233).

[0899] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX234).

[0900] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX235).

[0901] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX236).

[0902] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX237).

[0903] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX238).

[0904] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX239).

[0905] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX240).

[0906] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX241).

[0907] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 [Table L3] (hereinafter, referred to as Compound class SX242).

[0908] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.1 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX243).

[0909] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX244).

[0910] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX245).

[0911] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX246).

[0912] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX247).

[0913] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX248).

[0914] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX249).

[0915] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX250).

[0916] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX251).

[0917] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX252).

[0918] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX253).

[0919] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX254).

[0920] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX255).

[0921] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX256).

[0922] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX257).

[0923] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX258).

[0924] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX259).

[0925] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX260).

[0926] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX261).

[0927] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX262).

[0928] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX263).

[0929] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX264).

[0930] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX265).

[0931] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX266).

[0932] A present compound (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX267).

[0933] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX268).

[0934] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX269).

[0935] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX270).

[0936] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX271).

[0937] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX272).

[0938] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX273).

[0939] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX274).

[0940] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX275).

[0941] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX276).

[0942] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX277).

[0943] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX278).

[0944] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX279).

[0945] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX280).

[0946] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX281).

[0947] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX282).

[0948] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX283).

[0949] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX284).

[0950] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX285).

[0951] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX286).

[0952] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX287).

[0953] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX288).

[0954] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX289).

[0955] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX290).

[0956] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX291).

[0957] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX292).

[0958] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX293).

[0959] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX294).

[0960] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX295).

[0961] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX296).

[0962] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX297).

[0963] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX298).

[0964] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX299).

[0965] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX300).

[0966] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX301).

[0967] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX302).

[0968] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX303).

[0969] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX304).

[0970] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX305).

[0971] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX306).

[0972] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX307).

[0973] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX308).

[0974] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX309).

[0975] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX310).

[0976] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX311).

[0977] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX312).

[0978] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX313).

[0979] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX314).

[0980] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX315).

[0981] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX316).

[0982] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX317).

[0983] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX318).

[0984] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX319).

[0985] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX320).

[0986] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX321).

[0987] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX322).

[0988] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX323).

[0989] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX324).

[0990] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX325).

[0991] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX326).

[0992] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX327).

[0993] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX328).

[0994] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX329).

[0995] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX330).

[0996] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX331).

[0997] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX332).

[0998] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX333).

[0999] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX334).

[1000] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX335).

[1001] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX336).

[1002] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX337).

[1003] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX338).

[1004] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX339).

[1005] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX340).

[1006] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX341).

[1007] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX342).

[1008] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX343).

[1009] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX344).

[1010] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX345).

[1011] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX346).

[1012] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX347).

[1013] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX348).

[1014] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX349).

[1015] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX350).

[1016] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX351).

[1017] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX352).

[1018] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX353).

[1019] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX354).

[1020] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX355).

[1021] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX356).

[1022] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX357).

[1023] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX358).

[1024] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX359).

[1025] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX360).

[1026] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX361).

[1027] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX362).

[1028] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX363).

[1029] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX364).

[1030] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX365).

[1031] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX366).

[1032] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX367).

[1033] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX368).

[1034] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX369).

[1035] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX370).

[1036] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX371).

[1037] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX372).

[1038] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX373).

[1039] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX374).

[1040] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX375).

[1041] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX376).

[1042] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX377).

[1043] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX378).

[1044] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX379).

[1045] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX380).

[1046] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX381).

[1047] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX382).

[1048] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX383).

[1049] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX384).

[1050] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX385).

[1051] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX386).

[1052] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX387).

[1053] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX388).

[1054] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX389).

[1055] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX390).

[1056] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX391).

[1057] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX392).

[1058] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX393).

[1059] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX394).

[1060] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX395).

[1061] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX396).

[1062] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX397).

[1063] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX398).

[1064] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX399).

[1065] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX400).

[1066] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX401).

[1067] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX402).

[1068] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX403).

[1069] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX404).

[1070] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX405).

[1071] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX406).

[1072] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX407).

[1073] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX408).

[1074] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX409).

[1075] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX410).

[1076] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX411).

[1077] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX412).

[1078] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX413).

[1079] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX414).

[1080] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX415).

[1081] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX416).

[1082] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX417).

[1083] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX418).

[1084] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX419).

[1085] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX420).

[1086] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX421).

[1087] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX422).

[1088] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX423).

[1089] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX424).

[1090] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX425).

[1091] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX426).

[1092] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX427).

[1093] A present compound (L-1) wherein Rib represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX428).

[1094] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX429).

[1095] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX430).

[1096] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX431).

[1097] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX432).

[1098] A present compound (L-1) wherein Rib represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX433).

[1099] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX434).

[1100] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX435).

[1101] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.5 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX436).

[1102] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX437).

[1103] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX438).

[1104] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX439).

[1105] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX440).

[1106] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.5 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX441).

[1107] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX442).

[1108] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX443).

[1109] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX444).

[1110] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX445).

[1111] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX446).

[1112] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX447).

[1113] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX448).

[1114] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX449).

[1115] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX450).

[1116] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX451).

[1117] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX452).

[1118] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX453).

[1119] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX454).

[1120] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX455).

[1121] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX456).

[1122] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.J represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX457).

[1123] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX458).

[1124] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX459).

[1125] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX460).

[1126] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX461).

[1127] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX462).

[1128] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX463).

[1129] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX464).

[1130] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX465).

[1131] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX466).

[1132] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX467).

[1133] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX468).

[1134] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX469).

[1135] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX470).

[1136] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX471).

[1137] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX472).

[1138] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX473).

[1139] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX474).

[1140] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX475).

[1141] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX476).

[1142] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX477).

[1143] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX478).

[1144] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX479).

[1145] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX480).

[1146] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX481).

[1147] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX482).

[1148] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX483).

[1149] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX484).

[1150] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX485).

[1151] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX486).

[1152] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX487).

[1153] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX488).

[1154] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX489).

[1155] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX490).

[1156] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX491).

[1157] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX492).

[1158] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.11 represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX493).

[1159] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX494).

[1160] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX495).

[1161] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX496).

[1162] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX497).

[1163] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX498).

[1164] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX499).

[1165] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX500).

[1166] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX501).

[1167] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX502).

[1168] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX503).

[1169] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX504).

[1170] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX505).

[1171] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX506).

[1172] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX507).

[1173] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX508).

[1174] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX509).

[1175] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX510).

[1176] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX511).

[1177] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX512).

[1178] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX513).

[1179] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX514).

[1180] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX515).

[1181] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.5 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX516).

[1182] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX517).

[1183] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX518).

[1184] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX519).

[1185] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX520).

[1186] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX521).

[1187] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX522).

[1188] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX523).

[1189] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX524).

[1190] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX525).

[1191] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX526).

[1192] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX527).

[1193] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX528).

[1194] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX529).

[1195] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX530).

[1196] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX531).

[1197] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX532).

[1198] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX533).

[1199] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX534).

[1200] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX535).

[1201] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX536).

[1202] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX537).

[1203] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX538).

[1204] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX539).

[1205] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX540).

[1206] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX541).

[1207] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX542).

[1208] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX543).

[1209] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX544).

[1210] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX545).

[1211] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX546).

[1212] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX547).

[1213] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX548).

[1214] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX549).

[1215] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX550).

[1216] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX551).

[1217] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX552).

[1218] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX553).

[1219] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX554).

[1220] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX555).

[1221] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents any one group selected from a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX556).

[1222] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX557).

[1223] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX558).

[1224] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX559).

[1225] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX560).

[1226] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX561).

[1227] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX562).

[1228] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX563).

[1229] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX564).

[1230] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX565).

[1231] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX566).

[1232] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX567).

[1233] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX568).

[1234] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX569).

[1235] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX570).

[1236] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX571).

[1237] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX572).

[1238] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX573).

[1239] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX574).

[1240] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX575).

[1241] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX576).

[1242] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX577).

[1243] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX578).

[1244] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX579).

[1245] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX580).

[1246] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX581).

[1247] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX582).

[1248] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX583).

[1249] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX584).

[1250] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX585).

[1251] A present compound (L-1) wherein R.sup.1b and R.sup.1c represents CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX586).

[1252] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX587).

[1253] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX588).

[1254] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.1, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX589).

[1255] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3](hereinafter, referred to as Compound class SX590).

[1256] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX591).

[1257] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX592).

[1258] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX593).

[1259] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.1, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX594).

[1260] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX595).

[1261] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX596).

[1262] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX597).

[1263] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX598).

[1264] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX599).

[1265] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX600).

[1266] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX601).

[1267] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX602).

[1268] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX603).

[1269] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX604).

[1270] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX605).

[1271] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX606).

[1272] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX607).

[1273] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX608).

[1274] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX609).

[1275] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX610).

[1276] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX611).

[1277] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX612).

[1278] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX613).

[1279] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX614).

[1280] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX615).

[1281] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX616).

[1282] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX617).

[1283] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX618).

[1284] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX619).

[1285] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX620).

[1286] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX621).

[1287] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX622).

[1288] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX623).

[1289] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX624).

[1290] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX625).

[1291] A present compound (L-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX626).

[1292] A present compound (L-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX627).

[1293] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX628).

[1294] A present compound (L-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX629).

[1295] A present compound (L-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX630).

[1296] A present compound (L-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX631).

[1297] A present compound (L-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX632).

[1298] A present compound (L-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX633).

[1299] A present compound (L-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX634).

[1300] A present compound (L-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX635).

[1301] A present compound (L-1) wherein R.sup.1b represents CF.sub.3, R.sup.1b represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX636).

[1302] A present compound (L-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents any one group selected from a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, A.sup.1 represents a nitrogen atom, and A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH (hereinafter, referred to as Compound class SX637).

[1303] A compound represented by formula (L-2):

##STR00070##

(hereinafter, referred to as Compound (L-2))

[1304] wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX638).

TABLE-US-00023 TABLE L4 [00071] embedded image [00072] [00073] [00074] [00075] [00076]

TABLE-US-00024 TABLE L5 [00077] embedded image [00078] [00079] [00080] [00081] [00082]

TABLE-US-00025 TABLE L6 [00083] embedded image [00084] [00085] [00086] [00087] [00088]

TABLE-US-00026 TABLE L7 [00089] embedded image [00090] [00091] [00092] [00093] [00094] [00095] [00096]

TABLE-US-00027 TABLE L8 [00097] embedded image [00098] [00099] [00100] [00101] [00102] [00103] [00104]

TABLE-US-00028 TABLE L9 [00105] embedded image [00106] [00107] [00108] [00109] [00110] [00111] [00112]

[1305] A present compound (L-2) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX639).

[1306] A present compound (L-2) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX640).

[1307] A present compound (L-2) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX641).

[1308] A present compound (L-2) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX642).

[1309] A present compound (L-2) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX643).

[1310] A present compound (L-2) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX644).

[1311] A present compound (L-2) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX645).

[1312] A present compound (L-2) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX646).

[1313] A present compound (L-2) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX647).

[1314] A present compound (L-2) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX648).

[1315] A present compound (L-2) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX649).

[1316] A present compound (L-2) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX650).

[1317] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a fluorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX651).

[1318] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a chlorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX652).

[1319] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a bromine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX653).

[1320] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents an iodine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX654).

[1321] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a methyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX655).

[1322] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents an ethyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX656).

[1323] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a propyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX657).

[1324] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents an isopropyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX658).

[1325] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents a cyclopropyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX659).

[1326] A present compound (L-2) wherein R.sup.1b and R.sup.1c represents CF.sub.3, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX660).

[1327] A compound represented by formula (L-3):

##STR00113##

(hereinafter, referred to as Compound (L-3))

[1328] wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX661).

[1329] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX662).

[1330] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX663).

[1331] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX664).

[1332] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX665).

[1333] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX666).

[1334] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX667).

[1335] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX668).

[1336] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX669).

[1337] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX670).

[1338] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX671).

[1339] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX672).

[1340] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX673).

[1341] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX674).

[1342] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX675).

[1343] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX676).

[1344] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX677).

[1345] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX678).

[1346] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX679).

[1347] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX680).

[1348] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX681).

[1349] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX682).

[1350] A compound (L-3) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX683).

[1351] A present compound (L-3) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents any one group selected from a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, and A.sup.1, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH (hereinafter, referred to as Compound class SX684).

[1352] A compound represented by formula (L-4):

##STR00114##

(hereinafter, referred to as Compound (L-4))

[1353] wherein R.sup.1b and R.sup.1c represent a chlorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX685).

[1354] A compound represented by formula (L-5):

##STR00115##

(hereinafter, referred to as Compound (L-5))

[1355] wherein R.sup.1b and R.sup.1c represent a chlorine atom, and A.sup.2, A.sup.3, A.sup.4, and A.sup.J represent CH, and A.sup.1 represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX686).

[1356] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, and A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX687).

[1357] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, and A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX688).

[1358] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX689).

[1359] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX690).

[1360] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX691).

[1361] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX692).

[1362] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX693).

[1363] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX694).

[1364] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX695).

[1365] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX696).

[1366] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX697).

[1367] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX698).

[1368] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX699).

[1369] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX700).

[1370] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX701).

[1371] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX702).

[1372] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX703).

[1373] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX704).

[1374] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX705).

[1375] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX706).

[1376] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX707).

[1377] A compound (L-5) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX708).

[1378] A present compound (L-5) wherein Rib represents a chlorine atom, R.sup.1c represents any one group selected from a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, and A.sup.1, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH (hereinafter, referred to as Compound class SX709).

[1379] A compound represented by formula (L-6):

##STR00116##

(hereinafter, referred to as Compound (L-6))

[1380] wherein R.sup.1b and R.sup.1c represent a chlorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class SX710).

[1381] A compound represented by formula (K-1):

##STR00117##

(hereinafter, referred to as Compound (K-1))

[1382] wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.1 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX1)

[1383] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX2).

[1384] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX3).

[1385] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX4).

[1386] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX5).

[1387] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX6).

[1388] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX7).

[1389] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX8).

[1390] A compound (K-1) wherein Rib represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX9).

[1391] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX10).

[1392] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.11 represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX11).

[1393] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX12).

[1394] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX13).

[1395] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX14).

[1396] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX15).

[1397] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX16).

[1398] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX17).

[1399] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX18).

[1400] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX19).

[1401] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX20).

[1402] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX21).

[1403] A compound (K-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX22).

[1404] A compound (K-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX23).

[1405] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX24).

[1406] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX25).

[1407] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX26).

[1408] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX27).

[1409] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX28).

[1410] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX29).

[1411] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX30).

[1412] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX31).

[1413] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX32).

[1414] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX33).

[1415] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX34).

[1416] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.2, A.sup.1, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX35).

[1417] A compound (K-1) wherein Rib represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX36).

[1418] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX37).

[1419] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX38).

[1420] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX39).

[1421] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX40).

[1422] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX41).

[1423] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX42).

[1424] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX43).

[1425] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX44).

[1426] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX45).

[1427] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX46).

[1428] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX47).

[1429] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX48).

[1430] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX49).

[1431] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX50).

[1432] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX51).

[1433] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX52).

[1434] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX53).

[1435] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX54).

[1436] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX55).

[1437] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX56).

[1438] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX57).

[1439] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX58).

[1440] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX59).

[1441] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX60).

[1442] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX61).

[1443] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX62).

[1444] A compound (K-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX63).

[1445] A compound (K-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.11 represents a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX64).

[1446] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX65).

[1447] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX66).

[1448] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX67).

[1449] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX68).

[1450] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX69).

[1451] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX70).

[1452] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX71).

[1453] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX72).

[1454] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX73).

[1455] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX74).

[1456] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX75).

[1457] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX76).

[1458] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX77).

[1459] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX78).

[1460] A compound (K-1) wherein Rib represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX79).

[1461] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX80).

[1462] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX81).

[1463] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX82).

[1464] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX83).

[1465] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX84).

[1466] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX85).

[1467] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX86).

[1468] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX87).

[1469] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX88).

[1470] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX89).

[1471] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX90).

[1472] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX91).

[1473] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX92).

[1474] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX93).

[1475] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX94).

[1476] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX95).

[1477] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX96).

[1478] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX97).

[1479] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX98).

[1480] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX99).

[1481] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX100).

[1482] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX101).

[1483] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX102).

[1484] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX103).

[1485] A compound (K-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX104).

[1486] A compound (K-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX105).

[1487] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX106).

[1488] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX107).

[1489] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX108).

[1490] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX109).

[1491] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX110).

[1492] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX111).

[1493] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX112).

[1494] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX113).

[1495] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an iodine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX114).

[1496] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX115).

[1497] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX116).

[1498] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX117).

[1499] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an isopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX118).

[1500] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a cyclopropyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX119).

[1501] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents CF.sub.3, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX120).

[1502] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX121).

[1503] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX122).

[1504] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a propyl group, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX123).

[1505] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX124).

[1506] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX125).

[1507] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX126).

[1508] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX127).

[1509] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX128).

[1510] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX129).

[1511] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX130).

[1512] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX131).

[1513] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX132).

[1514] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX133).

[1515] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX134).

[1516] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX135).

[1517] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX136).

[1518] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX137).

[1519] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX138).

[1520] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX139).

[1521] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX140).

[1522] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX141).

[1523] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX142).

[1524] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX143).

[1525] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX144).

[1526] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX145).

[1527] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX146).

[1528] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX147).

[1529] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX148).

[1530] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX149).

[1531] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX150).

[1532] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX151).

[1533] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX152).

[1534] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX153).

[1535] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX154).

[1536] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX155).

[1537] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX156).

[1538] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX157).

[1539] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX158).

[1540] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX159).

[1541] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX160).

[1542] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX161).

[1543] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX162).

[1544] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX163).

[1545] A compound (K-1) wherein R.sup.b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX164).

[1546] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX165).

[1547] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX166).

[1548] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX167).

[1549] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX168).

[1550] A compound (K-1) wherein R.sup.b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX169).

[1551] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX170).

[1552] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX171).

[1553] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX172).

[1554] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX173).

[1555] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX174).

[1556] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX175).

[1557] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX176).

[1558] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX177).

[1559] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX178).

[1560] A compound (K-1) wherein R.sup.b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX179).

[1561] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX180).

[1562] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX181).

[1563] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX182).

[1564] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX183).

[1565] A compound (K-1) wherein R.sup.b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX183).

[1566] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX184).

[1567] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX185).

[1568] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX186).

[1569] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX187).

[1570] A compound (K-1) wherein R.sup.b represents a methyl group, R.sup.11 represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX188).

[1571] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX189).

[1572] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX190).

[1573] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX191).

[1574] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX191).

[1575] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.11 represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX192).

[1576] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX193).

[1577] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX194).

[1578] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX195).

[1579] A compound (K-1) wherein R.sup.b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX196).

[1580] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.11 represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX197).

[1581] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX198).

[1582] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX199).

[1583] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX200).

[1584] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX201).

[1585] A compound (K-1) wherein R.sup.b represents a methyl group, R.sup.11 represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX202).

[1586] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX203).

[1587] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX204).

[1588] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX205).

[1589] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX206).

[1590] A compound (K-1) wherein R.sup.b represents an ethyl group, R.sup.11 represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX207).

[1591] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX208).

[1592] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX209).

[1593] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX210).

[1594] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX211).

[1595] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX212).

[1596] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX213).

[1597] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX214).

[1598] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX215).

[1599] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX216).

[1600] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX217).

[1601] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX218).

[1602] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX219).

[1603] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX220).

[1604] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX221).

[1605] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX222).

[1606] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX223).

[1607] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX224).

[1608] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX225).

[1609] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX226).

[1610] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX227).

[1611] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.11 represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX228).

[1612] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX229).

[1613] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX230).

[1614] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX231).

[1615] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX232).

[1616] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX233).

[1617] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX234).

[1618] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX235).

[1619] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.3 represent CH, and A.sup.4 represents any one substituent substituent indicated in [Table L1] to [Table L3] indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX236).

[1620] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX237).

[1621] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX238).

[1622] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX239).

[1623] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.1, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX240).

[1624] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX241).

[1625] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX242).

[1626] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX243).

[1627] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX244).

[1628] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX245).

[1629] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX246).

[1630] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX247).

[1631] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX248).

[1632] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX249).

[1633] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX250).

[1634] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX251).

[1635] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX252).

[1636] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX253).

[1637] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX254).

[1638] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX255).

[1639] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX256).

[1640] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX257).

[1641] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX258).

[1642] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX259).

[1643] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.5 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX260).

[1644] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX261).

[1645] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX262).

[1646] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX263).

[1647] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX264).

[1648] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX265).

[1649] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX266).

[1650] A compound (K-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a hydrogen atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX267).

[1651] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX268).

[1652] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX269).

[1653] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX270).

[1654] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX271).

[1655] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX272).

[1656] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX273).

[1657] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX274).

[1658] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX275).

[1659] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX276).

[1660] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX277).

[1661] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX278).

[1662] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX279).

[1663] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX280).

[1664] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX281).

[1665] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX282).

[1666] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX283).

[1667] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX284).

[1668] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX285).

[1669] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX286).

[1670] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX287).

[1671] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX288).

[1672] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX289).

[1673] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX290).

[1674] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX291).

[1675] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.1 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX2 92).

[1676] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX293).

[1677] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX294).

[1678] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX295).

[1679] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 [Table L3] (hereinafter, referred to as Compound class CX296).

[1680] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX297).

[1681] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX298).

[1682] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX299).

[1683] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX300).

[1684] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 [Table L3] (hereinafter, referred to as Compound class CX301).

[1685] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX302).

[1686] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX303).

[1687] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX304).

[1688] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represents CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX305).

[1689] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX306).

[1690] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX307).

[1691] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX308).

[1692] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX309).

[1693] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX310).

[1694] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX311).

[1695] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX312).

[1696] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX313).

[1697] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX314).

[1698] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX315).

[1699] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX316).

[1700] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX317).

[1701] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX318).

[1702] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX319).

[1703] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX320).

[1704] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX321).

[1705] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX322).

[1706] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX323).

[1707] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX324).

[1708] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX325).

[1709] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX326).

[1710] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.1 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX327).

[1711] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX328).

[1712] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX329).

[1713] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX330).

[1714] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX331).

[1715] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX332).

[1716] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX333).

[1717] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX334).

[1718] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX335).

[1719] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX336).

[1720] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX337).

[1721] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX338).

[1722] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX339).

[1723] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX340).

[1724] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX341).

[1725] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX342).

[1726] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX343).

[1727] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX344).

[1728] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX345).

[1729] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX346).

[1730] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX347).

[1731] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX348).

[1732] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX349).

[1733] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX350).

[1734] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX351).

[1735] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX352).

[1736] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX353).

[1737] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX354).

[1738] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX355).

[1739] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX356).

[1740] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX357).

[1741] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX358).

[1742] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX359).

[1743] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX360).

[1744] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX361).

[1745] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX362).

[1746] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX363).

[1747] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX364).

[1748] A compound (K-1) wherein R.sup.1b and R.sup.1c(represent CF.sub.3, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX365).

[1749] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX366).

[1750] A compound (K-1) wherein Rib and R.sup.1c represent CF.sub.3, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX367).

[1751] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX368).

[1752] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX369).

[1753] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX370).

[1754] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 [Table L3] (hereinafter, referred to as Compound class CX371).

[1755] A compound (K-1) wherein Rib and R.sup.1c represent CF.sub.3, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX372).

[1756] A compound (K-1) wherein Rib and R.sup.1c represent CF.sub.3, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX373).

[1757] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX374).

[1758] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX375).

[1759] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX376).

[1760] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX377).

[1761] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX378).

[1762] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX379).

[1763] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX380).

[1764] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX381).

[1765] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX382).

[1766] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX383).

[1767] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX384).

[1768] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX385).

[1769] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX386).

[1770] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX387).

[1771] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX388).

[1772] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX389).

[1773] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX390).

[1774] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX391).

[1775] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX392).

[1776] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX393).

[1777] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX394).

[1778] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX395).

[1779] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX396).

[1780] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX397).

[1781] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX398).

[1782] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX399).

[1783] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX400).

[1784] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX401).

[1785] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX402).

[1786] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX403).

[1787] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX404).

[1788] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX405).

[1789] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX406).

[1790] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX407).

[1791] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX408).

[1792] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX409).

[1793] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX410).

[1794] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX411).

[1795] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX412).

[1796] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX413).

[1797] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX414).

[1798] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX415).

[1799] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX416).

[1800] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX417).

[1801] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX418).

[1802] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX419).

[1803] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX420).

[1804] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX421).

[1805] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX422).

[1806] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX423).

[1807] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX424).

[1808] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.5 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX425).

[1809] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX426).

[1810] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX427).

[1811] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX428).

[1812] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX429).

[1813] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX430).

[1814] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX431).

[1815] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX432).

[1816] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX433).

[1817] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX434).

[1818] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX435).

[1819] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX436).

[1820] A compound (K-1) wherein Rib represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX437).

[1821] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX438).

[1822] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX439).

[1823] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX440).

[1824] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX441).

[1825] A compound (K-1) wherein Rib represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX442).

[1826] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX443).

[1827] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX444).

[1828] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX445).

[1829] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX446).

[1830] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX447).

[1831] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX448).

[1832] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX449).

[1833] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX450).

[1834] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent to as Compound class CX451).

[1835] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX452).

[1836] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX453).

[1837] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX454).

[1838] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX455).

[1839] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX456).

[1840] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX457).

[1841] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX458).

[1842] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a methyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX459).

[1843] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX460).

[1844] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX461).

[1845] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX462).

[1846] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX463).

[1847] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX464).

[1848] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX465).

[1849] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX466).

[1850] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX467).

[1851] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX468).

[1852] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX469).

[1853] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX470).

[1854] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX471).

[1855] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX472).

[1856] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX473).

[1857] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX474).

[1858] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX475).

[1859] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX476).

[1860] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX477).

[1861] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX478).

[1862] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX479).

[1863] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX480).

[1864] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.3 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX481).

[1865] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX482).

[1866] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX483).

[1867] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX484).

[1868] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX485).

[1869] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX486).

[1870] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX487).

[1871] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX488).

[1872] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX489).

[1873] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX490).

[1874] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX491).

[1875] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX492).

[1876] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX493).

[1877] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX494).

[1878] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX495).

[1879] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX496).

[1880] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX497).

[1881] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX498).

[1882] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX499).

[1883] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX500).

[1884] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX501).

[1885] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX502).

[1886] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX503).

[1887] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX504).

[1888] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX505).

[1889] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX506).

[1890] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX507).

[1891] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX508).

[1892] A compound (K-1) wherein Rib represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX509).

[1893] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX510).

[1894] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX511).

[1895] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX512).

[1896] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX513).

[1897] A compound (K-1) wherein Rib represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX514).

[1898] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX515).

[1899] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX516).

[1900] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX517).

[1901] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX518).

[1902] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX519).

[1903] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX520).

[1904] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX521).

[1905] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX522).

[1906] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX523).

[1907] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX524).

[1908] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX525).

[1909] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX526).

[1910] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX527).

[1911] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX528).

[1912] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX529).

[1913] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX530).

[1914] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX531).

[1915] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX532).

[1916] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX533).

[1917] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX534).

[1918] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX535).

[1919] A compound (K-1) wherein R.sup.b represents a methyl group, R.sup.11 represents an ethyl group, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX536).

[1920] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX537).

[1921] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX538).

[1922] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents an ethyl group, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX539).

[1923] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CF, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX540).

[1924] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CCl, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX541).

[1925] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents an ethyl group, A.sup.2 represents CBr, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX542).

[1926] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CI, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX543).

[1927] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents C-Me, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX544).

[1928] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents COMe, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX545).

[1929] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents CCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX546).

[1930] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.2 represents COCF.sub.3, A.sup.1, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX547).

[1931] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CF, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX548).

[1932] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CCl, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX549).

[1933] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CBr, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX550).

[1934] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CI, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX551).

[1935] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents C-Me, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX552).

[1936] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents COMe, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX553).

[1937] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents CCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX554).

[1938] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a bromine atom, A.sup.3 represents COCF.sub.3, A.sup.1, A.sup.2, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX555).

[1939] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents any one of a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, and A.sup.1, A.sup.2, A.sup.1, A.sup.4, and A.sup.5 represent CH (hereinafter, referred to as Compound class CX556).

[1940] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX557).

[1941] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX558).

[1942] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX559).

[1943] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX560).

[1944] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX561).

[1945] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX562).

[1946] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX563).

[1947] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX564).

[1948] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX565).

[1949] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX566).

[1950] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX567).

[1951] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX568).

[1952] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX569).

[1953] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX570).

[1954] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX571).

[1955] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX572).

[1956] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX573).

[1957] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX574).

[1958] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX575).

[1959] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.4 represent CH, and A.sup.5 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX576).

[1960] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX578).

[1961] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX579).

[1962] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX580).

[1963] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX581).

[1964] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX582).

[1965] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX583).

[1966] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX584).

[1967] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX585).

[1968] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX586).

[1969] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX587).

[1970] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX588).

[1971] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX589).

[1972] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX590).

[1973] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX591).

[1974] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX592).

[1975] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX593).

[1976] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX594).

[1977] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX595).

[1978] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1b represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.3, and A.sup.5 represent CH, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX596).

[1979] A compound (K-1) wherein R.sup.11 and R.sup.1c represent a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX597).

[1980] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX598).

[1981] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX599).

[1982] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX600).

[1983] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX601).

[1984] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX602).

[1985] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX603).

[1986] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX604).

[1987] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX605).

[1988] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX606).

[1989] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX607).

[1990] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX608).

[1991] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX609).

[1992] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX610).

[1993] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX611).

[1994] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX612).

[1995] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX613).

[1996] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX614).

[1997] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX615).

[1998] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1b represents a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX616).

[1999] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a fluorine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX617).

[2000] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a chlorine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX618).

[2001] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a bromine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX619).

[2002] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an iodine atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX620).

[2003] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a methyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX621).

[2004] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an ethyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX622).

[2005] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a propyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX623).

[2006] A compound (K-1) wherein R.sup.1b and R.sup.1c represent an isopropyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX624).

[2007] A compound (K-1) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX625).

[2008] A compound (K-1) wherein R.sup.1b and R.sup.1c represent CF.sub.3, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX626).

[2009] A compound (K-1) wherein R.sup.1b represents a fluorine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX627).

[2010] A compound (K-1) wherein R.sup.1b represents a chlorine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX628).

[2011] A compound (K-1) wherein R.sup.1b represents a bromine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX629).

[2012] A compound (K-1) wherein R.sup.1b represents an iodine atom, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX630).

[2013] A compound (K-1) wherein R.sup.1b represents a methyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX631).

[2014] A compound (K-1) wherein R.sup.1b represents an ethyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX632).

[2015] A compound (K-1) wherein R.sup.1b represents a propyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX633).

[2016] A compound (K-1) wherein R.sup.1b represents an isopropyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX634).

[2017] A compound (K-1) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX635).

[2018] A compound (K-1) wherein R.sup.1b represents CF.sub.3, R.sup.1c represent a hydrogen atom, A.sup.1 represents a nitrogen atom, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class CX636).

[2019] A compound (K-1) wherein R.sup.1b represents chlorine atom, R.sup.1c represents any one of a hydrogen atom, a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, a methyl group, an ethyl group, a propyl group, an isopropyl group, a cyclopropyl group, or CF.sub.3, A.sup.1 represents a nitrogen atom, and A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH (hereinafter, referred to as Compound class CX637).

[2020] A compound represented by formula (K-2):

##STR00118##

(hereinafter, referred to as compound (K-2))
wherein R.sup.1b represents a fluorine atom, R.sup.1c represents a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX638).

[2021] A compound (K-2) wherein R.sup.1b represents a chlorine atom, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX639).

[2022] A compound (K-2) wherein R.sup.1b represents a bromine atom, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX640).

[2023] A compound (K-2) wherein R.sup.1b represents an iodine atom, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX641).

[2024] A compound (K-2) wherein R.sup.1b represents a methyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX642).

[2025] A compound (K-2) wherein R.sup.1b represents an ethyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX643).

[2026] A compound (K-2) wherein R.sup.1b represents a propyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX644).

[2027] A compound (K-2) wherein R.sup.1b represents an isopropyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX645).

[2028] A compound (K-2) wherein R.sup.1b represents a cyclopropyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX646).

[2029] A compound (K-2) wherein R.sup.1b represents CF.sub.3, R.sup.1b represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX647).

[2030] A compound (K-2) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX648).

[2031] A compound (K-2) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX649).

[2032] A compound (K-2) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a hydrogen atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX650).

[2033] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a fluorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX651).

[2034] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a chlorine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX652).

[2035] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a bromine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX653).

[2036] A compound (K-2) wherein R.sup.1b and R.sup.1c represent an iodine atom, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX654).

[2037] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a methyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX655).

[2038] A compound (K-2) wherein R.sup.1b and R.sup.1c represent an ethyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX656).

[2039] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a propyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX657).

[2040] A compound (K-2) wherein R.sup.1b and R.sup.1c represent an isopropyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX658).

[2041] A compound (K-2) wherein R.sup.1b and R.sup.1c represent a cyclopropyl group, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX659).

[2042] A compound (K-2) wherein R.sup.1b and R.sup.1c represent CF.sub.3, and Q represents any one substituent indicated in [Table L4] to [Table L9] (hereinafter, referred to as Compound class CX660).

[2043] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX711).

[2044] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a hydrogen atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX712).

[2045] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX713).

[2046] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX714).

[2047] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX715).

[2048] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX716).

[2049] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX717).

[2050] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX718).

[2051] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX719).

[2052] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX720).

[2053] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a fluorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX721).

[2054] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX722).

[2055] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX723).

[2056] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a chlorine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX724).

[2057] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX725).

[2058] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX726).

[2059] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a bromine atom, A.sup.2, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.1 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX727).

[2060] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX728).

[2061] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX729).

[2062] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX730).

[2063] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX731).

[2064] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX732).

[2065] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX733).

[2066] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.3c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX734).

[2067] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX735).

[2068] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX736).

[2069] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX737).

[2070] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX738).

[2071] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX739).

[2072] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX740).

[2073] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX741).

[2074] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX742).

[2075] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX743).

[2076] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.11 represent a bromine atom, A.sup.1, A.sup.3, A.sup.4, and A.sup.5 represent CH, and A.sup.2 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX744).

[2077] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX745).

[2078] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX746).

[2079] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX747).

[2080] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX748).

[2081] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX749).

[2082] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX750).

[2083] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX751).

[2084] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX752).

[2085] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX753).

[2086] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX754).

[2087] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX755).

[2088] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX756).

[2089] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX757).

[2090] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX758).

[2091] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.11 represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX759).

[2092] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX760).

[2093] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.2, A.sup.4, and A.sup.5 represent CH, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX761).

[2094] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX762).

[2095] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX763).

[2096] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX764).

[2097] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX765).

[2098] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX766).

[2099] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 [Table L3] (hereinafter, referred to as Compound class SX767).

[2100] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX768).

[2101] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX769).

[2102] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX770).

[2103] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX771).

[2104] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX772).

[2105] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX773).

[2106] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX774).

[2107] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represent a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX775).

[2108] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represent a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX776).

[2109] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX777).

[2110] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX778).

[2111] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX779).

[2112] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX780).

[2113] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX781).

[2114] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represent a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX782).

[2115] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX783).

[2116] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX784).

[2117] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX785).

[2118] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX786).

[2119] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX787).

[2120] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX788).

[2121] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX789).

[2122] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX790).

[2123] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX791).

[2124] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX792).

[2125] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX793).

[2126] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX794).

[2127] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX795).

[2128] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX796).

[2129] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX797).

[2130] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX798).

[2131] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX799).

[2132] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX800).

[2133] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX801).

[2134] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX802).

[2135] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX803).

[2136] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX804).

[2137] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX805).

[2138] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX806).

[2139] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX807).

[2140] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX808).

[2141] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX809).

[2142] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX810).

[2143] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX811).

[2144] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX812).

[2145] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX813).

[2146] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX814).

[2147] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX815).

[2148] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX816).

[2149] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX817).

[2150] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX818).

[2151] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX819).

[2152] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX820).

[2153] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX821).

[2154] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX822).

[2155] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX823).

[2156] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX824).

[2157] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX825).

[2158] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX826).

[2159] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX827).

[2160] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX828).

[2161] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX829).

[2162] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX830).

[2163] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX831).

[2164] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX832).

[2165] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX833).

[2166] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX834).

[2167] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX835).

[2168] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX836).

[2169] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX837).

[2170] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX838).

[2171] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX839).

[2172] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX840).

[2173] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX841).

[2174] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX842).

[2175] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX843).

[2176] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX844).

[2177] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX845).

[2178] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.4, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.3 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX846).

[2179] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX847).

[2180] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX848).

[2181] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX849).

[2182] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX850).

[2183] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX851).

[2184] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX852).

[2185] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX853).

[2186] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX854).

[2187] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX855).

[2188] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX856).

[2189] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX857).

[2190] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX858).

[2191] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX859).

[2192] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX860).

[2193] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX861).

[2194] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX862).

[2195] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CF, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX863).

[2196] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX864).

[2197] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX865).

[2198] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX866).

[2199] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX867).

[2200] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX868).

[2201] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX869).

[2202] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX870).

[2203] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX871).

[2204] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX872).

[2205] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX873).

[2206] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX874).

[2207] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX875).

[2208] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.11 represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX876).

[2209] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX877).

[2210] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX878).

[2211] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX879).

[2212] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCl, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX880).

[2213] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX881).

[2214] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX882).

[2215] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX883).

[2216] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX884).

[2217] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX885).

[2218] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX886).

[2219] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX887).

[2220] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX888).

[2221] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX889).

[2222] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX890).

[2223] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX891).

[2224] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX892).

[2225] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX893).

[2226] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX894).

[2227] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX895).

[2228] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX896).

[2229] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.1 represent CH, A.sup.2 represents C-Me, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX897).

[2230] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX898).

[2231] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX899).

[2232] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX900).

[2233] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX901).

[2234] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX902).

[2235] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX903).

[2236] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX904).

[2237] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX905).

[2238] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX906).

[2239] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX907).

[2240] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX908).

[2241] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX909).

[2242] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX910).

[2243] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX911).

[2244] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX912).

[2245] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.J represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX913).

[2246] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents CCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX914).

[2247] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX915).

[2248] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a hydrogen atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX916).

[2249] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX917).

[2250] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX918).

[2251] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX919).

[2252] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX920).

[2253] A compound represented by formula (L-1) wherein R.sup.1b represents a methoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX921).

[2254] A compound represented by formula (L-1) wherein R.sup.1b represents an ethoxy group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX922).

[2255] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX923).

[2256] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX924).

[2257] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a fluorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX925).

[2258] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX926).

[2259] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX927).

[2260] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfonyl group, R.sup.1c represents a chlorine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX928).

[2261] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfanyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX929).

[2262] A compound represented by formula (L-1) wherein R.sup.1b represents a methylsulfinyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX930).

[2263] A compound represented by formula (L-1) wherein Rib represents a methylsulfonyl group, R.sup.1c represents a bromine atom, A.sup.1, A.sup.3, and A.sup.5 represent CH, A.sup.2 represents COCF.sub.3, and A.sup.4 represents any one substituent indicated in [Table L1] to [Table L3] (hereinafter, referred to as Compound class SX931).

[2264] Next, the formulation examples of the compounds of the present invention are shown below. In the formulation examples, the parts represents part by weight unless otherwise specified. The present compound S represents the compounds described in the Compound Classes SX1 to SX931.

Formulation Example 1

[2265] Thirty five (35) parts of a mixture of ammonium polyoxyethylene alkyl ether sulfate and wet silica (weight ratio: 1:1), 10 parts of any one of the present compound S, and 55 parts of water are mixed, and the mixture is then finely-ground by a wet grinding method to obtain a formulation.

Formulation Example 2

[2266] Fifty (50) parts of any one of the present compound S, 3 parts of calcium lignin sulfonate, 2 parts of sodium lauryl sulfate, and 45 parts of silica are well mixed-grinding to obtain a formulation.

Formulation Example 3

[2267] Five (5) parts of any one of the present compound S, 9 parts of polyoxyethylene styryl phenyl ether, 5 parts of polyoxyethylene decyl ether (Number of ethylene oxide additions: 5), 6 parts of calcium dodecylbenzene sulfonate and 75 parts of xylene are well mixed to obtain a formulation.

Formulation Example 4

[2268] Two (2) parts of any one of the present compound S, 1 part of silica, 2 parts of calcium lignin sulfonate, 30 parts of bentonite and 65 parts of kaolin clay are mixed-grinding, and thereto is added an appropriate amount of water, and the mixture is well kneaded and is then granulated with a granulator and dried to obtain a formulation.

Formulation Example 5

[2269] Ten (10) parts of any one of the present compound S is mixed with a mixture of 18 parts of benzyl alcohol and 9 parts of DMSO, and thereto are added 6.3 parts of GERONOL (registered trademark) TE250, 2.7 parts of Ethylan (registered trademark)NS-500LQ, and 54 parts of Solvent naphtha, and the mixture is mixed to obtain a formulation.

Formulation Example 6

[2270] Zero point one (0.1) parts of any one of the present compound S and 39.9 parts of kerosene are dissolved while mixing, and the mixture is placed in an aerosol container, and 60 parts of liquefied petroleum gas (mixture of propane, butane and isobutane; saturated vapor pressure: 0.47 MPa (25? C.)) is filled in the container to obtain a formulation.

Formulation Example 7

[2271] Zero point two (0.2) parts of any one of the present compound S, 50 parts of pyrethrum extract dreg powder, 30 parts of Machilus thunbergii powder, and 19.8 parts of wood powder are mixed, and an appropriate amount of water is added thereto, and the mixture is well kneaded, and is extracted with an extruder into a plate-like sheet, and the resulting sheet is made a spiral-like form thereof with a punching machine to obtain a formulation.

[2272] Next, an efficacy of the present compound on controlling harmful arthropods is shown by Test examples. The following tests were conducted at 25? C.

Test Method 1

[2273] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2274] Cucumber (cucumber sativus) seedling (on the developmental stage of the second true leaf) is planted in a cup, and approximately 30 cotton aphids (Aphis gossypii) (all stages of life) are released onto the seedling. After one day, the diluted solutions are sprayed into the seedling at a ratio of 10 mL/seedling. After 5 days, the number of the surviving insects is examined and the controlling value is calculated by the following equation.

Controlling value (%)={1?(Cb?Tai)/(Cai?Tb)}?100

wherein the symbols in the equation represent the following descriptions.

[2275] Cb: Number of the test insects in untreated group;

[2276] Cai: Number of the surviving insects at the time of the examination in untreated group;

[2277] Tb: Number of the test insects in treated group;

[2278] Tai: Number of the surviving insects at the time of the examination in treated group;

[2279] Here the untreated group represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.

Test Example 1-1

[2280] The test was conducted according to the Test method 1 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value.

Present compound Nos: 1, 2, 3, 4, 7, 8, 9, 10, 11, 12, 14, 15, 17, 19, 23, 25, 28, 29, 30, 31, 32, 34, 35, 36, 38, 39, 40, 42, 45, 46, 49, 53, 54, 56, 60, 63, 64, 65, 67, 71, 72, 74, 77, 78, 79, 80, 81, 82, 83, 86, 87, 90, 91, 92, 94, 96, 100, 101, 108, 118, 123, 125, 129, 130, 135, 138, 139, 140, 143, 145, 146, 147, 148, 149

Test Method 2

[2281] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2282] Cucumber (cucumber sativus) seedling (on the developmental stage of the second true leaf) is planted in a cup, and approximately 30 cotton aphids (Aphis gossypii) (all stages of life) are released onto the seedling. After one day, the diluted solutions are sprayed into the seedling at a ratio of 10 mL/seedling. After 5 days, the number of the surviving insects is examined and the controlling value is calculated by the following equation.

[00001] $Controlling value (%) = {1 - (Cb ? Tai) / (Cai ? Tb)} ? 100$

wherein the symbols in the equation represent the following descriptions.

[2283] Cb: Number of the test insects in untreated group;

[2284] Cai: Number of the surviving insects at the time of the examination in untreated group;

[2285] Tb: Number of the test insects in treated group;

[2286] Tai: Number of the surviving insects at the time of the examination in treated group;

[2287] Here the untreated group represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.

Test Example 2-1

[2288] The test was conducted according to the Test method 2 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value.

Present compound Nos: 1, 2, 3, 4, 7, 8, 9, 10, 11, 12, 14, 15, 19, 23, 24, 27, 28, 29, 30, 32, 33, 34, 35, 36, 38, 39, 40, 42, 45, 46, 48, 49, 51, 53, 54, 56, 60, 61, 63, 65, 67, 68, 71, 72, 75, 76, 77, 78, 79, 80, 82, 83, 90, 91, 92, 94, 96, 97, 100, 108, 110, 112, 117, 118, 119, 120, 121, 123, 125, 129, 130, 135, 138, 139, 140, 143, 145, 146, 147, 148, 149

Test Method 3

[2289] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2290] Rice (Oryza sativa) seedling (on the developmental stage of the second true leaf) is planted in a container, and the diluted solutions are sprayed into the seedling in a ratio of 10 mL/seedling. Thereafter, 20 of 3rd instar larvae of brown planthoppers (Nilaparvata lugens) are released onto the rice leaves. After 5 days, the number of the surviving insects is examined and the mortality is calculated by the following equation.

[00002] $Mortality (%) = {1 - the number of the surviving insects / 20} ? 100$

Test Example 3-1

[2291] The test was conducted according to the Test method 3 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the mortality.

Present compound Nos: 3, 7, 9, 10, 11, 12, 13, 14, 15, 16, 17, 19, 20, 21, 22, 25, 27, 28, 30, 32, 35, 38, 39, 40, 41, 42, 45, 46, 48, 49, 51, 53, 54, 56, 58, 59, 64, 65, 67, 71, 72, 73, 74, 75, 76, 77, 78, 79, 80, 82, 83, 87, 90, 91, 92, 94, 96, 100, 106, 108, 118, 121, 122, 123, 125, 128, 129, 130, 131, 132, 133, 134, 135, 136, 138, 139, 140, 143, 145, 146, 147, 148, 149

Test Method 4

[2292] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2293] Rice (Oryza sativa) seedling (on the developmental stage of the second true leaf) is planted in a container, and the diluted solutions are sprayed into the seedling in a ratio of 10 mL/seedling. Thereafter, 20 of 3rd instar larvae of brown planthoppers (Nilaparvata lugens) are released onto the rice leaves. After 6 days, the number of the surviving insects is examined and the mortality is calculated by the following equation.

[00003] $Mortality (%) = {1 - the number of the surviving insects / 20} ? 100$

[2294] Test Example 4-1 The test was conducted according to the Test method 4 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the mortality.

Present compound Nos: 1, 2, 3, 4, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 32, 33, 35, 38, 39, 40, 41, 42, 46, 48, 49, 51, 53, 54, 56, 58, 59, 60, 61, 64, 65, 67, 70, 71, 72, 73, 74, 75, 76, 77, 78, 79, 80, 82, 83, 85, 86, 90, 91, 92, 94, 95, 96, 97, 98, 100, 106, 108, 110, 112, 117, 118, 119, 120, 121, 123, 125, 128, 131, 132, 133, 134, 135, 136, 138, 139, 140, 143, 145, 146, 147, 148, 149

Test Example 4-2

[2295] The test was conducted according to the Test method 4 by making the prescribed concentration 50 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the mortality.

Present compound Nos: 2, 92, 95, 102, 134, 138, 148

Test Method 5

[2296] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2297] Silverleaf whiteflies (Bemisia tabaci) are released on tomato (Lycopersicon esculentum) seedling that is planted in a container, and then spawn for about 24 hours. The seedling are stored for 8 days, and the larvae of silverleaf whiteflies are hatched from the laid eggs. The diluted solutions are sprayed into the seedling in a ratio of 10 mL/seedling. After 7 days, the number of the surviving insects is examined, and the controlling value is calculated by the following equation.

[00004] $Controlling value (%) = {1 - (Cb ? Tai) / (Cai ? Tb)} ? 100$

wherein the symbols in the formula represent the following descriptions.

[2298] Cb: Number of the insects shortly before the treatment in untreated group;

[2299] Cai: Number of the surviving insects at the time of the investigation in untreated group;

[2300] Tb: Number of the insects shortly before the treatment in treated group;

[2301] Tai: Number of the surviving insects at the time of the investigation in treated group;

[2302] Here the untreated group represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.

Test Example 5-1

[2303] The test was conducted according to the Test method 5 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value.

Present compound Nos: 2, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19, 20, 22, 27, 28, 29, 30, 33, 34, 35, 36, 38, 40, 41, 42, 46, 48, 49, 53, 54, 56, 58, 59, 60, 61, 63, 64, 65, 68, 69, 71, 72, 73, 74, 75, 76, 77, 78, 79, 80, 83, 90, 91, 92, 94, 96, 97, 98, 100, 108, 109, 110, 111, 112, 117, 118, 119, 120, 121, 123, 125, 129, 132, 134, 135, 136, 138, 139, 140, 143, 145, 146, 147, 148, 149

Test Example 5-2

[2304] The test was conducted according to the Test method 5 by making the prescribed concentration 50 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value.

Present compound Nos: 2, 19, 94, 95, 117, 139, 145, 147

Test Method 6

[2305] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.

[2306] Into the diluted solution, 30 common house mosquito (Culex pipiens pallens) at the last instar larval stage are released, and after 1 day, the state of the house mosquito larvae is examined, and the mortality of insects is calculated by the following equation.

Mortality (%)=(the Number of the dead insects/the Number of tested insects)?100

Test Example 6-1

[2307] The test was conducted according to the Test method 6 by making the prescribed concentration 3.5 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 91% or more as the mortality.

Present compound Nos: 4, 7, 12, 15, 16, 17, 18, 19, 21, 28, 30, 36, 38, 39, 42, 46, 53, 56, 58, 60, 77, 78, 79, 82, 88, 91, 92, 107, 108, 121, 145, 146

Test Method 7

[2308] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.

[2309] Into the diluted solution, 30 common house mosquito (Culex pipiens pallens) at the last instar larval stage are released, and after 8 days, the state of the house mosquito larvae is examined, and the mortality of insects is calculated by the following equation.

Mortality (%)=(the Number of the dead insects/the Number of tested insects)?100

Test Example 7-1

[2310] The test was conducted according to the Test method 7 by making the prescribed concentration 3.5 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 91% or more as the mortality.

Present compound Nos: 5, 6, 8, 9, 10, 11, 13, 14, 20, 22, 23, 24, 25, 26, 27, 29, 31, 32, 34, 37, 41, 43, 47, 49, 50, 51, 52, 54, 55, 57, 59, 62, 63, 64, 65, 66, 67, 68, 71, 72, 73, 74, 76, 83, 84, 86, 90, 96, 99, 100, 114, 115, 116, 122, 130, 135, 139, 140, 145, 146

Test Method 8

[2311] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2312] Cabbage (Brassicae oleracea) seedling (on the developmental stage of the second to third true leaf) is planted in a cup, and the diluted solutions are sprayed into the seedling at a ratio of 20 mL/seedling. Thereafter, the stem and leaf thereof is cut out and then is installed into a cup that is covered with filter paper. Five (5) tobacco cutworm (Spodoptera litura) at the second instar larval stage are released into the cup. After 5 days, the number of the surviving insects is counted, and the mortality of insects is calculated by the following equation.

[00005] $Mortality (%) = (1 - the Number of the surviving insects / 5) ? 100$

Test Example 8-1

[2313] The test was conducted according to the Test method 8 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality.

Present compound Nos: 23, 28, 31, 32, 35, 38, 67, 77, 88, 89, 91, 100, 106, 118, 143

Test Method 9

[2314] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 1, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2315] Cabbage (Brassicae oleracea) seedling (on the developmental stage of the second to third true leaf) is planted in a cup, and the diluted solutions are sprayed into the seedling at a ratio of 20 mL/seedling. Thereafter, the stem and leaf thereof is cut out and then is installed into a cup that is covered with filter paper. Five (5) diamondback moth (Plutella xylostella) at the second instar larval stage are released into the cup. After 5 days, the number of the surviving insects is counted, and the mortality of insects is calculated by the following equation.

[00006] $Mortality (%) = (1 - the Number of the surviving insects / 5) ? 100$

Test Example 9-1

[2316] The test was conducted according to the Test method 9 by making the prescribed concentration 500 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 80% or more as the mortality.

Present compound Nos: 6, 12, 26, 28, 77, 79, 88, 89, 91, 99, 100, 101, 137

Test Method 10

[2317] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.

[2318] Cucumber (cucumber sativus) seedling (on the developmental stage of the second true leaf) is planted in a cup, and the diluted solutions are drenched to the foot of the seedling at a ratio of 5 mL/seedling. After 7 days, approximately 30 cotton aphids (Aphis gossypii) (all stages of life) are released onto the leaf of the seedling. After 6 days, the number of the surviving insects is examined and the controlling value is calculated by the following equation.

[00007] $Controlling value (%) = {1 - (Cb ? Tai) / (Cai ? Tb)} ? 100$

wherein the symbols in the equation represent the following descriptions.

[2319] Cb: Number of the test insects in untreated group;

[2320] Cai: Number of the surviving insects at the time of the examination in untreated group;

[2321] Tb: Number of the test insects in treated group;

[2322] Tai: Number of the surviving insects at the time of the examination in treated group;

[2323] Here the untreated group represents a group where a similar treatment procedure to that of treated group except not using the test compound is done.

Test Example 10-1

[2324] The test was conducted according to the Test method 10 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the controlling value.

Present compound Nos.: 14, 77

Test Method 11

[2325] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water to prepare a diluted solution containing a prescribed concentration of the test compound.

[2326] Five (5) mL of the diluted solution described above is added to a container, and therein is installed Rice (Oryza sativa) seedling (on the developmental stage of the second true leaf) that is planted in a container having a hole in the bottom. After 7 days, 20 3rd instar larvae of brown planthoppers (Nilaparvata lugens) are released. After 6 days, the number of the surviving insects is examined, and the mortality is calculated by the following equation.

[00008] $Mortality (%) = (1 - the Number of the surviving insects / 20) ? 100$

Test Example 11-1

[2327] The test was conducted according to the Test method 11 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the mortality.

Present compound Nos.: 2, 28, 29, 79, 98, 135

Test Method 12

[2328] Test compounds are made to a formulation according to a similar method to that described in the Formulation example 5, and thereto is added water containing 0.03 v/v % of Shindain (registered trademark) to prepare a diluted solution containing a prescribed concentration of the test compound.

[2329] Cucumber (Brassicae oleracea) seedling (on the developmental stage of the second leaf) is planted in a cup, and the diluted solutions are sprayed into the seedling at a ratio of 10 mL/seedling. Thereafter, the second true leaf thereof is cut out and then is installed into a cup, and about twenty (20) instar larvae of Western flower thrips (Frankliniella occidentalis) are released. After 6 days, the number of the surviving insects is examined, and the mortality is calculated by the following equation.

[00009] $Mortality (%) = (1 - the Number of the surviving insects / 20) ? 100$

Test Example 12-1

[2330] The test was conducted according to the Test method 12 by making the prescribed concentration 200 ppm and using the below-mentioned present compounds as a test compound, and, as the result of the test, the below-mentioned present compounds showed 90% or more as the mortality.

Present compound Nos: 11, 42, 88, 98

Test Method 13

[2331] An acetone solution which is adjusted to 2,000 ppm of the test compound is poured into a container having 20 mL contents, and the test compound is coated uniformly on inner face of the container such that the concentration of the test compound is made 100 mg/m.sup.2, and the container is then allowed to dry.

[2332] Five (5) larvae of Haemaphysalis longicornis are placed in the container, and the container is then covered with the lid. After the prescribed time has been passed, the state of the Haemaphysalis longicornis is examined, and the mortality is obtained. The mortality is calculated by the following equation.

[00010] $Mortality (%) = (the Number of dead insects / the Number of tested insects) ? 100$

Test Example 13-1

[2333] The test results obtained by the case when the test was conducted according to the Test Method 13 is shown below. The test was conducted by making the prescribed time two (2) days and by using the below-mentioned present compound as a test compound, and as the result of the test, the below-mentioned present compound showed 80% or more as the mortality.

Present compound Nos.: 12, 15, 23, 35, 47, 79, 83, 91, 94, 118, 138

Test Method 14

[2334] An acetone solution which is adjusted to 200 ppm of the test compound is poured into a container having 20 mL contents, and the test compound is coated uniformly on inner face of the container such that the concentration of the test compound is made 10 mg/m.sup.2, and the container is then allowed to dry.

[2335] Five (5) female adult of common house mosquito (Culex pipiens pallens) are placed in the container, and the container is then covered with the lid. After the prescribed time has been passed, the state of the common house mosquito is examined, and the mortality is obtained. The mortality is calculated by the following equation.

[00011] $Mortality (%) = (the Number of dead insects / the Number of tested insects) ? 100$

Test Example 14-1

[2336] The test results obtained by the case when the test was conducted according to the Test Method 14 is shown below. The test was conducted by making the prescribed time one (1) hour and by using the below-mentioned present compounds as a test compound, and as the result of the test, any of the below-mentioned present compounds showed 80% or more as the mortality.

Present compound No: 83

Test Example 14-2

[2337] The test results obtained by the case when the test was conducted according to the Test Method 14 is shown below. The test was conducted by making the prescribed time one (1) day and by using the below-mentioned present compounds as a test compound, and as the result of the test, any of the below-mentioned present compounds showed 80% or more as the mortality.

Present compound Nos: 12, 28, 49, 79, 83

Test Method 15

[2338] An acetone solution which is adjusted to 800 ppm of the test compound is poured into a container having 20 mL contents, and the test compound is coated uniformly on inner face of the container such that the concentration of the test compound is made 40 mg/m.sup.2, and the container is then allowed to dry.

[2339] Five (5) female adult housefly (Musca domestica) are placed in the container, and the container is then covered with the lid. After the prescribed time has been passed, the state of the housefly is examined, and the mortality is obtained. The mortality is calculated by the following equation.

[00012] $Mortality (%) = (the Number of dead insects / the Number of tested insects) ? 100$

Test Example 15-1

[2340] The test results obtained by the case when the test was conducted according to the Test Method 15 is shown below. The test was conducted by making the prescribed time one (1) day and by using the below-mentioned present compounds as a test compound, and as the result of the test, any of the below-mentioned present compounds showed 80% or more as the mortality.

Present compound Nos: 19, 28, 72, 78, 79, 143, 145

Test Method 16

[2341] An acetone solution which is adjusted to 800 ppm of the test compound is poured into a container having 50 mL contents, and the test compound is coated uniformly on inner face of the container such that the concentration of the test compound is made 40 mg/m.sup.2, and the container is then allowed to dry.

[2342] Five (5) male adult German cockroach (Blattella germanica) are placed in the container, and the container is then covered with the lid. After the prescribed time has been passed, the state of the housefly is examined, and the mortality is obtained. The mortality is calculated by the following equation.

[00013] $Mortality (%) = (the Number of dead insects / the Number of tested insects) ? 100$

Test Example 16-1

[2343] The test results obtained by the case when the test was conducted according to the Test Method 16 is shown below. The test was conducted by making the prescribed time three (3) days and by using the below-mentioned present compounds as a test compound, and as the result of the test, any of the below-mentioned present compounds showed 80% or more as the mortality.

Present compound No: 56

Test Method 17

[2344] Each 1 mg of the present compounds is dissolved into 10 ?L of a mixed solution of xylene, DMF, and a surfactant (xylene:DMF:surfactant=4:4:1 (v/v ratio)). Thereto is added water containing 0.02% by volume of a spreader to prepare diluted solution A containing a prescribed concentration of the present compound.

[2345] Each 1 mg of the present ingredients is dissolved into 10 ?L of a mixed solution of xylene, DMF, and a surfactant (xylene:DMF:surfactant=4:4:1 (v/v ratio)). Thereto is added water containing 0.02% by volume of a spreader to prepare diluted solution B containing a prescribed concentration of the present ingredient.

[2346] The diluted solution A is mixed with the diluted solution B to prepare diluted solution C.

[2347] Leaf discs of Cucumber (cucumber sativus) cotyledon (length 1.5 cm) are placed in each well of 24-well microplate. Two (2) apterous adults and 8 larvae of cotton aphids (Aphis gossypii) per one well are released and the diluted solution C is sprayed at 20 ?L per one well. The group is defined as treated group. A well that is sprayed with 20 ?L of water containing 0.02% by volume of a spreader instead of the diluted solution C is defined as untreated group.

[2348] After drying the diluted solution C, the upper microplate is covered with a film sheet. After 5 days, the number of the surviving insects in each well is examined.

[2349] The controlling value is calculated by the following equation.

Controlling value (%)={1?(Tai)/(Cai)}?100

wherein the symbols in the equation represent the following descriptions.

[2350] Cai: Number of the surviving insects at the time of the examination in untreated group;

[2351] Tai: Number of the surviving insects at the time of the examination in treated group.

[2352] Specific diluted solutions C, which can confirm their effect according to the Test method 17, are described in the following 1) to 5).

1) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 200 ppm and a concentration of the present ingredient is 2,000 ppm. In List A, Comp X represents any compound selected from the present compounds 1 to 136.

List A:

[2353] Comp X+Clothianidin; Comp X+thiamethoxam; Comp X+imidacloprid; Comp X+thiacloprid;
Comp X+flupyradifurone; Comp X+sulfoxaflor; Comp X+triflumezopyrim; Comp X+dicloromezotiaz; Comp X+beta-cyfluthrin; Comp X+tefluthrin; Comp X+fipronil; Comp X+chlorantraniliprole; Comp X+cyantraniliprole; Comp X+tetraniliprole; Comp X+thiodicarb; Comp X+carbofuran; Comp X+fluxametamide; Comp X+afoxolaner; Comp X+fluralaner; Comp X+broflanilide; Comp X+abamectin; Comp X+fluopyram; Comp X+fluensulfone; Comp X+fluazaindolizine; Comp X+tioxazafen; Comp X+flupyrimin; Comp X+Mycorrhizal Fungi; Comp X+Bradyrhizobium japonicum TA-11; Comp X+Bacillus firmus; Comp X+Bacillus firmus I-1582; Comp X+Bacillus amyloliquefaciens; Comp X+Bacillus amyloliquefaciens FZB42; Comp X+Pasteuria nishizawae; Comp X+Pasteuria nishizawae Pnl; Comp X+Pasteuria penetrans; Comp X+tebuconazole; Comp X+prothioconazole; Comp X+metconazole; Comp X+ipconazole; Comp X+triticonazole; Comp X+difenoconazole; Comp X+imazalil; Comp X+triadimenol; Comp X+tetraconazole; Comp X+flutriafol; Comp X+mandestrobin; Comp X+azoxystrobin; Comp X+pyraclostrobin; Comp X+trifloxystrobin; Comp X+fluoxastrobin; Comp X+picoxystrobin; Comp X+fenamidone; Comp X+metalaxyl; Comp X+metalaxyl-M; Comp X+fludioxonil; Comp X+sedaxane; Comp X+penflufen; Comp X+fluxapyroxad; Camp X+benzovindiflupyr; Camp X+boscalid; Comp X+carboxin; Comp X+penthiopyrad; Comp X+flutolanil; Comp X+captan; Comp X+thiram; Comp X+tolclofos-methyl; Camp X+thiabendazole; Camp X+ethaboxam; Comp X+mancozeb; Comp X+picarbutrazox; Comp X+oxathiapiprolin; Comp X+silthiofam; Comp X+inpyrfluxam.
2) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 200 ppm, and a concentration of the present ingredient is 200 ppm.
3) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 50 ppm.
4) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 5 ppm.
5) The diluted solution C comprises the combination recited in List A wherein a concentration of the present compound is 500 ppm, and a concentration of the present ingredient is 0.5 ppm.

INDUSTRIAL APPLICABILITY

[2354] The compound of the present invention has excellent control effect on harmful arthropods.

HETEROCYCLIC COMPOUND AND HARMFUL-ARTHROPOD-CONTROLLING COMPOSITION CONTAINING SAME

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