C07D209/54

Intermediate compounds and methods

The present invention relates to compounds of (II) and an acceptable salt or hydrate thereof method of making same. ##STR00001##

SSAO inhibitors and use thereof

The application relates to a compound of Formula (I′) or (I): ##STR00001##
or a pharmaceutically acceptable salt, hydrate, solvate, prodrug, stereoisomer, or tautomer thereof, which modulates the activity of SSAO, a pharmaceutical composition comprising a compound of Formula (I′) or (I), and a method of treating or preventing a disease in which SSAO plays a role.

INHIBITORS OF NOROVIRUS AND CORONAVIRUS REPLICATION
20230159453 · 2023-05-25 ·

Compounds of Formula (I) and methods of inhibiting the replication of viruses in a biological sample or patient, of reducing the amount of viruses in a biological sample or patient, and of treating a vims infection in a patient, comprising administering to said biological sample or patient an effective amount of a compound represented by Formula (I), a compound of Table A or B or a pharmaceutically acceptable salt thereof.

##STR00001##

INHIBITORS OF NOROVIRUS AND CORONAVIRUS REPLICATION
20230159453 · 2023-05-25 ·

Compounds of Formula (I) and methods of inhibiting the replication of viruses in a biological sample or patient, of reducing the amount of viruses in a biological sample or patient, and of treating a vims infection in a patient, comprising administering to said biological sample or patient an effective amount of a compound represented by Formula (I), a compound of Table A or B or a pharmaceutically acceptable salt thereof.

##STR00001##

Fluorinated Derivatives of Gabapentin and Methods of Use Thereof
20230150922 · 2023-05-18 ·

Described herein are fluorinated derivatives of gabapentin and methods of synthesis and methods of use thereof, e.g., in imaging and therapy.

Fluorinated Derivatives of Gabapentin and Methods of Use Thereof
20230150922 · 2023-05-18 ·

Described herein are fluorinated derivatives of gabapentin and methods of synthesis and methods of use thereof, e.g., in imaging and therapy.

Process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis-alkoxy-substituted spirocyclic 1H-pyrrolidine-2,4-dione derivatives

The present invention relates to a novel process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis-alkoxy-substituted spirocyclic 1H-pyrrolidine-2,4-dione derivatives, and also to novel intermediates and starting materials which are produced and/or used in the process according to the invention.

Process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis-alkoxy-substituted spirocyclic 1H-pyrrolidine-2,4-dione derivatives

The present invention relates to a novel process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis-alkoxy-substituted spirocyclic 1H-pyrrolidine-2,4-dione derivatives, and also to novel intermediates and starting materials which are produced and/or used in the process according to the invention.

INTERMEDIATE COMPOUNDS AND METHODS

The present invention relates to compounds of (II) and an acceptable salt or hydrate thereof method of making same.

##STR00001##

INTERMEDIATE COMPOUNDS AND METHODS

The present invention relates to compounds of (II) and an acceptable salt or hydrate thereof method of making same.

##STR00001##