C07D473/14

BRK inhibitory compound

The present invention relates to a Brk inhibitory compound represented by general formula (I) (wherein, all symbols represent the same meanings as the symbols set forth in the specification), a salt thereof, an N-oxide thereof, a solvate thereof, or a prodrug of any of these. ##STR00001##

METHOD OF ISOLATING THEACRINE AND COMPOSITION COMPRISING THEACRINE

Disclosed are improved methods for producing solid powdered theacrine compositions that are virtually flavorless and improved theacrine compositions.

METHOD OF ISOLATING THEACRINE AND COMPOSITION COMPRISING THEACRINE

Disclosed are improved methods for producing solid powdered theacrine compositions that are virtually flavorless and improved theacrine compositions.

NOVEL COCRYSTALS OF METHYLXANTHINES, THEIR POLYMORPHS AND PROCESS THEREOF

The present invention relates to cocrystals of Methylxanthines with Stilbenoids as coformers, their polymorphic forms and to the process for preparation thereof. The debittering of Methylxanthines is carried out by co-crystallization using Stilbenoids as coformers. The invention further relates to the preparation of polymorphic forms of debittered cocrystals and their use in nutraceutical and pharmaceutical compositions.

NOVEL COCRYSTALS OF METHYLXANTHINES, THEIR POLYMORPHS AND PROCESS THEREOF

The present invention relates to cocrystals of Methylxanthines with Stilbenoids as coformers, their polymorphic forms and to the process for preparation thereof. The debittering of Methylxanthines is carried out by co-crystallization using Stilbenoids as coformers. The invention further relates to the preparation of polymorphic forms of debittered cocrystals and their use in nutraceutical and pharmaceutical compositions.